Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 4675
TargetProto-oncogene tyrosine-protein kinase Src(Mouse)
Ariad Pharmaceuticals

LigandPNGBDBM50318870(2,6,9-Trisubstituted Purine, AP23451 | 2,6,9-Trisu...)
Affinity DataIC50: 68nMAssay Description:2,6,9-Trisubstituted purines were evaluated for their src kinase inhibitory activities using an ELISA assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2011
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Mouse)
Ariad Pharmaceuticals

LigandPNGBDBM81725(2,6,9-Trisubstituted Purine, AP23517)
Affinity DataIC50: 73nMAssay Description:2,6,9-Trisubstituted purines were evaluated for their src kinase inhibitory activities using an ELISA assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2011
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Mouse)
Ariad Pharmaceuticals

LigandPNGBDBM81723(2,6,9-Trisubstituted Purine, 10)
Affinity DataIC50: 101nMAssay Description:2,6,9-Trisubstituted purines were evaluated for their src kinase inhibitory activities using an ELISA assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2011
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Mouse)
Ariad Pharmaceuticals

LigandPNGBDBM81722(2,6,9-Trisubstituted Purine, 9)
Affinity DataIC50: 205nMAssay Description:2,6,9-Trisubstituted purines were evaluated for their src kinase inhibitory activities using an ELISA assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2011
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Mouse)
Ariad Pharmaceuticals

LigandPNGBDBM50318870(2,6,9-Trisubstituted Purine, AP23451 | 2,6,9-Trisu...)
Affinity DataIC50: 273nMAssay Description:2,6,9-Trisubstituted purines were evaluated for their src kinase inhibitory activities using an ELISA assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2011
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Mouse)
Ariad Pharmaceuticals

LigandPNGBDBM81718(2,6,9-Trisubstituted Purine, 4)
Affinity DataIC50: 665nMAssay Description:2,6,9-Trisubstituted purines were evaluated for their src kinase inhibitory activities using an ELISA assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2011
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Mouse)
Ariad Pharmaceuticals

LigandPNGBDBM81720(2,6,9-Trisubstituted Purine, 6)
Affinity DataIC50: 1.01E+3nMAssay Description:2,6,9-Trisubstituted purines were evaluated for their src kinase inhibitory activities using an ELISA assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2011
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Mouse)
Ariad Pharmaceuticals

LigandPNGBDBM81724(2,6,9-Trisubstituted Purine, 11)
Affinity DataIC50: 2.11E+3nMAssay Description:2,6,9-Trisubstituted purines were evaluated for their src kinase inhibitory activities using an ELISA assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2011
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Mouse)
Ariad Pharmaceuticals

LigandPNGBDBM81721(2,6,9-Trisubstituted Purine, 7)
Affinity DataIC50: 2.30E+3nMAssay Description:2,6,9-Trisubstituted purines were evaluated for their src kinase inhibitory activities using an ELISA assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2011
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Mouse)
Ariad Pharmaceuticals

LigandPNGBDBM81719(2,6,9-Trisubstituted Purine, 5)
Affinity DataIC50: 2.31E+3nMAssay Description:2,6,9-Trisubstituted purines were evaluated for their src kinase inhibitory activities using an ELISA assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2011
Entry Details Article
PubMed