Compile Data Set for Download or QSAR
Report error Found 19 Enz. Inhib. hit(s) with all data for entry = 50038088
TargetGrowth hormone secretagogue receptor type 1(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50235838((4-hydroxy-butyl)-carbamic acid 2-{5-[(S)-1-(2-ami...)
Affinity DataEC50:  0.340nMAssay Description:Inhibition of human growth hormone secretagogue receptor assessed as measuring intracellular calcium level by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50235845((S)-2-(5-(2-(2,4-difluorobenzyloxy)-1-(2-amino-2-m...)
Affinity DataEC50:  0.420nMAssay Description:Inhibition of human growth hormone secretagogue receptor assessed as measuring intracellular calcium level by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50235842((S)-2-(5-(2-(2-chlorobenzyloxy)-1-(2-amino-2-methy...)
Affinity DataEC50:  0.450nMAssay Description:Inhibition of human growth hormone secretagogue receptor assessed as measuring intracellular calcium level by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50235849((4-hydroxy-butyl)-carbamic acid 2-{5-[(S)-1-(2-ami...)
Affinity DataEC50:  0.510nMAssay Description:Inhibition of human growth hormone secretagogue receptor assessed as measuring intracellular calcium level by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50235854((S)-2-(5-(2-(2,3-dichlorobenzyloxy)-1-(2-amino-2-m...)
Affinity DataEC50:  0.610nMAssay Description:Inhibition of human growth hormone secretagogue receptor assessed as measuring intracellular calcium level by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50235840((S)-2-(5-(2-(2-(trifluoromethyl)benzyloxy)-1-(2-am...)
Affinity DataEC50:  0.720nMAssay Description:Inhibition of human growth hormone secretagogue receptor assessed as measuring intracellular calcium level by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50235850(2-(5-((S)-2-(2-(3,5-dimethylisoxazol-4-yl)benzylox...)
Affinity DataEC50:  1.04nMAssay Description:Inhibition of human growth hormone secretagogue receptor assessed as measuring intracellular calcium level by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50235839((S)-2-(5-(2-(2-methoxybenzyloxy)-1-(2-amino-2-meth...)
Affinity DataEC50:  1.11nMAssay Description:Inhibition of human growth hormone secretagogue receptor assessed as measuring intracellular calcium level by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50235852(2-(5-((S)-2-(2-(pyridin-3-yl)benzyloxy)-1-(2-amino...)
Affinity DataEC50:  1.18nMAssay Description:Inhibition of human growth hormone secretagogue receptor assessed as measuring intracellular calcium level by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50235853((S)-2-(5-(2-(2-cyanobenzyloxy)-1-(2-amino-2-methyl...)
Affinity DataEC50:  1.26nMAssay Description:Inhibition of human growth hormone secretagogue receptor assessed as measuring intracellular calcium level by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50366689(GHRELIN)
Affinity DataEC50:  1.41nMAssay Description:Inhibition of human growth hormone secretagogue receptor assessed as measuring intracellular calcium level by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50235843((S)-2-(5-(2-(3-chlorobenzyloxy)-1-(2-amino-2-methy...)
Affinity DataEC50:  1.60nMAssay Description:Inhibition of human growth hormone secretagogue receptor assessed as measuring intracellular calcium level by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50235847((S)-2-(5-(1-(2-amino-2-methylpropanamido)-2-(cyclo...)
Affinity DataEC50:  1.66nMAssay Description:Inhibition of human growth hormone secretagogue receptor assessed as measuring intracellular calcium level by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50235841((S)-2-(5-(2-(3-(trifluoromethyl)benzyloxy)-1-(2-am...)
Affinity DataEC50:  1.79nMAssay Description:Inhibition of human growth hormone secretagogue receptor assessed as measuring intracellular calcium level by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM21941(2-{5-[(1S)-1-(2-amino-2-methylpropanamido)-2-(benz...)
Affinity DataEC50:  1.92nMAssay Description:Inhibition of human growth hormone secretagogue receptor assessed as measuring intracellular calcium level by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50235846((S)-2-(5-(2-(3-(trifluoromethoxy)benzyloxy)-1-(2-a...)
Affinity DataEC50:  3.10nMAssay Description:Inhibition of human growth hormone secretagogue receptor assessed as measuring intracellular calcium level by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50235848((S)-2-(5-(2-(3,5-dichlorobenzyloxy)-1-(2-amino-2-m...)
Affinity DataEC50:  6.75nMAssay Description:Inhibition of human growth hormone secretagogue receptor assessed as measuring intracellular calcium level by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50235851((S)-2-(5-(2-(4-(trifluoromethoxy)benzyloxy)-1-(2-a...)
Affinity DataEC50:  33.2nMAssay Description:Inhibition of human growth hormone secretagogue receptor assessed as measuring intracellular calcium level by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50235844((S)-2-(5-(2-(3,5-bis(trifluoromethyl)benzyloxy)-1-...)
Affinity DataEC50:  34nMAssay Description:Inhibition of human growth hormone secretagogue receptor assessed as measuring intracellular calcium level by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed