Compile Data Set for Download or QSAR
Report error Found 40 Enz. Inhib. hit(s) with all data for entry = 50022549
TargetMitogen-activated protein kinase 11(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50236473((R)-2-(sec-butylamino)-N-(2-methyl-5-(methylcarbam...)
Affinity DataIC50: 1.5nMAssay Description:Inhibition of human p38betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50236476(N-(5-(ethylcarbamoyl)-2-methylphenyl)-2-(propylami...)
Affinity DataIC50: 2nMAssay Description:Inhibition of human p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50236483((S)-2-(sec-butylamino)-N-(2-methyl-5-(methylcarbam...)
Affinity DataIC50: 2.30nMAssay Description:Inhibition of human p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50236490(N-(5-carbamoyl-2-methylphenyl)-2-(isopropylamino)t...)
Affinity DataIC50: 3.20nMAssay Description:Inhibition of human p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50236474(N-(5-(ethylcarbamoyl)-2-methylphenyl)-2-(isopropyl...)
Affinity DataIC50: 3.40nMAssay Description:Inhibition of human p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50236473((R)-2-(sec-butylamino)-N-(2-methyl-5-(methylcarbam...)
Affinity DataIC50: 3.5nMAssay Description:Inhibition of human p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50236475(2-(isopropylamino)-N-(2-methyl-5-(methylcarbamoyl)...)
Affinity DataIC50: 3.5nMAssay Description:Inhibition of human p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50236487(2-(isopropylamino)-N-(5-(isoxazol-3-ylcarbamoyl)-2...)
Affinity DataIC50: 3.80nMAssay Description:Inhibition of human p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50236488(N-(5-carbamoyl-2-methylphenyl)-2-(propylamino)thia...)
Affinity DataIC50: 4.10nMAssay Description:Inhibition of human p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50236478(N-(5-((1H-pyrazol-5-yl)carbamoyl)-2-methylphenyl)-...)
Affinity DataIC50: 4.20nMAssay Description:Inhibition of human p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50236480(N-(2-methyl-5-(methylcarbamoyl)phenyl)-2-(propylam...)
Affinity DataIC50: 4.5nMAssay Description:Inhibition of human p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50236485(2-(isopropylamino)-N-(2-methyl-5-((1-methyl-1H-pyr...)
Affinity DataIC50: 5.40nMAssay Description:Inhibition of human p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50236482(N-(2-chloro-6-methylphenyl)-2-(isopropylamino)thia...)
Affinity DataIC50: 13nMAssay Description:Inhibition of human p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50236477(2-(2-methoxyethylamino)-N-(2-methyl-5-(methylcarba...)
Affinity DataIC50: 22nMAssay Description:Inhibition of human p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50236486(N-(2-chloro-6-methylphenyl)-2-(propylamino)thiazol...)
Affinity DataIC50: 28nMAssay Description:Inhibition of human p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50236479(N-ethyl-3-(2-(isopropylamino)-6-oxo-4H-pyrrolo[3,4...)
Affinity DataIC50: 34nMAssay Description:Inhibition of human p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50236484(N-(2-chloro-6-methylphenyl)-2-(cyclobutylamino)thi...)
Affinity DataIC50: 36nMAssay Description:Inhibition of human p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50236481(N-(2-chloro-6-methylphenyl)-2-(cyclopropylamino)th...)
Affinity DataIC50: 39nMAssay Description:Inhibition of human p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50236471(3-(2-(cyclopentylamino)-6-oxo-3a,4,6,6a-tetrahydro...)
Affinity DataIC50: 53nMAssay Description:Inhibition of human p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50156469(N-(2-chloro-6-methylphenyl)-2-(phenylamino)thiazol...)
Affinity DataIC50: 62nMAssay Description:Inhibition of human p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50236491(3-(2-(cyclopentylamino)-6-oxo-4H-pyrrolo[3,4-d]thi...)
Affinity DataIC50: 110nMAssay Description:Inhibition of human p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50236495(3-(2-(isopropylamino)-6-oxo-4H-pyrrolo[3,4-d]thiaz...)
Affinity DataIC50: 110nMAssay Description:Inhibition of human p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50236472(N-(5-(ethylcarbamoyl)-2-methylphenyl)-4-methyl-2-(...)
Affinity DataIC50: 130nMAssay Description:Inhibition of human p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50236493(N-(2-chloro-6-methylphenyl)-2-(ethylamino)thiazole...)
Affinity DataIC50: 140nMAssay Description:Inhibition of human p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50236481(N-(2-chloro-6-methylphenyl)-2-(cyclopropylamino)th...)
Affinity DataIC50: 140nMAssay Description:Inhibition of LckMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50236494(N-ethyl-4-methyl-3-(6-oxo-2-(propylamino)-4H-pyrro...)
Affinity DataIC50: 160nMAssay Description:Inhibition of human p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50236492(N,4-dimethyl-3-(6-oxo-2-(propylamino)-3a,4,6,6a-te...)
Affinity DataIC50: 270nMAssay Description:Inhibition of human p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50236489(2-(ethylamino)-N-(5-(ethylcarbamoyl)-2-methylpheny...)
Affinity DataIC50: 330nMAssay Description:Inhibition of human p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50236487(2-(isopropylamino)-N-(5-(isoxazol-3-ylcarbamoyl)-2...)
Affinity DataIC50: 380nMAssay Description:Inhibition of LckMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50236476(N-(5-(ethylcarbamoyl)-2-methylphenyl)-2-(propylami...)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of LckMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50236484(N-(2-chloro-6-methylphenyl)-2-(cyclobutylamino)thi...)
Affinity DataIC50: 3.31E+3nMAssay Description:Inhibition of LckMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50236480(N-(2-methyl-5-(methylcarbamoyl)phenyl)-2-(propylam...)
Affinity DataIC50: 4.80E+3nMAssay Description:Inhibition of LckMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50236485(2-(isopropylamino)-N-(2-methyl-5-((1-methyl-1H-pyr...)
Affinity DataIC50: 5.80E+3nMAssay Description:Inhibition of LckMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50236473((R)-2-(sec-butylamino)-N-(2-methyl-5-(methylcarbam...)
Affinity DataIC50: 2.20E+4nMAssay Description:Inhibition of LckMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 13(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50236473((R)-2-(sec-butylamino)-N-(2-methyl-5-(methylcarbam...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of human p38deltaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 12(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50236473((R)-2-(sec-butylamino)-N-(2-methyl-5-(methylcarbam...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of human p38-gammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50236474(N-(5-(ethylcarbamoyl)-2-methylphenyl)-2-(isopropyl...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of LckMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50236490(N-(5-carbamoyl-2-methylphenyl)-2-(isopropylamino)t...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of LckMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50236475(2-(isopropylamino)-N-(2-methyl-5-(methylcarbamoyl)...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of LckMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50236483((S)-2-(sec-butylamino)-N-(2-methyl-5-(methylcarbam...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of LckMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed