Compile Data Set for Download or QSAR
Report error Found 33 Enz. Inhib. hit(s) with all data for entry = 50041538
TargetC-C chemokine receptor type 8(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50423492(CHEMBL409648)
Affinity DataIC50: 12nMAssay Description:Antagonist activity at CCR8 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50414964(CHEMBL271128)
Affinity DataIC50: 12nMAssay Description:Antagonist activity at CCR8 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50411749(CHEMBL271127)
Affinity DataIC50: 16nMAssay Description:Antagonist activity at CCR8 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50414967(CHEMBL271801)
Affinity DataIC50: 18nMAssay Description:Antagonist activity at CCR8 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50414957(CHEMBL429436)
Affinity DataIC50: 19nMAssay Description:Antagonist activity at CCR8 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50423493(CHEMBL411651)
Affinity DataIC50: 27nMAssay Description:Antagonist activity at CCR8 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50414968(CHEMBL410885)
Affinity DataIC50: 28nMAssay Description:Antagonist activity at CCR8 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50414969(CHEMBL272022)
Affinity DataIC50: 33nMAssay Description:Antagonist activity at CCR8 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50423496(CHEMBL271768)
Affinity DataIC50: 33nMAssay Description:Antagonist activity at CCR8 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50414959(CHEMBL409224)
Affinity DataIC50: 35nMAssay Description:Antagonist activity at CCR8 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50423495(CHEMBL270969)
Affinity DataIC50: 79nMAssay Description:Antagonist activity at CCR8 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50414958(CHEMBL259243)
Affinity DataIC50: 81nMAssay Description:Antagonist activity at CCR8 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50414965(CHEMBL270971)
Affinity DataIC50: 115nMAssay Description:Antagonist activity at CCR8 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
LigandPNGBDBM50411749(CHEMBL271127)
Affinity DataIC50: 120nMAssay Description:Displacement of [3H]dofetilide from human recombinant ERG potassium channel expressed in HEK293 cells by patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50423494(CHEMBL409849)
Affinity DataIC50: 166nMAssay Description:Antagonist activity at CCR8 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
LigandPNGBDBM50411754(CHEMBL410862)
Affinity DataIC50: 5.13E+8nMAssay Description:Displacement of [3H]dofetilide from human recombinant ERG potassium channel expressed in HEK293 cells by patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
LigandPNGBDBM50411756(CHEMBL272241)
Affinity DataIC50: 2.95E+6nMAssay Description:Displacement of [3H]dofetilide from human recombinant ERG potassium channel expressed in HEK293 cells by patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
LigandPNGBDBM50411755(CHEMBL408483)
Affinity DataIC50: 9.55E+8nMAssay Description:Displacement of [3H]dofetilide from human recombinant ERG potassium channel expressed in HEK293 cells by patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
LigandPNGBDBM50411738(CHEMBL272842)
Affinity DataIC50: 7.59E+8nMAssay Description:Displacement of [3H]dofetilide from human recombinant ERG potassium channel expressed in HEK293 cells by patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
LigandPNGBDBM50411753(CHEMBL429924)
Affinity DataIC50: 1.58E+8nMAssay Description:Displacement of [3H]dofetilide from human recombinant ERG potassium channel expressed in HEK293 cells by patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
LigandPNGBDBM50411752(CHEMBL271971)
Affinity DataIC50: 2.82E+7nMAssay Description:Displacement of [3H]dofetilide from human recombinant ERG potassium channel expressed in HEK293 cells by patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
LigandPNGBDBM50411751(CHEMBL271998)
Affinity DataIC50: 6.61E+7nMAssay Description:Displacement of [3H]dofetilide from human recombinant ERG potassium channel expressed in HEK293 cells by patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
LigandPNGBDBM50411750(CHEMBL270116)
Affinity DataIC50: 5.13E+8nMAssay Description:Displacement of [3H]dofetilide from human recombinant ERG potassium channel expressed in HEK293 cells by patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
LigandPNGBDBM50411748(CHEMBL409449)
Affinity DataIC50: 6.46E+8nMAssay Description:Displacement of [3H]dofetilide from human recombinant ERG potassium channel expressed in HEK293 cells by patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
LigandPNGBDBM50411747(CHEMBL402450)
Affinity DataIC50: 2.04E+7nMAssay Description:Displacement of [3H]dofetilide from human recombinant ERG potassium channel expressed in HEK293 cells by patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
LigandPNGBDBM50411746(CHEMBL271405)
Affinity DataIC50: 3.31E+7nMAssay Description:Displacement of [3H]dofetilide from human recombinant ERG potassium channel expressed in HEK293 cells by patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
LigandPNGBDBM50411745(CHEMBL411448)
Affinity DataIC50: 3.72E+7nMAssay Description:Displacement of [3H]dofetilide from human recombinant ERG potassium channel expressed in HEK293 cells by patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
LigandPNGBDBM50411744(CHEMBL406028)
Affinity DataIC50: 6.46E+7nMAssay Description:Displacement of [3H]dofetilide from human recombinant ERG potassium channel expressed in HEK293 cells by patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
LigandPNGBDBM50411743(CHEMBL429581)
Affinity DataIC50: 8.51E+7nMAssay Description:Displacement of [3H]dofetilide from human recombinant ERG potassium channel expressed in HEK293 cells by patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
LigandPNGBDBM50411742(CHEMBL272242)
Affinity DataIC50: 9.77E+7nMAssay Description:Displacement of [3H]dofetilide from human recombinant ERG potassium channel expressed in HEK293 cells by patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
LigandPNGBDBM50411741(CHEMBL429763)
Affinity DataIC50: 1.00E+8nMAssay Description:Displacement of [3H]dofetilide from human recombinant ERG potassium channel expressed in HEK293 cells by patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
LigandPNGBDBM50411740(CHEMBL272441)
Affinity DataIC50: 4.37E+7nMAssay Description:Displacement of [3H]dofetilide from human recombinant ERG potassium channel expressed in HEK293 cells by patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
LigandPNGBDBM50411739(CHEMBL271766)
Affinity DataIC50: 2.51E+8nMAssay Description:Displacement of [3H]dofetilide from human recombinant ERG potassium channel expressed in HEK293 cells by patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed