Compile Data Set for Download or QSAR
Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 50035907
TargetD(2) dopamine receptor(Rat)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50452985(CHEMBL2114234)
Affinity DataKi:  6.70nMAssay Description:Binding affinity towards dopamine receptor D2 using as [3H]-spiperone radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50452983(CHEMBL2114236)
Affinity DataKi:  9.40nMAssay Description:Binding affinity towards dopamine receptor D2 using as [3H]-spiperone radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50452981(CHEMBL2115231)
Affinity DataKi:  9.60nMAssay Description:Binding affinity towards dopamine receptor D2 using as [3H]-spiperone radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50452980(CHEMBL2115232)
Affinity DataKi:  21nMAssay Description:Binding affinity towards dopamine receptor D2 using as [3H]-spiperone radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50452984(CHEMBL2114235)
Affinity DataKi:  23nMAssay Description:Binding affinity towards dopamine receptor D2 using as [3H]-spiperone radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM81774(Sulpiride-S | CAS_15676-16-1 | Sulpiride-l | SULPI...)
Affinity DataKi:  29nMAssay Description:Binding affinity towards dopamine receptor D2 using as [3H]-spiperone radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50284586(N-((S)-1-Butyl-pyrrolidin-2-ylmethyl)-2-methoxy-5-...)
Affinity DataKi:  51nMAssay Description:Binding affinity towards dopamine receptor D2 using as [3H]-spiperone radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50452990(CHEMBL2114240)
Affinity DataKi:  59nMAssay Description:Binding affinity towards dopamine receptor D2 using as [3H]-spiperone radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50452982(CHEMBL2115229)
Affinity DataKi:  95nMAssay Description:Binding affinity towards dopamine receptor D2 using as [3H]-spiperone radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50452987(CHEMBL2115228)
Affinity DataKi:  210nMAssay Description:Binding affinity towards dopamine receptor D2 using as [3H]-spiperone radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50284609(N-((R)-1-Butyl-pyrrolidin-2-ylmethyl)-2-methoxy-5-...)
Affinity DataKi:  230nMAssay Description:Binding affinity towards dopamine receptor D2 using as [3H]-spiperone radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50452988(CHEMBL2114238)
Affinity DataKi:  400nMAssay Description:Binding affinity towards dopamine receptor D2 using as [3H]-spiperone radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50452986(CHEMBL2115227)
Affinity DataKi:  630nMAssay Description:Binding affinity towards dopamine receptor D2 using as [3H]-spiperone radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50452989(CHEMBL2114239)
Affinity DataKi:  650nMAssay Description:Binding affinity towards dopamine receptor D2 using as [3H]-spiperone radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50452979(CHEMBL2115233)
Affinity DataKi:  1.40E+3nMAssay Description:Binding affinity towards dopamine receptor D2 using as [3H]-spiperone radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM81775(Sulpiride-R | Sulpiride-d | Sulpiride-low,(-) | Su...)
Affinity DataKi:  2.70E+3nMAssay Description:Binding affinity towards dopamine receptor D2 using as [3H]-spiperone radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed