Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 4615
Target3-phosphoinositide-dependent protein kinase 1(Human)
University of Munich

LigandPNGBDBM7401(6-bromoindirubin-3 -oxime | (3E)-6-bromo-3-[3-(hyd...)
Affinity DataIC50: 1.50E+3nMpH: 7.5 T: 2°CAssay Description:PDK1 protein kinase was expressed in Sf9 insect cells as human recombinant GST-fusion protein by means of the baculovirus expression systems. Protei...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2011
Entry Details Article
PubMed
Target3-phosphoinositide-dependent protein kinase 1(Human)
University of Munich

LigandPNGBDBM7393(Indirubin-3 -monoxime | 3-[(2Z,3E)-3-(hydroxyimino...)
Affinity DataIC50: 1.00E+5nMpH: 7.5 T: 2°CAssay Description:PDK1 protein kinase was expressed in Sf9 insect cells as human recombinant GST-fusion protein by means of the baculovirus expression systems. Protei...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2011
Entry Details Article
PubMed
Target3-phosphoinositide-dependent protein kinase 1(Human)
University of Munich

LigandPNGBDBM81296(5BIO)
Affinity DataIC50: 1.00E+5nMpH: 7.5 T: 2°CAssay Description:PDK1 protein kinase was expressed in Sf9 insect cells as human recombinant GST-fusion protein by means of the baculovirus expression systems. Protei...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2011
Entry Details Article
PubMed
Target3-phosphoinositide-dependent protein kinase 1(Human)
University of Munich

LigandPNGBDBM50218894(CHEMBL1092509 | 7BIO | 7-bromoindirubin-3-oxime)
Affinity DataIC50: 1.00E+5nMpH: 7.5 T: 2°CAssay Description:PDK1 protein kinase was expressed in Sf9 insect cells as human recombinant GST-fusion protein by means of the baculovirus expression systems. Protei...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2011
Entry Details Article
PubMed