Compile Data Set for Download or QSAR
Report error Found 82 Enz. Inhib. hit(s) with all data for entry = 50022295
TargetC-X-C chemokine receptor type 2(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233576((R)-3-(2-(1-(4-bromofuran-2-yl)propylamino)-3,4-di...)
Affinity DataIC50: 2nMAssay Description:Inhibition of CXCR2-mediated chemotaxis in Ba/F3 cells expressing human CXCR2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233586(2-hydroxy-3-(2-(1-(5-(hydroxymethyl)furan-2-yl)pro...)
Affinity DataIC50: 2.80nMAssay Description:Inhibition of CXCR2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233554((R)-3-(3,4-dioxo-2-(1-(pyridin-2-yl)propylamino)cy...)
Affinity DataIC50: 3.30nMAssay Description:Inhibition of CXCR2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233561((R)-3-(3,4-dioxo-2-(1-(thiophen-3-yl)propylamino)c...)
Affinity DataIC50: 3.40nMAssay Description:Inhibition of CXCR2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233560(3-(2-(1-(benzofuran-2-yl)propylamino)-3,4-dioxocyc...)
Affinity DataIC50: 3.5nMAssay Description:Inhibition of CXCR2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233576((R)-3-(2-(1-(4-bromofuran-2-yl)propylamino)-3,4-di...)
Affinity DataIC50: 3.5nMAssay Description:Inhibition of CXCR2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233574((R)-3-(2-(1-(4-chlorofuran-2-yl)propylamino)-3,4-d...)
Affinity DataIC50: 3.80nMAssay Description:Inhibition of CXCR2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233592(3-(2-(1-(5-ethylfuran-2-yl)propylamino)-3,4-dioxoc...)
Affinity DataIC50: 4.10nMAssay Description:Inhibition of CXCR2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233554((R)-3-(3,4-dioxo-2-(1-(pyridin-2-yl)propylamino)cy...)
Affinity DataIC50: 4.5nMAssay Description:Inhibition of CXCR2-mediated chemotaxis in Ba/F3 cells expressing human CXCR2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233589(3-(2-(1-(4-chlorofuran-2-yl)propylamino)-3,4-dioxo...)
Affinity DataIC50: 4.5nMAssay Description:Inhibition of CXCR2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233572((R)-3-(2-(1-(5-chlorofuran-2-yl)propylamino)-3,4-d...)
Affinity DataIC50: 4.60nMAssay Description:Inhibition of CXCR2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233588(3-(2-(1-(5-bromofuran-2-yl)propylamino)-3,4-dioxoc...)
Affinity DataIC50: 4.70nMAssay Description:Inhibition of CXCR2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233581(3-(2-(1-(5-chlorofuran-2-yl)propylamino)-3,4-dioxo...)
Affinity DataIC50: 4.80nMAssay Description:Inhibition of CXCR2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233563(3-(2-(1-(furan-2-yl)propylamino)-3,4-dioxocyclobut...)
Affinity DataIC50: 5nMAssay Description:Inhibition of CXCR2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233577(3-(2-(1-(4-bromofuran-2-yl)propylamino)-3,4-dioxoc...)
Affinity DataIC50: 5nMAssay Description:Inhibition of CXCR2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233553(2-hydroxy-N,N-dimethyl-3-(2-(1-(5-methylfuran-2-yl...)
Affinity DataIC50: 5.70nMAssay Description:Inhibition of CXCR2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233584(3-(3,4-dioxo-2-(1-(thiophen-3-yl)propylamino)cyclo...)
Affinity DataIC50: 5.80nMAssay Description:Inhibition of CXCR2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233570(3-(3,4-dioxo-2-(1-(4-phenylfuran-2-yl)propylamino)...)
Affinity DataIC50: 6.10nMAssay Description:Inhibition of CXCR2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233580(3-(3,4-dioxo-2-(1-(thiophen-2-yl)propylamino)cyclo...)
Affinity DataIC50: 6.20nMAssay Description:Inhibition of CXCR2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233557(3-(2-(1-(5-chlorothiophen-2-yl)propylamino)-3,4-di...)
Affinity DataIC50: 6.20nMAssay Description:Inhibition of CXCR2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233558((R)-2-hydroxy-N,N-dimethyl-3-(2-(1-(5-methylisoxaz...)
Affinity DataIC50: 6.30nMAssay Description:Inhibition of CXCR2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233568(3-(2-(1-(5-(difluoromethyl)furan-2-yl)propylamino)...)
Affinity DataIC50: 6.80nMAssay Description:Inhibition of CXCR2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233567(2-hydroxy-N,N-dimethyl-3-(2-(1-(5-methylisoxazol-3...)
Affinity DataIC50: 7.5nMAssay Description:Inhibition of CXCR2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233590(3-(2-(1-(4-(3,5-dimethylisoxazol-4-yl)furan-2-yl)p...)
Affinity DataIC50: 7.60nMAssay Description:Inhibition of CXCR2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233552(3-(2-(1-(furan-3-yl)propylamino)-3,4-dioxocyclobut...)
Affinity DataIC50: 8nMAssay Description:Inhibition of CXCR2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233556(2-hydroxy-N,N-dimethyl-3-(2-(1-(3-methyl-1,2,4-oxa...)
Affinity DataIC50: 8.20nMAssay Description:Inhibition of CXCR2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233562(3-(3,4-dioxo-2-(1-(4-(thiophen-3-yl)furan-2-yl)pro...)
Affinity DataIC50: 8.20nMAssay Description:Inhibition of CXCR2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233565(2-hydroxy-N,N-dimethyl-3-(2-(1-(oxazol-2-yl)propyl...)
Affinity DataIC50: 8.60nMAssay Description:Inhibition of CXCR2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233587(3-(3,4-dioxo-2-(1-(4-(pyridin-4-yl)furan-2-yl)prop...)
Affinity DataIC50: 9.5nMAssay Description:Inhibition of CXCR2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233583(3-(3,4-dioxo-2-(1-(thiazol-2-yl)propylamino)cyclob...)
Affinity DataIC50: 9.80nMAssay Description:Inhibition of CXCR2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233578(2-hydroxy-3-(2-(1-(isoxazol-5-yl)propylamino)-3,4-...)
Affinity DataIC50: 9.80nMAssay Description:Inhibition of CXCR2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233569(2-hydroxy-N,N-dimethyl-3-(2-(1-(oxazol-4-yl)propyl...)
Affinity DataIC50: 10.9nMAssay Description:Inhibition of CXCR2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233558((R)-2-hydroxy-N,N-dimethyl-3-(2-(1-(5-methylisoxaz...)
Affinity DataIC50: 12.2nMAssay Description:Inhibition of CXCR2-mediated chemotaxis in Ba/F3 cells expressing human CXCR2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233579(3-(2-(1-(3-bromofuran-2-yl)propylamino)-3,4-dioxoc...)
Affinity DataIC50: 16.5nMAssay Description:Inhibition of CXCR2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233566(3-(3,4-dioxo-2-(1-(5-(trifluoromethyl)furan-2-yl)p...)
Affinity DataIC50: 17.2nMAssay Description:Inhibition of CXCR2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233564(3-(2-(1-(3-chlorothiophen-2-yl)propylamino)-3,4-di...)
Affinity DataIC50: 21nMAssay Description:Inhibition of CXCR2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233591(3-(2-(1-(5-(2-chlorophenyl)furan-2-yl)propylamino)...)
Affinity DataIC50: 49nMAssay Description:Inhibition of CXCR2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233555(3-(3,4-dioxo-2-(1-(pyridin-4-yl)propylamino)cyclob...)
Affinity DataIC50: 50nMAssay Description:Inhibition of CXCR2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233576((R)-3-(2-(1-(4-bromofuran-2-yl)propylamino)-3,4-di...)
Affinity DataIC50: 55nMAssay Description:Inhibition of CXCR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233573(3-(2-(1-(5-(3-chlorophenyl)furan-2-yl)propylamino)...)
Affinity DataIC50: 58nMAssay Description:Inhibition of CXCR2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233574((R)-3-(2-(1-(4-chlorofuran-2-yl)propylamino)-3,4-d...)
Affinity DataIC50: 62nMAssay Description:Inhibition of CXCR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233563(3-(2-(1-(furan-2-yl)propylamino)-3,4-dioxocyclobut...)
Affinity DataIC50: 67nMAssay Description:Inhibition of CXCR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233582(3-(3,4-dioxo-2-(1-(5-(3-(trifluoromethyl)phenyl)fu...)
Affinity DataIC50: 87nMAssay Description:Inhibition of CXCR2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233577(3-(2-(1-(4-bromofuran-2-yl)propylamino)-3,4-dioxoc...)
Affinity DataIC50: 93nMAssay Description:Inhibition of CXCR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233559(3-(2-(1-(5-((dimethylamino)methyl)furan-2-yl)propy...)
Affinity DataIC50: 94nMAssay Description:Inhibition of CXCR2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233553(2-hydroxy-N,N-dimethyl-3-(2-(1-(5-methylfuran-2-yl...)
Affinity DataIC50: 99nMAssay Description:Inhibition of CXCR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233589(3-(2-(1-(4-chlorofuran-2-yl)propylamino)-3,4-dioxo...)
Affinity DataIC50: 100nMAssay Description:Inhibition of CXCR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233561((R)-3-(3,4-dioxo-2-(1-(thiophen-3-yl)propylamino)c...)
Affinity DataIC50: 104nMAssay Description:Inhibition of CXCR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233554((R)-3-(3,4-dioxo-2-(1-(pyridin-2-yl)propylamino)cy...)
Affinity DataIC50: 148nMAssay Description:Inhibition of CXCR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50233570(3-(3,4-dioxo-2-(1-(4-phenylfuran-2-yl)propylamino)...)
Affinity DataIC50: 150nMAssay Description:Inhibition of CXCR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
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