Compile Data Set for Download or QSAR
Report error Found 70 Enz. Inhib. hit(s) with all data for entry = 50022534
LigandPNGBDBM50236266(7-[(1E)-1-(methoxyimino)ethyl]-19-methyl-3,13,19,2...)
Affinity DataIC50: 1nMAssay Description:Inhibition of human recombinant VEGFR2 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
LigandPNGBDBM50236260(7-[(1E)-1-(hydroxyimino)ethyl]-19-methyl-3,13,19,2...)
Affinity DataIC50: 1nMAssay Description:Inhibition of human recombinant VEGFR2 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
LigandPNGBDBM50236262(7-[(1E)-1-(methoxyimino)ethyl]-19-methyl-3-propyl-...)
Affinity DataIC50: 1nMAssay Description:Inhibition of human recombinant VEGFR2 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
LigandPNGBDBM50236262(7-[(1E)-1-(methoxyimino)ethyl]-19-methyl-3-propyl-...)
Affinity DataIC50: 1nMAssay Description:Inhibition of VEGF-stimulated VEGFR2 autophosphorylation in HUVEC cells at 50 nM relative to controlMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50236270(1-(4-(4-amino-6-(4-methoxyphenyl)furo[2,3-d]pyrimi...)
Affinity DataIC50: 2nMAssay Description:Inhibition of human recombinant TIE2 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
LigandPNGBDBM50236263(19-methyl-7-[(1E)-1-[(2-methylpropoxy)imino]ethyl]...)
Affinity DataIC50: 2nMAssay Description:Inhibition of VEGF-stimulated VEGFR2 autophosphorylation in HUVEC cells at 50 nM relative to controlMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
LigandPNGBDBM50236246(7-[(1E)-1-(ethoxyimino)ethyl]-19-methyl-3,13,19,20...)
Affinity DataIC50: 2nMAssay Description:Inhibition of human recombinant VEGFR2 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
LigandPNGBDBM50236259(3-ethyl-19-methyl-7-[(1E)-1-[(2-methylpropoxy)imin...)
Affinity DataIC50: 3nMAssay Description:Inhibition of VEGF-stimulated VEGFR2 autophosphorylation in HUVEC cells at 50 nM relative to controlMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
LigandPNGBDBM50236264(19-methyl-7-[(1E)-1-[(propan-2-yloxy)imino]ethyl]-...)
Affinity DataIC50: 3nMAssay Description:Inhibition of human recombinant VEGFR2 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
LigandPNGBDBM50236270(1-(4-(4-amino-6-(4-methoxyphenyl)furo[2,3-d]pyrimi...)
Affinity DataIC50: 3nMAssay Description:Inhibition of human recombinant VEGFR2 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
LigandPNGBDBM50236258(19-methyl-7-[(1E)-1-[(2-methylpropoxy)imino]ethyl]...)
Affinity DataIC50: 4nMAssay Description:Inhibition of VEGF-stimulated VEGFR2 autophosphorylation in HUVEC cells at 50 nM relative to controlMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
LigandPNGBDBM50236246(7-[(1E)-1-(ethoxyimino)ethyl]-19-methyl-3,13,19,20...)
Affinity DataIC50: 4nMAssay Description:Inhibition of VEGF-stimulated VEGFR2 autophosphorylation in HUVEC cells at 50 nM relative to controlMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
LigandPNGBDBM50236267(7-[(1E)-1-(methoxyimino)-2-methylpropyl]-19-methyl...)
Affinity DataIC50: 4nMAssay Description:Inhibition of human recombinant VEGFR2 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
LigandPNGBDBM50236256(3-ethyl-7-[(1E)-1-(methoxyimino)ethyl]-19-methyl-3...)
Affinity DataIC50: 4nMAssay Description:Inhibition of human recombinant VEGFR2 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
LigandPNGBDBM50236264(19-methyl-7-[(1E)-1-[(propan-2-yloxy)imino]ethyl]-...)
Affinity DataIC50: 4nMAssay Description:Inhibition of VEGF-stimulated VEGFR2 autophosphorylation in HUVEC cells at 50 nM relative to controlMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
LigandPNGBDBM50236268(7-[(1E)-1-(ethoxyimino)ethyl]-19-methyl-3-(2-methy...)
Affinity DataIC50: 4nMAssay Description:Inhibition of human recombinant VEGFR2 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
LigandPNGBDBM50236252(7-[(1E)-1-(methoxyimino)ethyl]-19-methyl-3-(propan...)
Affinity DataIC50: 4nMAssay Description:Inhibition of human recombinant VEGFR2 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
LigandPNGBDBM50236254(7-[(1E)-1-(ethoxyimino)ethyl]-19-methyl-3-(propan-...)
Affinity DataIC50: 4nMAssay Description:Inhibition of human recombinant VEGFR2 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
LigandPNGBDBM50236248(7-[(1E)-(ethoxyimino)methyl]-19-methyl-3,13,19,20-...)
Affinity DataIC50: 4nMAssay Description:Inhibition of human recombinant VEGFR2 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
LigandPNGBDBM50236268(7-[(1E)-1-(ethoxyimino)ethyl]-19-methyl-3-(2-methy...)
Affinity DataIC50: 4nMAssay Description:Inhibition of VEGF-stimulated VEGFR2 autophosphorylation in HUVEC cells at 50 nM relative to controlMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
LigandPNGBDBM50236257(19-methyl-3-(2-methylpropyl)-7-[(1E)-1-[(propan-2-...)
Affinity DataIC50: 4nMAssay Description:Inhibition of VEGF-stimulated VEGFR2 autophosphorylation in HUVEC cells at 50 nM relative to controlMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
LigandPNGBDBM50236251(7-[(1E)-1-(methoxyimino)ethyl]-19-methyl-3-(2-meth...)
Affinity DataIC50: 4nMAssay Description:Inhibition of VEGF-stimulated VEGFR2 autophosphorylation in HUVEC cells at 50 nM relative to controlMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
LigandPNGBDBM50236254(7-[(1E)-1-(ethoxyimino)ethyl]-19-methyl-3-(propan-...)
Affinity DataIC50: 4nMAssay Description:Inhibition of VEGF-stimulated VEGFR2 autophosphorylation in HUVEC cells at 50 nM relative to controlMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
LigandPNGBDBM50236269(19-methyl-3-(propan-2-yl)-7-[(1E)-1-[(propan-2-ylo...)
Affinity DataIC50: 4nMAssay Description:Inhibition of VEGF-stimulated VEGFR2 autophosphorylation in HUVEC cells at 50 nM relative to controlMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
LigandPNGBDBM50236253(7-[(1E)-1-(methoxyimino)ethyl]-3,19-dimethyl-3,13,...)
Affinity DataIC50: 5nMAssay Description:Inhibition of human recombinant VEGFR2 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
LigandPNGBDBM50236251(7-[(1E)-1-(methoxyimino)ethyl]-19-methyl-3-(2-meth...)
Affinity DataIC50: 7nMAssay Description:Inhibition of human recombinant VEGFR2 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
LigandPNGBDBM50236251(7-[(1E)-1-(methoxyimino)ethyl]-19-methyl-3-(2-meth...)
Affinity DataIC50: 8nMAssay Description:Inhibition of VEGFR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
LigandPNGBDBM50236258(19-methyl-7-[(1E)-1-[(2-methylpropoxy)imino]ethyl]...)
Affinity DataIC50: 10nMAssay Description:Inhibition of human recombinant VEGFR2 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50236258(19-methyl-7-[(1E)-1-[(2-methylpropoxy)imino]ethyl]...)
Affinity DataIC50: 10nMAssay Description:Inhibition of human recombinant TIE2 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
LigandPNGBDBM50236251(7-[(1E)-1-(methoxyimino)ethyl]-19-methyl-3-(2-meth...)
Affinity DataIC50: 10nMAssay Description:Inhibition of VEGFR3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
LigandPNGBDBM25115(3-[(4-bromo-2,6-difluorophenyl)methoxy]-5-({[4-(py...)
Affinity DataIC50: 11nMAssay Description:Inhibition of human recombinant VEGFR2 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
LigandPNGBDBM50236269(19-methyl-3-(propan-2-yl)-7-[(1E)-1-[(propan-2-ylo...)
Affinity DataIC50: 11nMAssay Description:Inhibition of human recombinant VEGFR2 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
LigandPNGBDBM50236247(3-butyl-7-[(1E)-1-(methoxyimino)ethyl]-19-methyl-3...)
Affinity DataIC50: 12nMAssay Description:Inhibition of human recombinant VEGFR2 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50236254(7-[(1E)-1-(ethoxyimino)ethyl]-19-methyl-3-(propan-...)
Affinity DataIC50: 14nMAssay Description:Inhibition of c-srcMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
LigandPNGBDBM50236249(7-[(1E)-(methoxyimino)methyl]-19-methyl-3,13,19,20...)
Affinity DataIC50: 18nMAssay Description:Inhibition of human recombinant VEGFR2 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM25115(3-[(4-bromo-2,6-difluorophenyl)methoxy]-5-({[4-(py...)
Affinity DataIC50: 18nMAssay Description:Inhibition of human recombinant TIE2 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
LigandPNGBDBM50236261(7-[(1E)-1-(ethoxyimino)-2-methylpropyl]-19-methyl-...)
Affinity DataIC50: 23nMAssay Description:Inhibition of human recombinant VEGFR2 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50236265(19-methyl-7-[(1E)-1-[(2-methylpropoxy)imino]ethyl]...)
Affinity DataIC50: 23nMAssay Description:Inhibition of human recombinant TIE2 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50236246(7-[(1E)-1-(ethoxyimino)ethyl]-19-methyl-3,13,19,20...)
Affinity DataIC50: 23nMAssay Description:Inhibition of human recombinant TIE2 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
LigandPNGBDBM50236259(3-ethyl-19-methyl-7-[(1E)-1-[(2-methylpropoxy)imin...)
Affinity DataIC50: 24nMAssay Description:Inhibition of human recombinant VEGFR2 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50236268(7-[(1E)-1-(ethoxyimino)ethyl]-19-methyl-3-(2-methy...)
Affinity DataIC50: 25nMAssay Description:Inhibition of human recombinant TIE2 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50236254(7-[(1E)-1-(ethoxyimino)ethyl]-19-methyl-3-(propan-...)
Affinity DataIC50: 26nMAssay Description:Inhibition of human recombinant TIE2 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50236264(19-methyl-7-[(1E)-1-[(propan-2-yloxy)imino]ethyl]-...)
Affinity DataIC50: 28nMAssay Description:Inhibition of human recombinant TIE2 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50236262(7-[(1E)-1-(methoxyimino)ethyl]-19-methyl-3-propyl-...)
Affinity DataIC50: 30nMAssay Description:Inhibition of human recombinant TIE2 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50236251(7-[(1E)-1-(methoxyimino)ethyl]-19-methyl-3-(2-meth...)
Affinity DataIC50: 30nMAssay Description:Inhibition of human recombinant TIE2 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
LigandPNGBDBM50236257(19-methyl-3-(2-methylpropyl)-7-[(1E)-1-[(propan-2-...)
Affinity DataIC50: 31nMAssay Description:Inhibition of human recombinant VEGFR2 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
LigandPNGBDBM50236250(7-[(1E)-1-[(tert-butoxy)imino]ethyl]-19-methyl-3,1...)
Affinity DataIC50: 31nMAssay Description:Inhibition of human recombinant VEGFR2 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50236251(7-[(1E)-1-(methoxyimino)ethyl]-19-methyl-3-(2-meth...)
Affinity DataIC50: 43nMAssay Description:Inhibition of c-srcMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50236260(7-[(1E)-1-(hydroxyimino)ethyl]-19-methyl-3,13,19,2...)
Affinity DataIC50: 44nMAssay Description:Inhibition of human recombinant TIE2 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50236259(3-ethyl-19-methyl-7-[(1E)-1-[(2-methylpropoxy)imin...)
Affinity DataIC50: 45nMAssay Description:Inhibition of human recombinant TIE2 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
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