Compile Data Set for Download or QSAR
Report error Found 17 Enz. Inhib. hit(s) with all data for entry = 50022021
TargetTransketolase(Human)
Array Biopharma

Curated by ChEMBL
LigandPNGBDBM50230591(3-(acetylthio)-4-(N-((2-amino-6-methylpyridin-3-yl...)
Affinity DataEC50:  8nMAssay Description:Inhibition of transketolase in human HCT116 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetTransketolase(Human)
Array Biopharma

Curated by ChEMBL
LigandPNGBDBM50230590(N-(2-amino-6-chloro-pyridin-3-ylmethyl)-N-{2-[2-[(...)
Affinity DataEC50:  8nMAssay Description:Inhibition of transketolase in human HCT116 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetTransketolase(Human)
Array Biopharma

Curated by ChEMBL
LigandPNGBDBM50230593(CHEMBL270613 | CHEMBL401948 | 3-(2-amino-6-chloro-...)
Affinity DataEC50:  9nMAssay Description:Inhibition of transketolase in human HCT116 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetTransketolase(Human)
Array Biopharma

Curated by ChEMBL
LigandPNGBDBM50230587(N-(2-amino-6-methyl-pyridin-3-ylmethyl)-N-{2-[2-[(...)
Affinity DataEC50:  12nMAssay Description:Inhibition of transketolase in human HCT116 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetTransketolase(Human)
Array Biopharma

Curated by ChEMBL
LigandPNGBDBM50230598(N-((2-amino-6-methylpyridin-3-yl)methyl)-N-(5-hydr...)
Affinity DataEC50:  13nMAssay Description:Inhibition of transketolase in human HCT116 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetTransketolase(Human)
Array Biopharma

Curated by ChEMBL
LigandPNGBDBM50230586(N-((2-amino-6-methylpyridin-3-yl)methyl)-N-(1-(2-o...)
Affinity DataEC50:  15nMAssay Description:Inhibition of transketolase in human HCT116 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetTransketolase(Human)
Array Biopharma

Curated by ChEMBL
LigandPNGBDBM50230600(3-(6-methyl-2-amino-pyridin-3-ylmethyl)-5-(2-hydro...)
Affinity DataEC50:  18nMAssay Description:Inhibition of transketolase in human HCT116 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetTransketolase(Human)
Array Biopharma

Curated by ChEMBL
LigandPNGBDBM50230597(4-(N-((2-amino-6-methylpyridin-3-yl)methyl)formami...)
Affinity DataEC50:  28nMAssay Description:Inhibition of transketolase in human HCT116 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetTransketolase(Human)
Array Biopharma

Curated by ChEMBL
LigandPNGBDBM50230588(CHEMBL252441 | CHEMBL402329 | 3-(2-amino-6-methyl-...)
Affinity DataEC50:  28nMAssay Description:Inhibition of transketolase in human HCT116 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetTransketolase(Human)
Array Biopharma

Curated by ChEMBL
LigandPNGBDBM50230595(N-{2-[2-[acetyl-(2-amino-6-methyl-pyridin-3-ylmeth...)
Affinity DataEC50:  32nMAssay Description:Inhibition of transketolase in human HCT116 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetTransketolase(Human)
Array Biopharma

Curated by ChEMBL
LigandPNGBDBM50230599(3-(2-(4-(N-((2-amino-6-methylpyridin-3-yl)methyl)f...)
Affinity DataEC50:  52nMAssay Description:Inhibition of transketolase in human HCT116 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetTransketolase(Human)
Array Biopharma

Curated by ChEMBL
LigandPNGBDBM50230589(CHEMBL252637 | CHEMBL403365 | 3-(2-amino-pyridin-3...)
Affinity DataEC50:  110nMAssay Description:Inhibition of transketolase in human HCT116 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetTransketolase(Human)
Array Biopharma

Curated by ChEMBL
LigandPNGBDBM50230594((4-(N-((2-amino-6-methylpyridin-3-yl)methyl)formam...)
Affinity DataEC50:  116nMAssay Description:Inhibition of transketolase in human HCT116 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetTransketolase(Human)
Array Biopharma

Curated by ChEMBL
LigandPNGBDBM50230592(N-(2-amino-pyridin-3-ylmethyl)-N-{2-[2-[(2-amino-p...)
Affinity DataEC50:  479nMAssay Description:Inhibition of transketolase in human HCT116 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetTransketolase(Human)
Array Biopharma

Curated by ChEMBL
LigandPNGBDBM50230601(N-((2-amino-6-methylpyridin-3-yl)methyl)-N-(3-(but...)
Affinity DataEC50:  6.00E+3nMAssay Description:Inhibition of transketolase in human HCT116 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetTransketolase(Human)
Array Biopharma

Curated by ChEMBL
LigandPNGBDBM50230596(CHEMBL256454 | CHEMBL252842 | 3-(2-amino-6-methyl-...)
Affinity DataEC50:  9.54E+3nMAssay Description:Inhibition of transketolase in human HCT116 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetTransketolase(Human)
Array Biopharma

Curated by ChEMBL
LigandPNGBDBM50230602(N-(2-amino-6-methyl-pyridin-3-ylmethyl)-N-(2-{1-[1...)
Affinity DataEC50:  1.02E+5nMAssay Description:Inhibition of transketolase in human HCT116 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed