Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 50038414
TargetSerine/threonine-protein kinase Chk1(Human)
Blaise Pascal University

Curated by ChEMBL
LigandPNGBDBM50220067(11H-2,5,11-triaza-benzo[a]trindene-1,3,4,6-tetraon...)
Affinity DataIC50: 20nMAssay Description:Inhibition of human Chk1More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Chk1(Human)
Blaise Pascal University

Curated by ChEMBL
LigandPNGBDBM50376170(CHEMBL265446)
Affinity DataIC50: 24nMAssay Description:Inhibition of human Chk1More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Chk1(Human)
Blaise Pascal University

Curated by ChEMBL
LigandPNGBDBM50236805(4,5-dihydro-11H-2,5,11-triaza-benzo[a]trindene-1,3...)
Affinity DataIC50: 51nMAssay Description:Inhibition of human Chk1More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Chk1(Human)
Blaise Pascal University

Curated by ChEMBL
LigandPNGBDBM50216165(1,11-dihydro-1,3,5,11-tetraaza-benzo[a]trindene-4,...)
Affinity DataIC50: 81nMAssay Description:Inhibition of human Chk1More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Chk1(Human)
Blaise Pascal University

Curated by ChEMBL
LigandPNGBDBM50216157(11H-2,5,11,11b-Tetraaza-benzo[a]trindene-4,6-dione...)
Affinity DataIC50: 100nMAssay Description:Inhibition of human Chk1More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Chk1(Human)
Blaise Pascal University

Curated by ChEMBL
LigandPNGBDBM50220074(benzo[a]pyrrolo[3,4-c]carbazole-1,3,4,7(2H,8H)-tet...)
Affinity DataIC50: 269nMAssay Description:Inhibition of human Chk1More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Chk1(Human)
Blaise Pascal University

Curated by ChEMBL
LigandPNGBDBM50220068(4,7-dihydroxybenzo[a]pyrrolo[3,4-c]carbazole-1,3(2...)
Affinity DataIC50: 311nMAssay Description:Inhibition of human Chk1More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Chk1(Human)
Blaise Pascal University

Curated by ChEMBL
LigandPNGBDBM50376169(CHEMBL259432)
Affinity DataIC50: 1.92E+3nMAssay Description:Inhibition of human Chk1More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Chk1(Human)
Blaise Pascal University

Curated by ChEMBL
LigandPNGBDBM50376171(CHEMBL265691)
Affinity DataIC50: 1.45E+4nMAssay Description:Inhibition of human Chk1More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed