Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 2454
TargetHeat shock protein HSP 90-alpha(Human)
Wyeth Research

LigandPNGBDBM20732(geldanomycin | GM-BODIPY | Geldanamycin | CHEMBL27...)
Affinity DataIC50: 20nMpH: 7.3 T: 2°CAssay Description:Compounds were assayed over a threefold dilution series in a 96-well plate format to determine IC50 values. The reaction was allowed to proceed with ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2008
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
Wyeth Research

LigandPNGBDBM20739(CHEMBL404630 | 4-chloro-6-(5-{[2-(morpholin-4-yl)e...)
Affinity DataIC50: 30nMpH: 7.3 T: 2°CAssay Description:Compounds were assayed over a threefold dilution series in a 96-well plate format to determine IC50 values. The reaction was allowed to proceed with ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2008
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
Wyeth Research

LigandPNGBDBM20737(4-bromo-6-(5-{[2-(morpholin-4-yl)ethyl]amino}-1,2-...)
Affinity DataIC50: 40nMpH: 7.3 T: 2°CAssay Description:Compounds were assayed over a threefold dilution series in a 96-well plate format to determine IC50 values. The reaction was allowed to proceed with ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2008
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
Wyeth Research

LigandPNGBDBM20734(CHEMBL362307 | 4-chloro-6-(6-hydroxy-1,2-benzoxazo...)
Affinity DataIC50: 60nMpH: 7.3 T: 2°CAssay Description:Compounds were assayed over a threefold dilution series in a 96-well plate format to determine IC50 values. The reaction was allowed to proceed with ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2008
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
Wyeth Research

LigandPNGBDBM20731(4-bromo-6-(6-hydroxy-1,2-benzoxazol-3-yl)benzene-1...)
Affinity DataIC50: 190nMpH: 7.3 T: 2°CAssay Description:Compounds were assayed over a threefold dilution series in a 96-well plate format to determine IC50 values. The reaction was allowed to proceed with ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2008
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
Wyeth Research

LigandPNGBDBM20736(4-chloro-6-[5-(4-methylpiperazin-1-yl)-1,2-benzoxa...)
Affinity DataIC50: 800nMpH: 7.3 T: 2°CAssay Description:Compounds were assayed over a threefold dilution series in a 96-well plate format to determine IC50 values. The reaction was allowed to proceed with ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2008
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
Wyeth Research

LigandPNGBDBM20733(CHEMBL360410 | 4-(6-hydroxy-1,2-benzoxazol-3-yl)be...)
Affinity DataIC50: 1.52E+4nMpH: 7.3 T: 2°CAssay Description:Compounds were assayed over a threefold dilution series in a 96-well plate format to determine IC50 values. The reaction was allowed to proceed with ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2008
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
Wyeth Research

LigandPNGBDBM20735(3-(5-chloro-2,4-dimethoxyphenyl)-6-methoxy-1,2-ben...)
Affinity DataIC50: 2.00E+4nMpH: 7.3 T: 2°CAssay Description:Compounds were assayed over a threefold dilution series in a 96-well plate format to determine IC50 values. The reaction was allowed to proceed with ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2008
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
Wyeth Research

LigandPNGBDBM20738(3-(5-chloro-2,4-dimethoxyphenyl)-N-[2-(morpholin-4...)
Affinity DataIC50: 2.00E+4nMpH: 7.3 T: 2°CAssay Description:Compounds were assayed over a threefold dilution series in a 96-well plate format to determine IC50 values. The reaction was allowed to proceed with ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2008
Entry Details Article
PubMed