Compile Data Set for Download or QSAR
Report error Found 64 Enz. Inhib. hit(s) with all data for entry = 50025793
TargetPeroxisome proliferator-activated receptor gamma(Human)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50103960(3-(4-(2-(5-(3-fluorophenyl)-1,2,4-oxadiazol-3-yl)e...)
Affinity DataEC50:  2nMAssay Description:Agonist activity at human PPARgamma expressed in african green monkey CV1 cells co-transfected with Gal4 assessed as reporter activity by transient t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50103955(3-{4-[5-(4-tert-Butyl-phenyl)-[1,2,4]oxadiazol-3-y...)
Affinity DataEC50:  3nMAssay Description:Agonist activity at human PPARgamma expressed in african green monkey CV1 cells co-transfected with Gal4 assessed as reporter activity by transient t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50103953(3-(4-{2-[5-(3-Chloro-phenyl)-[1,2,4]oxadiazol-3-yl...)
Affinity DataEC50:  4nMAssay Description:Agonist activity at human PPARgamma expressed in african green monkey CV1 cells co-transfected with Gal4 assessed as reporter activity by transient t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50103957(3-(4-(2-(5-(3,5-bis(trifluoromethyl)phenyl)-1,2,4-...)
Affinity DataEC50:  4nMAssay Description:Agonist activity at human PPARgamma expressed in african green monkey CV1 cells co-transfected with Gal4 assessed as reporter activity by transient t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50103950(2-isopropoxy-3-(4-((5-(4-isopropylphenyl)-1,2,4-ox...)
Affinity DataEC50:  4nMAssay Description:Agonist activity at human PPARgamma expressed in african green monkey CV1 cells co-transfected with Gal4 assessed as reporter activity by transient t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50103941(2-isopropoxy-3-(4-(2-(5-(3-(trifluoromethyl)phenyl...)
Affinity DataEC50:  6nMAssay Description:Agonist activity at human PPARgamma expressed in african green monkey CV1 cells co-transfected with Gal4 assessed as reporter activity by transient t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50103940(3-(4-((5-(3,5-bis(trifluoromethyl)phenyl)-1,2,4-ox...)
Affinity DataEC50:  6nMAssay Description:Agonist activity at human PPARalpha expressed in african green monkey CV1 cells co-transfected with Gal4 assessed as reporter activity by transient t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50103954(2-isopropoxy-3-(4-(2-(5-phenyl-1,2,4-oxadiazol-3-y...)
Affinity DataEC50:  13nMAssay Description:Agonist activity at human PPARgamma expressed in african green monkey CV1 cells co-transfected with Gal4 assessed as reporter activity by transient t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50103943(3-{4-[5-(4-Chloro-phenyl)-[1,2,4]oxadiazol-3-ylmet...)
Affinity DataEC50:  13nMAssay Description:Agonist activity at human PPARalpha expressed in african green monkey CV1 cells co-transfected with Gal4 assessed as reporter activity by transient t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50103950(2-isopropoxy-3-(4-((5-(4-isopropylphenyl)-1,2,4-ox...)
Affinity DataEC50:  13nMAssay Description:Agonist activity at human PPARalpha expressed in african green monkey CV1 cells co-transfected with Gal4 assessed as reporter activity by transient t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50103948(2-isopropoxy-3-(4-((5-p-tolyl-1,2,4-oxadiazol-3-yl...)
Affinity DataEC50:  16nMAssay Description:Agonist activity at human PPARgamma expressed in african green monkey CV1 cells co-transfected with Gal4 assessed as reporter activity by transient t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50103959(2-isopropoxy-3-(4-((5-(4-(trifluoromethoxy)phenyl)...)
Affinity DataEC50:  20nMAssay Description:Agonist activity at human PPARalpha expressed in african green monkey CV1 cells co-transfected with Gal4 assessed as reporter activity by transient t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50103943(3-{4-[5-(4-Chloro-phenyl)-[1,2,4]oxadiazol-3-ylmet...)
Affinity DataEC50:  20nMAssay Description:Agonist activity at human PPARgamma expressed in african green monkey CV1 cells co-transfected with Gal4 assessed as reporter activity by transient t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50103948(2-isopropoxy-3-(4-((5-p-tolyl-1,2,4-oxadiazol-3-yl...)
Affinity DataEC50:  25nMAssay Description:Agonist activity at human PPARalpha expressed in african green monkey CV1 cells co-transfected with Gal4 assessed as reporter activity by transient t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50103944(3-(4-(2-(5-(4-chlorophenyl)-1,2,4-oxadiazol-3-yl)e...)
Affinity DataEC50:  25nMAssay Description:Agonist activity at human PPARgamma expressed in african green monkey CV1 cells co-transfected with Gal4 assessed as reporter activity by transient t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50103949(2-Isopropoxy-3-{4-[5-(4-trifluoromethyl-phenyl)-[1...)
Affinity DataEC50:  25nMAssay Description:Agonist activity at human PPARgamma expressed in african green monkey CV1 cells co-transfected with Gal4 assessed as reporter activity by transient t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50103940(3-(4-((5-(3,5-bis(trifluoromethyl)phenyl)-1,2,4-ox...)
Affinity DataEC50:  32nMAssay Description:Agonist activity at human PPARgamma expressed in african green monkey CV1 cells co-transfected with Gal4 assessed as reporter activity by transient t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50103949(2-Isopropoxy-3-{4-[5-(4-trifluoromethyl-phenyl)-[1...)
Affinity DataEC50:  32nMAssay Description:Agonist activity at human PPARalpha expressed in african green monkey CV1 cells co-transfected with Gal4 assessed as reporter activity by transient t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50103947(3-{4-[5-(4-Bromo-phenyl)-[1,2,4]oxadiazol-3-ylmeth...)
Affinity DataEC50:  32nMAssay Description:Agonist activity at human PPARgamma expressed in african green monkey CV1 cells co-transfected with Gal4 assessed as reporter activity by transient t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50103939(2-isopropoxy-3-(4-((5-o-tolyl-1,2,4-oxadiazol-3-yl...)
Affinity DataEC50:  40nMAssay Description:Agonist activity at human PPARalpha expressed in african green monkey CV1 cells co-transfected with Gal4 assessed as reporter activity by transient t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50103951(3-(4-{2-[5-(4-Fluoro-phenyl)-[1,2,4]oxadiazol-3-yl...)
Affinity DataEC50:  40nMAssay Description:Agonist activity at human PPARgamma expressed in african green monkey CV1 cells co-transfected with Gal4 assessed as reporter activity by transient t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50103947(3-{4-[5-(4-Bromo-phenyl)-[1,2,4]oxadiazol-3-ylmeth...)
Affinity DataEC50:  40nMAssay Description:Agonist activity at human PPARalpha expressed in african green monkey CV1 cells co-transfected with Gal4 assessed as reporter activity by transient t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50103946(3-(4-((5-(3,5-difluorophenyl)-1,2,4-oxadiazol-3-yl...)
Affinity DataEC50:  40nMAssay Description:Agonist activity at human PPARalpha expressed in african green monkey CV1 cells co-transfected with Gal4 assessed as reporter activity by transient t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50103955(3-{4-[5-(4-tert-Butyl-phenyl)-[1,2,4]oxadiazol-3-y...)
Affinity DataEC50:  40nMAssay Description:Agonist activity at human PPARalpha expressed in african green monkey CV1 cells co-transfected with Gal4 assessed as reporter activity by transient t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50103957(3-(4-(2-(5-(3,5-bis(trifluoromethyl)phenyl)-1,2,4-...)
Affinity DataEC50:  50nMAssay Description:Agonist activity at human PPARalpha expressed in african green monkey CV1 cells co-transfected with Gal4 assessed as reporter activity by transient t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50103956(2-Isopropoxy-3-[4-(5-m-tolyl-[1,2,4]oxadiazol-3-yl...)
Affinity DataEC50:  50nMAssay Description:Agonist activity at human PPARgamma expressed in african green monkey CV1 cells co-transfected with Gal4 assessed as reporter activity by transient t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50103959(2-isopropoxy-3-(4-((5-(4-(trifluoromethoxy)phenyl)...)
Affinity DataEC50:  63nMAssay Description:Agonist activity at human PPARgamma expressed in african green monkey CV1 cells co-transfected with Gal4 assessed as reporter activity by transient t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50103956(2-Isopropoxy-3-[4-(5-m-tolyl-[1,2,4]oxadiazol-3-yl...)
Affinity DataEC50:  79nMAssay Description:Agonist activity at human PPARalpha expressed in african green monkey CV1 cells co-transfected with Gal4 assessed as reporter activity by transient t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50103938(2-isopropoxy-3-(4-((5-phenyl-1,2,4-oxadiazol-3-yl)...)
Affinity DataEC50:  79nMAssay Description:Agonist activity at human PPARgamma expressed in african green monkey CV1 cells co-transfected with Gal4 assessed as reporter activity by transient t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50103958(3-{4-[5-(3-Fluoro-phenyl)-[1,2,4]oxadiazol-3-ylmet...)
Affinity DataEC50:  79nMAssay Description:Agonist activity at human PPARalpha expressed in african green monkey CV1 cells co-transfected with Gal4 assessed as reporter activity by transient t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50103946(3-(4-((5-(3,5-difluorophenyl)-1,2,4-oxadiazol-3-yl...)
Affinity DataEC50:  100nMAssay Description:Agonist activity at human PPARgamma expressed in african green monkey CV1 cells co-transfected with Gal4 assessed as reporter activity by transient t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50103958(3-{4-[5-(3-Fluoro-phenyl)-[1,2,4]oxadiazol-3-ylmet...)
Affinity DataEC50:  100nMAssay Description:Agonist activity at human PPARgamma expressed in african green monkey CV1 cells co-transfected with Gal4 assessed as reporter activity by transient t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50103939(2-isopropoxy-3-(4-((5-o-tolyl-1,2,4-oxadiazol-3-yl...)
Affinity DataEC50:  100nMAssay Description:Agonist activity at human PPARgamma expressed in african green monkey CV1 cells co-transfected with Gal4 assessed as reporter activity by transient t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50103953(3-(4-{2-[5-(3-Chloro-phenyl)-[1,2,4]oxadiazol-3-yl...)
Affinity DataEC50:  100nMAssay Description:Agonist activity at human PPARdelta expressed in african green monkey CV1 cells co-transfected with Gal4 assessed as reporter activity by transient t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50103946(3-(4-((5-(3,5-difluorophenyl)-1,2,4-oxadiazol-3-yl...)
Affinity DataEC50:  160nMAssay Description:Agonist activity at human PPARdelta expressed in african green monkey CV1 cells co-transfected with Gal4 assessed as reporter activity by transient t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50103945(2-Isopropoxy-3-(4-{2-[5-(2-trifluoromethyl-phenyl)...)
Affinity DataEC50:  160nMAssay Description:Agonist activity at human PPARgamma expressed in african green monkey CV1 cells co-transfected with Gal4 assessed as reporter activity by transient t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50103938(2-isopropoxy-3-(4-((5-phenyl-1,2,4-oxadiazol-3-yl)...)
Affinity DataEC50:  160nMAssay Description:Agonist activity at human PPARalpha expressed in african green monkey CV1 cells co-transfected with Gal4 assessed as reporter activity by transient t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50103952(3-(4-((5-(4-fluorophenyl)-1,2,4-oxadiazol-3-yl)met...)
Affinity DataEC50:  160nMAssay Description:Agonist activity at human PPARalpha expressed in african green monkey CV1 cells co-transfected with Gal4 assessed as reporter activity by transient t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50103941(2-isopropoxy-3-(4-(2-(5-(3-(trifluoromethyl)phenyl...)
Affinity DataEC50:  200nMAssay Description:Agonist activity at human PPARalpha expressed in african green monkey CV1 cells co-transfected with Gal4 assessed as reporter activity by transient t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50103952(3-(4-((5-(4-fluorophenyl)-1,2,4-oxadiazol-3-yl)met...)
Affinity DataEC50:  200nMAssay Description:Agonist activity at human PPARgamma expressed in african green monkey CV1 cells co-transfected with Gal4 assessed as reporter activity by transient t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50103942(3-(4-((5-cyclohexyl-1,2,4-oxadiazol-3-yl)methoxy)p...)
Affinity DataEC50:  230nMAssay Description:Agonist activity at human PPARgamma expressed in african green monkey CV1 cells co-transfected with Gal4 assessed as reporter activity by transient t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50103942(3-(4-((5-cyclohexyl-1,2,4-oxadiazol-3-yl)methoxy)p...)
Affinity DataEC50:  240nMAssay Description:Agonist activity at human PPARalpha expressed in african green monkey CV1 cells co-transfected with Gal4 assessed as reporter activity by transient t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50103953(3-(4-{2-[5-(3-Chloro-phenyl)-[1,2,4]oxadiazol-3-yl...)
Affinity DataEC50:  320nMAssay Description:Agonist activity at human PPARalpha expressed in african green monkey CV1 cells co-transfected with Gal4 assessed as reporter activity by transient t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50103940(3-(4-((5-(3,5-bis(trifluoromethyl)phenyl)-1,2,4-ox...)
Affinity DataEC50:  320nMAssay Description:Agonist activity at human PPARdelta expressed in african green monkey CV1 cells co-transfected with Gal4 assessed as reporter activity by transient t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50103945(2-Isopropoxy-3-(4-{2-[5-(2-trifluoromethyl-phenyl)...)
Affinity DataEC50:  400nMAssay Description:Agonist activity at human PPARalpha expressed in african green monkey CV1 cells co-transfected with Gal4 assessed as reporter activity by transient t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50103944(3-(4-(2-(5-(4-chlorophenyl)-1,2,4-oxadiazol-3-yl)e...)
Affinity DataEC50:  400nMAssay Description:Agonist activity at human PPARalpha expressed in african green monkey CV1 cells co-transfected with Gal4 assessed as reporter activity by transient t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50103943(3-{4-[5-(4-Chloro-phenyl)-[1,2,4]oxadiazol-3-ylmet...)
Affinity DataEC50:  500nMAssay Description:Agonist activity at human PPARdelta expressed in african green monkey CV1 cells co-transfected with Gal4 assessed as reporter activity by transient t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50103949(2-Isopropoxy-3-{4-[5-(4-trifluoromethyl-phenyl)-[1...)
Affinity DataEC50:  500nMAssay Description:Agonist activity at human PPARdelta expressed in african green monkey CV1 cells co-transfected with Gal4 assessed as reporter activity by transient t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50103941(2-isopropoxy-3-(4-(2-(5-(3-(trifluoromethyl)phenyl...)
Affinity DataEC50:  500nMAssay Description:Agonist activity at human PPARdelta expressed in african green monkey CV1 cells co-transfected with Gal4 assessed as reporter activity by transient t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
National Institute of Pharmaceutical Education and Research

Curated by ChEMBL
LigandPNGBDBM50103960(3-(4-(2-(5-(3-fluorophenyl)-1,2,4-oxadiazol-3-yl)e...)
Affinity DataEC50:  500nMAssay Description:Agonist activity at human PPARalpha expressed in african green monkey CV1 cells co-transfected with Gal4 assessed as reporter activity by transient t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
Displayed 1 to 50 (of 64 total ) | Next | Last >>
Jump to: