Compile Data Set for Download or QSAR
Report error Found 44 Enz. Inhib. hit(s) with all data for entry = 50038326
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50374938(CHEMBL402163)
Affinity DataIC50: 0.210nMAssay Description:Inhibition of human recombinant DPP4 expressed in insect cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50374941(CHEMBL445674)
Affinity DataIC50: 3.20nMAssay Description:Inhibition of human recombinant DPP4 expressed in insect cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50237207((2S)-3-(3-(2-chloro-4-(methylsulfonyl)phenyl)-1,2,...)
Affinity DataIC50: 7.5nMAssay Description:Inhibition of human recombinant DPP4 expressed in insect cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50374939(CHEMBL404079)
Affinity DataIC50: 12nMAssay Description:Inhibition of human recombinant DPP4 expressed in insect cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM11676((2S,3S)-3-[3-(2-chloro-4-methanesulfonylphenyl)-1,...)
Affinity DataIC50: 13nMAssay Description:Inhibition of human recombinant DPP4 expressed in insect cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM11666((2S,3S)-2-amino-3-[3-(2-chloro-4-methanesulfonylph...)
Affinity DataIC50: 17nMAssay Description:Inhibition of human recombinant DPP4 expressed in insect cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM11681((2S,3S)-4-cyclopropyl-3-[3-(2-fluoro-4-methanesulf...)
Affinity DataIC50: 19nMAssay Description:Inhibition of human recombinant DPP4 expressed in insect cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50374942(CHEMBL1162974)
Affinity DataIC50: 21nMAssay Description:Inhibition of human recombinant DPP4 expressed in insect cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM11675(oxadiazole based amide | (2S,3S)-3-[3-(2-chloro-4-...)
Affinity DataIC50: 40nMAssay Description:Inhibition of human recombinant DPP4 expressed in insect cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50374943(CHEMBL429757)
Affinity DataIC50: 50nMAssay Description:Inhibition of human recombinant DPP4 expressed in insect cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50374944(CHEMBL256172)
Affinity DataIC50: 57nMAssay Description:Inhibition of human recombinant DPP4 expressed in insect cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM11678((2S,3S)-3-[3-(2-chloro-4-methanesulfonylphenyl)-1,...)
Affinity DataIC50: 70nMAssay Description:Inhibition of human recombinant DPP4 expressed in insect cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50374946(CHEMBL257709)
Affinity DataIC50: 90nMAssay Description:Inhibition of human recombinant DPP4 expressed in insect cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50374940(CHEMBL255591)
Affinity DataIC50: 93nMAssay Description:Inhibition of human recombinant DPP4 expressed in insect cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM11658((2S,3S)-2-amino-3-[3-(4-methanesulfonylphenyl)-1,2...)
Affinity DataIC50: 122nMAssay Description:Inhibition of human recombinant DPP4 expressed in insect cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50374938(CHEMBL402163)
Affinity DataIC50: 130nMAssay Description:Inhibition of human recombinant QPP expressed in baculovirus systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50374947(CHEMBL256603)
Affinity DataIC50: 140nMAssay Description:Inhibition of human recombinant QPP expressed in baculovirus systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM11662((2S,3S)-2-amino-3-[3-(2,4-dichlorophenyl)-1,2,4-ox...)
Affinity DataIC50: 203nMAssay Description:Inhibition of human recombinant DPP4 expressed in insect cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50374939(CHEMBL404079)
Affinity DataIC50: 210nMAssay Description:Inhibition of human recombinant QPP expressed in baculovirus systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50374949(CHEMBL437026)
Affinity DataIC50: 250nMAssay Description:Inhibition of human recombinant QPP expressed in baculovirus systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50374944(CHEMBL256172)
Affinity DataIC50: 330nMAssay Description:Inhibition of human recombinant QPP expressed in baculovirus systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50237207((2S)-3-(3-(2-chloro-4-(methylsulfonyl)phenyl)-1,2,...)
Affinity DataIC50: 330nMAssay Description:Inhibition of human recombinant QPP expressed in baculovirus systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50374943(CHEMBL429757)
Affinity DataIC50: 420nMAssay Description:Inhibition of human recombinant QPP expressed in baculovirus systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50374942(CHEMBL1162974)
Affinity DataIC50: 460nMAssay Description:Inhibition of human recombinant QPP expressed in baculovirus systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50374948(CHEMBL255351)
Affinity DataIC50: 525nMAssay Description:Inhibition of human recombinant DPP4 expressed in insect cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50374947(CHEMBL256603)
Affinity DataIC50: 645nMAssay Description:Inhibition of human recombinant DPP4 expressed in insect cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50374941(CHEMBL445674)
Affinity DataIC50: 1.16E+3nMAssay Description:Inhibition of human recombinant QPP expressed in baculovirus systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50374949(CHEMBL437026)
Affinity DataIC50: 1.17E+3nMAssay Description:Inhibition of human recombinant DPP4 expressed in insect cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM11662((2S,3S)-2-amino-3-[3-(2,4-dichlorophenyl)-1,2,4-ox...)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of human recombinant QPP expressed in baculovirus systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50374940(CHEMBL255591)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of human recombinant QPP expressed in baculovirus systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50374945(CHEMBL401932)
Affinity DataIC50: 1.49E+3nMAssay Description:Inhibition of human recombinant DPP4 expressed in insect cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50374948(CHEMBL255351)
Affinity DataIC50: 1.66E+3nMAssay Description:Inhibition of human recombinant QPP expressed in baculovirus systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50374945(CHEMBL401932)
Affinity DataIC50: 3.44E+3nMAssay Description:Inhibition of human recombinant QPP expressed in baculovirus systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM11675(oxadiazole based amide | (2S,3S)-3-[3-(2-chloro-4-...)
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of human recombinant QPP expressed in baculovirus systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50374946(CHEMBL257709)
Affinity DataIC50: 3.91E+3nMAssay Description:Inhibition of human recombinant QPP expressed in baculovirus systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM11666((2S,3S)-2-amino-3-[3-(2-chloro-4-methanesulfonylph...)
Affinity DataIC50: 6.40E+3nMAssay Description:Inhibition of human recombinant QPP expressed in baculovirus systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
LigandPNGBDBM50374938(CHEMBL402163)
Affinity DataIC50: 7.10E+3nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM11658((2S,3S)-2-amino-3-[3-(4-methanesulfonylphenyl)-1,2...)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of human recombinant QPP expressed in baculovirus systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM11676((2S,3S)-3-[3-(2-chloro-4-methanesulfonylphenyl)-1,...)
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibition of human recombinant QPP expressed in baculovirus systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM11681((2S,3S)-4-cyclopropyl-3-[3-(2-fluoro-4-methanesulf...)
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of human recombinant QPP expressed in baculovirus systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
LigandPNGBDBM50237207((2S)-3-(3-(2-chloro-4-(methylsulfonyl)phenyl)-1,2,...)
Affinity DataIC50: 1.90E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
LigandPNGBDBM11666((2S,3S)-2-amino-3-[3-(2-chloro-4-methanesulfonylph...)
Affinity DataIC50: 3.70E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM11678((2S,3S)-3-[3-(2-chloro-4-methanesulfonylphenyl)-1,...)
Affinity DataIC50: 4.50E+4nMAssay Description:Inhibition of human recombinant QPP expressed in baculovirus systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
LigandPNGBDBM50374941(CHEMBL445674)
Affinity DataIC50: 4.70E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed