Compile Data Set for Download or QSAR
Report error Found 80 Enz. Inhib. hit(s) with all data for entry = 515
TargetProtein kinase C eta type(Human)
Sphinx Pharmaceuticals

LigandPNGBDBM3153(CHEMBL52529 | 2-{[2,6-dihydroxy-4-({[(1R,2R)-2-[(4...)
Affinity DataIC50: 0.600nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2005
Entry Details Article

TargetProtein kinase C delta type(Human)
Sphinx Pharmaceuticals

LigandPNGBDBM3153(CHEMBL52529 | 2-{[2,6-dihydroxy-4-({[(1R,2R)-2-[(4...)
Affinity DataIC50: 0.900nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2005
Entry Details Article

TargetProtein kinase C eta type(Human)
Sphinx Pharmaceuticals

LigandPNGBDBM3252((1R,2R)-2-[(4-hydroxybenzene)amido]cyclopentyl 3,5...)
Affinity DataIC50: 4nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2005
Entry Details Article

TargetProtein kinase C eta type(Human)
Sphinx Pharmaceuticals

LigandPNGBDBM3248((3R,4R)-4-[(4-hydroxybenzene)amido]pyrrolidin-3-yl...)
Affinity DataIC50: 4nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2005
Entry Details Article

TargetProtein kinase C eta type(Human)
Sphinx Pharmaceuticals

LigandPNGBDBM3152(2-{[2,6-dihydroxy-4-({[(3R,4R)-4-[(4-hydroxybenzen...)
Affinity DataIC50: 4nMpH: 7.5 T: 2°CAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2005
Entry Details Article

TargetProtein kinase C delta type(Human)
Sphinx Pharmaceuticals

LigandPNGBDBM3252((1R,2R)-2-[(4-hydroxybenzene)amido]cyclopentyl 3,5...)
Affinity DataIC50: 5nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2005
Entry Details Article

TargetProtein kinase C delta type(Human)
Sphinx Pharmaceuticals

LigandPNGBDBM3152(2-{[2,6-dihydroxy-4-({[(3R,4R)-4-[(4-hydroxybenzen...)
Affinity DataIC50: 5nMpH: 7.5 T: 2°CAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2005
Entry Details Article

TargetProtein kinase C epsilon type(Human)
Sphinx Pharmaceuticals

LigandPNGBDBM3152(2-{[2,6-dihydroxy-4-({[(3R,4R)-4-[(4-hydroxybenzen...)
Affinity DataIC50: 10nMpH: 7.5 T: 2°CAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2005
Entry Details Article

TargetProtein kinase C delta type(Human)
Sphinx Pharmaceuticals

LigandPNGBDBM3248((3R,4R)-4-[(4-hydroxybenzene)amido]pyrrolidin-3-yl...)
Affinity DataIC50: 10nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2005
Entry Details Article

TargetProtein kinase C eta type(Human)
Sphinx Pharmaceuticals

LigandPNGBDBM3249((3R,4R)-4-[(4-hydroxybenzene)amido]pyrrolidin-3-yl...)
Affinity DataIC50: 14nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2005
Entry Details Article

TargetProtein kinase C eta type(Human)
Sphinx Pharmaceuticals

LigandPNGBDBM3243((3R,4R)-4-[(4-hydroxybenzene)amido]pyrrolidin-3-yl...)
Affinity DataIC50: 16nMpH: 7.5 T: 2°CAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2005
Entry Details Article

TargetProtein kinase C delta type(Human)
Sphinx Pharmaceuticals

LigandPNGBDBM3243((3R,4R)-4-[(4-hydroxybenzene)amido]pyrrolidin-3-yl...)
Affinity DataIC50: 18nMpH: 7.5 T: 2°CAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2005
Entry Details Article

TargetProtein kinase C beta type(Human)
Sphinx Pharmaceuticals

LigandPNGBDBM3248((3R,4R)-4-[(4-hydroxybenzene)amido]pyrrolidin-3-yl...)
Affinity DataIC50: 20nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2005
Entry Details Article

TargetProtein kinase C eta type(Human)
Sphinx Pharmaceuticals

LigandPNGBDBM3244((3R,4R)-4-[(4-hydroxybenzene)amido]pyrrolidin-3-yl...)
Affinity DataIC50: 20nMpH: 7.5 T: 2°CAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2005
Entry Details Article

TargetProtein kinase C beta type(Human)
Sphinx Pharmaceuticals

LigandPNGBDBM3249((3R,4R)-4-[(4-hydroxybenzene)amido]pyrrolidin-3-yl...)
Affinity DataIC50: 20nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2005
Entry Details Article

TargetProtein kinase C eta type(Human)
Sphinx Pharmaceuticals

LigandPNGBDBM3149(Acyclic Balanol Analog (-)-1 | 2-{[2,6-dihydroxy-4...)
Affinity DataIC50: 22nMpH: 7.5 T: 2°CAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2005
Entry Details Article

TargetProtein kinase C alpha type(Human)
Sphinx Pharmaceuticals

LigandPNGBDBM3152(2-{[2,6-dihydroxy-4-({[(3R,4R)-4-[(4-hydroxybenzen...)
Affinity DataIC50: 22nMpH: 7.5 T: 2°CAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2005
Entry Details Article

TargetProtein kinase C delta type(Human)
Sphinx Pharmaceuticals

LigandPNGBDBM3249((3R,4R)-4-[(4-hydroxybenzene)amido]pyrrolidin-3-yl...)
Affinity DataIC50: 24nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2005
Entry Details Article

TargetProtein kinase C delta type(Human)
Sphinx Pharmaceuticals

LigandPNGBDBM3250(2-[(4-hydroxybenzene)amido]cyclopentyl 3,5-dihydro...)
Affinity DataIC50: 30nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2005
Entry Details Article

TargetProtein kinase C eta type(Human)
Sphinx Pharmaceuticals

LigandPNGBDBM3250(2-[(4-hydroxybenzene)amido]cyclopentyl 3,5-dihydro...)
Affinity DataIC50: 30nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2005
Entry Details Article

TargetProtein kinase C delta type(Human)
Sphinx Pharmaceuticals

LigandPNGBDBM50285231(3,5-Dihydroxy-4-(2-hydroxy-6-methoxycarbonyl-benzo...)
Affinity DataIC50: 30nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2005
Entry Details Article

TargetProtein kinase C delta type(Human)
Sphinx Pharmaceuticals

LigandPNGBDBM3149(Acyclic Balanol Analog (-)-1 | 2-{[2,6-dihydroxy-4...)
Affinity DataIC50: 32nMpH: 7.5 T: 2°CAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2005
Entry Details Article

TargetProtein kinase C beta type(Human)
Sphinx Pharmaceuticals

LigandPNGBDBM3152(2-{[2,6-dihydroxy-4-({[(3R,4R)-4-[(4-hydroxybenzen...)
Affinity DataIC50: 33nMpH: 7.5 T: 2°CAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2005
Entry Details Article

TargetProtein kinase C epsilon type(Human)
Sphinx Pharmaceuticals

LigandPNGBDBM3248((3R,4R)-4-[(4-hydroxybenzene)amido]pyrrolidin-3-yl...)
Affinity DataIC50: 34nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2005
Entry Details Article

TargetProtein kinase C beta type(Human)
Sphinx Pharmaceuticals

LigandPNGBDBM3252((1R,2R)-2-[(4-hydroxybenzene)amido]cyclopentyl 3,5...)
Affinity DataIC50: 40nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2005
Entry Details Article

TargetProtein kinase C beta type(Human)
Sphinx Pharmaceuticals

LigandPNGBDBM50285231(3,5-Dihydroxy-4-(2-hydroxy-6-methoxycarbonyl-benzo...)
Affinity DataIC50: 40nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2005
Entry Details Article

TargetProtein kinase C alpha type(Human)
Sphinx Pharmaceuticals

LigandPNGBDBM3153(CHEMBL52529 | 2-{[2,6-dihydroxy-4-({[(1R,2R)-2-[(4...)
Affinity DataIC50: 40nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2005
Entry Details Article

TargetProtein kinase C eta type(Human)
Sphinx Pharmaceuticals

LigandPNGBDBM3245((3R,4R)-4-[(4-hydroxybenzene)amido]pyrrolidin-3-yl...)
Affinity DataIC50: 40nMpH: 7.5 T: 2°CAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2005
Entry Details Article

TargetProtein kinase C beta type(Human)
Sphinx Pharmaceuticals

LigandPNGBDBM3149(Acyclic Balanol Analog (-)-1 | 2-{[2,6-dihydroxy-4...)
Affinity DataIC50: 44nMpH: 7.5 T: 2°CAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2005
Entry Details Article

TargetProtein kinase C epsilon type(Human)
Sphinx Pharmaceuticals

LigandPNGBDBM3149(Acyclic Balanol Analog (-)-1 | 2-{[2,6-dihydroxy-4...)
Affinity DataIC50: 49nMpH: 7.5 T: 2°CAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2005
Entry Details Article

TargetProtein kinase C delta type(Human)
Sphinx Pharmaceuticals

LigandPNGBDBM3254((1R,2R)-2-[(4-hydroxybenzene)amido]cyclopentyl 3,5...)
Affinity DataIC50: 50nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2005
Entry Details Article

TargetProtein kinase C beta type(Human)
Sphinx Pharmaceuticals

LigandPNGBDBM3153(CHEMBL52529 | 2-{[2,6-dihydroxy-4-({[(1R,2R)-2-[(4...)
Affinity DataIC50: 50nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2005
Entry Details Article

TargetProtein kinase C delta type(Human)
Sphinx Pharmaceuticals

LigandPNGBDBM3244((3R,4R)-4-[(4-hydroxybenzene)amido]pyrrolidin-3-yl...)
Affinity DataIC50: 50nMpH: 7.5 T: 2°CAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2005
Entry Details Article

TargetProtein kinase C eta type(Human)
Sphinx Pharmaceuticals

LigandPNGBDBM3247((3R,4R)-4-[(4-hydroxybenzene)amido]pyrrolidin-3-yl...)
Affinity DataIC50: 50nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2005
Entry Details Article

TargetProtein kinase C eta type(Human)
Sphinx Pharmaceuticals

LigandPNGBDBM3246((3R,4R)-4-[(4-hydroxybenzene)amido]pyrrolidin-3-yl...)
Affinity DataIC50: 50nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2005
Entry Details Article

TargetProtein kinase C epsilon type(Human)
Sphinx Pharmaceuticals

LigandPNGBDBM3153(CHEMBL52529 | 2-{[2,6-dihydroxy-4-({[(1R,2R)-2-[(4...)
Affinity DataIC50: 50nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2005
Entry Details Article

TargetProtein kinase C eta type(Human)
Sphinx Pharmaceuticals

LigandPNGBDBM3253((1R,2R)-2-[(4-hydroxybenzene)amido]cyclopentyl 4-{...)
Affinity DataIC50: 52nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2005
Entry Details Article

TargetProtein kinase C delta type(Human)
Sphinx Pharmaceuticals

LigandPNGBDBM3253((1R,2R)-2-[(4-hydroxybenzene)amido]cyclopentyl 4-{...)
Affinity DataIC50: 67nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2005
Entry Details Article

TargetProtein kinase C alpha type(Human)
Sphinx Pharmaceuticals

LigandPNGBDBM3149(Acyclic Balanol Analog (-)-1 | 2-{[2,6-dihydroxy-4...)
Affinity DataIC50: 74nMpH: 7.5 T: 2°CAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2005
Entry Details Article

TargetProtein kinase C delta type(Human)
Sphinx Pharmaceuticals

LigandPNGBDBM3245((3R,4R)-4-[(4-hydroxybenzene)amido]pyrrolidin-3-yl...)
Affinity DataIC50: 80nMpH: 7.5 T: 2°CAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2005
Entry Details Article

TargetProtein kinase C alpha type(Human)
Sphinx Pharmaceuticals

LigandPNGBDBM3249((3R,4R)-4-[(4-hydroxybenzene)amido]pyrrolidin-3-yl...)
Affinity DataIC50: 130nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2005
Entry Details Article

TargetProtein kinase C epsilon type(Human)
Sphinx Pharmaceuticals

LigandPNGBDBM3249((3R,4R)-4-[(4-hydroxybenzene)amido]pyrrolidin-3-yl...)
Affinity DataIC50: 130nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2005
Entry Details Article

TargetProtein kinase C alpha type(Human)
Sphinx Pharmaceuticals

LigandPNGBDBM3248((3R,4R)-4-[(4-hydroxybenzene)amido]pyrrolidin-3-yl...)
Affinity DataIC50: 160nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2005
Entry Details Article

TargetProtein kinase C epsilon type(Human)
Sphinx Pharmaceuticals

LigandPNGBDBM3243((3R,4R)-4-[(4-hydroxybenzene)amido]pyrrolidin-3-yl...)
Affinity DataIC50: 170nMpH: 7.5 T: 2°CAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2005
Entry Details Article

TargetProtein kinase C delta type(Human)
Sphinx Pharmaceuticals

LigandPNGBDBM3246((3R,4R)-4-[(4-hydroxybenzene)amido]pyrrolidin-3-yl...)
Affinity DataIC50: 200nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2005
Entry Details Article

TargetProtein kinase C alpha type(Human)
Sphinx Pharmaceuticals

LigandPNGBDBM3252((1R,2R)-2-[(4-hydroxybenzene)amido]cyclopentyl 3,5...)
Affinity DataIC50: 210nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2005
Entry Details Article

TargetProtein kinase C delta type(Human)
Sphinx Pharmaceuticals

LigandPNGBDBM3251((1S,2S)-2-[(4-hydroxybenzene)amido]cyclopentyl 3,5...)
Affinity DataIC50: 250nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2005
Entry Details Article

TargetProtein kinase C alpha type(Human)
Sphinx Pharmaceuticals

LigandPNGBDBM3243((3R,4R)-4-[(4-hydroxybenzene)amido]pyrrolidin-3-yl...)
Affinity DataIC50: 250nMpH: 7.5 T: 2°CAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2005
Entry Details Article

TargetProtein kinase C epsilon type(Human)
Sphinx Pharmaceuticals

LigandPNGBDBM3250(2-[(4-hydroxybenzene)amido]cyclopentyl 3,5-dihydro...)
Affinity DataIC50: 260nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2005
Entry Details Article

TargetProtein kinase C eta type(Human)
Sphinx Pharmaceuticals

LigandPNGBDBM3254((1R,2R)-2-[(4-hydroxybenzene)amido]cyclopentyl 3,5...)
Affinity DataIC50: 260nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2005
Entry Details Article

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