Compile Data Set for Download or QSAR
Report error Found 29 Enz. Inhib. hit(s) with all data for entry = 2807
TargetRAC-beta serine/threonine-protein kinase(Human)
Merck Research Laboratories

LigandPNGBDBM24887(5-{5-phenyl-6-[4-({4-[5-(pyridin-2-yl)-1H-1,2,4-tr...)
Affinity DataIC50: 22nMpH: 7.5 T: 2°CAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2008
Entry Details Article
PubMed
TargetRAC-beta serine/threonine-protein kinase(Human)
Merck Research Laboratories

LigandPNGBDBM24890(5-(6-{4-[(4-{4-amino-1H-pyrazolo[3,4-d]pyrimidin-1...)
Affinity DataIC50: 22nMpH: 7.5 T: 2°CAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2008
Entry Details Article
PubMed
TargetRAC-beta serine/threonine-protein kinase(Human)
Merck Research Laboratories

LigandPNGBDBM24886(5-{5-phenyl-6-[4-({4-[5-(pyridin-2-yl)-1H-pyrazol-...)
Affinity DataIC50: 28nMpH: 7.5 T: 2°CAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2008
Entry Details Article
PubMed
TargetRAC-beta serine/threonine-protein kinase(Human)
Merck Research Laboratories

LigandPNGBDBM24892(3-[({4-[5-(5-amino-1,3,4-thiadiazol-2-yl)-3-phenyl...)
Affinity DataIC50: 30nMpH: 7.5 T: 2°CAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2008
Entry Details Article
PubMed
TargetRAC-beta serine/threonine-protein kinase(Human)
Merck Research Laboratories

LigandPNGBDBM24885(5-{5-phenyl-6-[4-({4-[5-(pyridin-4-yl)-1H-pyrazol-...)
Affinity DataIC50: 38nMpH: 7.5 T: 2°CAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2008
Entry Details Article
PubMed
TargetRAC-beta serine/threonine-protein kinase(Human)
Merck Research Laboratories

LigandPNGBDBM24889(5-{5-phenyl-6-[4-({4-[4-(pyrazin-2-yl)-1H-pyrazol-...)
Affinity DataIC50: 51nMpH: 7.5 T: 2°CAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2008
Entry Details Article
PubMed
TargetRAC-beta serine/threonine-protein kinase(Human)
Merck Research Laboratories

LigandPNGBDBM24895(1-[1-({4-[3-phenyl-5-(pyrimidin-2-yl)pyridin-2-yl]...)
Affinity DataIC50: 62nMpH: 7.5 T: 2°CAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2008
Entry Details Article
PubMed
TargetRAC-beta serine/threonine-protein kinase(Human)
Merck Research Laboratories

LigandPNGBDBM24894(1-[1-({4-[3-phenyl-5-(1,3-thiazol-2-yl)pyridin-2-y...)
Affinity DataIC50: 64nMpH: 7.5 T: 2°CAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2008
Entry Details Article
PubMed
TargetRAC-beta serine/threonine-protein kinase(Human)
Merck Research Laboratories

LigandPNGBDBM24891(1-[1-({4-[5-(5-amino-1,3,4-thiadiazol-2-yl)-3-phen...)
Affinity DataIC50: 73nMpH: 7.5 T: 2°CAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2008
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

LigandPNGBDBM24887(5-{5-phenyl-6-[4-({4-[5-(pyridin-2-yl)-1H-1,2,4-tr...)
Affinity DataIC50: 85nMpH: 7.5 T: 2°CAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2008
Entry Details Article
PubMed
TargetRAC-beta serine/threonine-protein kinase(Human)
Merck Research Laboratories

LigandPNGBDBM24888(5-{5-phenyl-6-[4-({4-[4-(pyridin-2-yl)-1H-pyrazol-...)
Affinity DataIC50: 90nMpH: 7.5 T: 2°CAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2008
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

LigandPNGBDBM24886(5-{5-phenyl-6-[4-({4-[5-(pyridin-2-yl)-1H-pyrazol-...)
Affinity DataIC50: 95nMpH: 7.5 T: 2°CAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2008
Entry Details Article
PubMed
TargetRAC-beta serine/threonine-protein kinase(Human)
Merck Research Laboratories

LigandPNGBDBM24897(1-[1-({4-[3-phenyl-5-(1H-1,2,4-triazol-3-yl)pyridi...)
Affinity DataIC50: 101nMpH: 7.5 T: 2°CAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2008
Entry Details Article
PubMed
TargetRAC-beta serine/threonine-protein kinase(Human)
Merck Research Laboratories

LigandPNGBDBM24884(9-[1-({4-[3-phenyl-5-(1H-1,2,3,4-tetrazol-5-yl)pyr...)
Affinity DataIC50: 105nMpH: 7.5 T: 2°CAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2008
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

LigandPNGBDBM24892(3-[({4-[5-(5-amino-1,3,4-thiadiazol-2-yl)-3-phenyl...)
Affinity DataIC50: 114nMpH: 7.5 T: 2°CAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2008
Entry Details Article
PubMed
TargetRAC-beta serine/threonine-protein kinase(Human)
Merck Research Laboratories

LigandPNGBDBM24896(1-[1-({4-[5-(1,2,4-oxadiazol-3-yl)-3-phenylpyridin...)
Affinity DataIC50: 121nMpH: 7.5 T: 2°CAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2008
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

LigandPNGBDBM24885(5-{5-phenyl-6-[4-({4-[5-(pyridin-4-yl)-1H-pyrazol-...)
Affinity DataIC50: 123nMpH: 7.5 T: 2°CAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2008
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

LigandPNGBDBM24890(5-(6-{4-[(4-{4-amino-1H-pyrazolo[3,4-d]pyrimidin-1...)
Affinity DataIC50: 126nMpH: 7.5 T: 2°CAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2008
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

LigandPNGBDBM24889(5-{5-phenyl-6-[4-({4-[4-(pyrazin-2-yl)-1H-pyrazol-...)
Affinity DataIC50: 172nMpH: 7.5 T: 2°CAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2008
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

LigandPNGBDBM24896(1-[1-({4-[5-(1,2,4-oxadiazol-3-yl)-3-phenylpyridin...)
Affinity DataIC50: 180nMpH: 7.5 T: 2°CAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2008
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

LigandPNGBDBM24897(1-[1-({4-[3-phenyl-5-(1H-1,2,4-triazol-3-yl)pyridi...)
Affinity DataIC50: 182nMpH: 7.5 T: 2°CAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2008
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

LigandPNGBDBM24884(9-[1-({4-[3-phenyl-5-(1H-1,2,3,4-tetrazol-5-yl)pyr...)
Affinity DataIC50: 210nMpH: 7.5 T: 2°CAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2008
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

LigandPNGBDBM24888(5-{5-phenyl-6-[4-({4-[4-(pyridin-2-yl)-1H-pyrazol-...)
Affinity DataIC50: 214nMpH: 7.5 T: 2°CAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2008
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

LigandPNGBDBM24894(1-[1-({4-[3-phenyl-5-(1,3-thiazol-2-yl)pyridin-2-y...)
Affinity DataIC50: 264nMpH: 7.5 T: 2°CAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2008
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

LigandPNGBDBM24895(1-[1-({4-[3-phenyl-5-(pyrimidin-2-yl)pyridin-2-yl]...)
Affinity DataIC50: 306nMpH: 7.5 T: 2°CAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2008
Entry Details Article
PubMed
TargetRAC-beta serine/threonine-protein kinase(Human)
Merck Research Laboratories

LigandPNGBDBM24893(1-[1-({4-[3-phenyl-5-(pyridin-2-yl)pyridin-2-yl]ph...)
Affinity DataIC50: 370nMpH: 7.5 T: 2°CAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2008
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

LigandPNGBDBM24891(1-[1-({4-[5-(5-amino-1,3,4-thiadiazol-2-yl)-3-phen...)
Affinity DataIC50: 434nMpH: 7.5 T: 2°CAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2008
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

LigandPNGBDBM24893(1-[1-({4-[3-phenyl-5-(pyridin-2-yl)pyridin-2-yl]ph...)
Affinity DataIC50: 1.63E+3nMpH: 7.5 T: 2°CAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2008
Entry Details Article
PubMed
TargetRAC-gamma serine/threonine-protein kinase(Human)
Merck Research Laboratories

LigandPNGBDBM24884(9-[1-({4-[3-phenyl-5-(1H-1,2,3,4-tetrazol-5-yl)pyr...)
Affinity DataIC50: 5.00E+4nMpH: 7.5 T: 2°CAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2008
Entry Details Article
PubMed