Compile Data Set for Download or QSAR
Report error Found 20 Enz. Inhib. hit(s) with all data for entry = 50038273
TargetMuscarinic acetylcholine receptor M1(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50165008(2-[(1R)-3-(diisopropylamino)-1-phenylpropyl]-4-met...)
Affinity DataKi:  1.40nMAssay Description:Displacement of [3H]N-methyl Scopolamine from human cloned muscarinic M1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50165008(2-[(1R)-3-(diisopropylamino)-1-phenylpropyl]-4-met...)
Affinity DataKi:  2.20nMAssay Description:Displacement of [3H]N-methyl Scopolamine from human cloned muscarinic M5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50165008(2-[(1R)-3-(diisopropylamino)-1-phenylpropyl]-4-met...)
Affinity DataKi:  2.70nMAssay Description:Displacement of [3H]N-methyl Scopolamine from human cloned muscarinic M2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M4(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50165008(2-[(1R)-3-(diisopropylamino)-1-phenylpropyl]-4-met...)
Affinity DataKi:  3.10nMAssay Description:Displacement of [3H]N-methyl Scopolamine from human cloned muscarinic M4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50165008(2-[(1R)-3-(diisopropylamino)-1-phenylpropyl]-4-met...)
Affinity DataKi:  3.60nMAssay Description:Displacement of [3H]N-methyl Scopolamine from human cloned muscarinic M3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50374004(CHEMBL271108)
Affinity DataKi:  4.60nMAssay Description:Displacement of [3H]N-methyl Scopolamine from human cloned muscarinic M1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M4(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50374004(CHEMBL271108)
Affinity DataKi:  6.30nMAssay Description:Displacement of [3H]N-methyl Scopolamine from human cloned muscarinic M4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50374004(CHEMBL271108)
Affinity DataKi:  9nMAssay Description:Displacement of [3H]N-methyl Scopolamine from human cloned muscarinic M2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50374004(CHEMBL271108)
Affinity DataKi:  10.3nMAssay Description:Displacement of [3H]N-methyl Scopolamine from human cloned muscarinic M3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50374004(CHEMBL271108)
Affinity DataKi:  17.5nMAssay Description:Displacement of [3H]N-methyl Scopolamine from human cloned muscarinic M5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50374006(CHEMBL257643)
Affinity DataKi:  24nMAssay Description:Displacement of [3H]N-methyl Scopolamine from human cloned muscarinic M3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50374005(CHEMBL257431)
Affinity DataKi:  30nMAssay Description:Displacement of [3H]N-methyl Scopolamine from human cloned muscarinic M3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50374006(CHEMBL257643)
Affinity DataKi:  34nMAssay Description:Displacement of [3H]N-methyl Scopolamine from human cloned muscarinic M1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50374006(CHEMBL257643)
Affinity DataKi:  38nMAssay Description:Displacement of [3H]N-methyl Scopolamine from human cloned muscarinic M2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50374005(CHEMBL257431)
Affinity DataKi:  44nMAssay Description:Displacement of [3H]N-methyl Scopolamine from human cloned muscarinic M1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50374005(CHEMBL257431)
Affinity DataKi:  55nMAssay Description:Displacement of [3H]N-methyl Scopolamine from human cloned muscarinic M2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50374005(CHEMBL257431)
Affinity DataKi:  83nMAssay Description:Displacement of [3H]N-methyl Scopolamine from human cloned muscarinic M5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M4(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50374005(CHEMBL257431)
Affinity DataKi:  103nMAssay Description:Displacement of [3H]N-methyl Scopolamine from human cloned muscarinic M4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M4(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50374006(CHEMBL257643)
Affinity DataKi:  121nMAssay Description:Displacement of [3H]N-methyl Scopolamine from human cloned muscarinic M4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50374006(CHEMBL257643)
Affinity DataKi:  228nMAssay Description:Displacement of [3H]N-methyl Scopolamine from human cloned muscarinic M5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed