Compile Data Set for Download or QSAR
Report error Found 33 Enz. Inhib. hit(s) with all data for entry = 5541
TargetCannabinoid receptor 1(Human)
F. Hoffmann-La Roche

Curated by PDSP Ki Database
LigandPNGBDBM86998(CAS_22475030 | NSC_22475030 | (2,2-bis(2,4-difluor...)
In Depth
Date in BDB:
6/12/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
F. Hoffmann-La Roche

Curated by PDSP Ki Database
LigandPNGBDBM87007(CAS_10391336 | NSC_10391336 | (2-(2,4-dichlorophen...)
In Depth
Date in BDB:
6/12/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
F. Hoffmann-La Roche

Curated by PDSP Ki Database
LigandPNGBDBM86984(CAS_24828562 | NSC_24828563 | CAS_24828563 | [2-(2...)
In Depth
Date in BDB:
6/12/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
F. Hoffmann-La Roche

Curated by PDSP Ki Database
LigandPNGBDBM86989(CAS_22475232 | NSC_22475232 | 1-(2,2-bis(2,4-diflu...)
In Depth
Date in BDB:
6/12/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
F. Hoffmann-La Roche

Curated by PDSP Ki Database
LigandPNGBDBM86984(CAS_24828562 | NSC_24828563 | CAS_24828563 | [2-(2...)
Affinity DataKi:  3.30nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
F. Hoffmann-La Roche

Curated by PDSP Ki Database
LigandPNGBDBM86984(CAS_24828562 | NSC_24828563 | CAS_24828563 | [2-(2...)
In Depth
Date in BDB:
6/12/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
F. Hoffmann-La Roche

Curated by PDSP Ki Database
LigandPNGBDBM86995(CAS_24828287 | NSC_24828287 | (2-(2,4-dichlorophen...)
In Depth
Date in BDB:
6/12/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
F. Hoffmann-La Roche

Curated by PDSP Ki Database
LigandPNGBDBM87003(CAS_10254993 | NSC_10254993 | (2-(2,4-dichlorophen...)
In Depth
Date in BDB:
6/12/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
F. Hoffmann-La Roche

Curated by PDSP Ki Database
LigandPNGBDBM21278(SR141716 | 5-(4-chlorophenyl)-1-(2,4-dichloropheny...)
In Depth
Date in BDB:
6/12/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
F. Hoffmann-La Roche

Curated by PDSP Ki Database
LigandPNGBDBM86997(NSC_22475102 | CAS_22475102 | (6-fluoro-2,2-bis(4-...)
In Depth
Date in BDB:
6/12/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
F. Hoffmann-La Roche

Curated by PDSP Ki Database
LigandPNGBDBM86992(NSC_22475130 | CAS_22475130 | (2,2-bis(2,4-difluor...)
In Depth
Date in BDB:
6/12/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
F. Hoffmann-La Roche

Curated by PDSP Ki Database
LigandPNGBDBM29094(3-(4-chlorophenyl)-N''''-(4-chlorophenylsulfonyl)-...)
In Depth
Date in BDB:
6/12/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
F. Hoffmann-La Roche

Curated by PDSP Ki Database
LigandPNGBDBM87009(NSC_22475238 | CAS_22475238 | 4-(2-(2,4-dichloroph...)
In Depth
Date in BDB:
6/12/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
F. Hoffmann-La Roche

Curated by PDSP Ki Database
LigandPNGBDBM86986(NSC_10024106 | CAS_10024106 | (6-fluoro-2,2-diphen...)
Affinity DataKi:  11nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
F. Hoffmann-La Roche

Curated by PDSP Ki Database
LigandPNGBDBM86999(CAS_24828561 | NSC_24828561 | (2,2-diphenyl-[1,3]d...)
Affinity DataKi:  13nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
F. Hoffmann-La Roche

Curated by PDSP Ki Database
LigandPNGBDBM87000(CAS_10097960 | NSC_10097960 | 1-(2,2-diphenyl-benz...)
Affinity DataKi:  13nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
F. Hoffmann-La Roche

Curated by PDSP Ki Database
LigandPNGBDBM86993(CAS_10024236 | NSC_10024236 | (6-fluoro-2,2-diphen...)
Affinity DataKi:  15nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
F. Hoffmann-La Roche

Curated by PDSP Ki Database
LigandPNGBDBM87006(CAS_22475173 | NSC_22475173 | (6-fluoro-2,2-bis(4-...)
Affinity DataKi:  18nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
F. Hoffmann-La Roche

Curated by PDSP Ki Database
LigandPNGBDBM87012(NSC_22475055 | CAS_22475055 | 4-(2,2-bis(2,4-diflu...)
Affinity DataKi:  25nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
F. Hoffmann-La Roche

Curated by PDSP Ki Database
LigandPNGBDBM86991(CAS_10045631 | NSC_10045631 | (2,2-diphenylbenzo[d...)
Affinity DataKi:  28nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
F. Hoffmann-La Roche

Curated by PDSP Ki Database
LigandPNGBDBM87001(CAS_22475058 | NSC_22475058 | (2-(2,4-dichlorophen...)
Affinity DataKi:  30nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
F. Hoffmann-La Roche

Curated by PDSP Ki Database
LigandPNGBDBM86984(CAS_24828562 | NSC_24828563 | CAS_24828563 | [2-(2...)
Affinity DataKi:  35nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
F. Hoffmann-La Roche

Curated by PDSP Ki Database
LigandPNGBDBM87004(NSC_10342137 | CAS_10342137 | 1-(2,2-diphenyl-benz...)
Affinity DataKi:  38nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
F. Hoffmann-La Roche

Curated by PDSP Ki Database
LigandPNGBDBM87011(CAS_44450433 | NSC_44450433 | (S)-(2,2-bis(2,4-dif...)
Affinity DataKi:  46nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
F. Hoffmann-La Roche

Curated by PDSP Ki Database
LigandPNGBDBM87008(NSC_10452791 | CAS_10452791 | (2,2-diphenylbenzo[d...)
Affinity DataKi:  50nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
F. Hoffmann-La Roche

Curated by PDSP Ki Database
LigandPNGBDBM87005(CAS_44450450 | NSC_44450450 | (6-(methylsulfonyl)-...)
Affinity DataKi:  110nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
F. Hoffmann-La Roche

Curated by PDSP Ki Database
LigandPNGBDBM86988(NSC_22475064 | CAS_22475064 | (6-chloro-2,2-diphen...)
Affinity DataKi:  216nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
F. Hoffmann-La Roche

Curated by PDSP Ki Database
LigandPNGBDBM86990(NSC_22475161 | CAS_22475161 | 6-(morpholine-4-carb...)
Affinity DataKi:  277nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
F. Hoffmann-La Roche

Curated by PDSP Ki Database
LigandPNGBDBM86994(CAS_24828424 | NSC_24828424 | (6-methyl-2,2-diphen...)
Affinity DataKi:  509nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
F. Hoffmann-La Roche

Curated by PDSP Ki Database
LigandPNGBDBM86985(NSC_22475120 | CAS_22475120 | (6-bromo-2,2-dipheny...)
Affinity DataKi:  873nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
F. Hoffmann-La Roche

Curated by PDSP Ki Database
LigandPNGBDBM86996(CAS_24828288 | NSC_24828288 | 4-[6-fluoro-2,2-bis-...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
F. Hoffmann-La Roche

Curated by PDSP Ki Database
LigandPNGBDBM87010(CAS_44450451 | NSC_44450451 | 1-(4-(4-chlorophenyl...)
Affinity DataKi:  1.50E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
F. Hoffmann-La Roche

Curated by PDSP Ki Database
LigandPNGBDBM87000(CAS_10097960 | NSC_10097960 | 1-(2,2-diphenyl-benz...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2012
Entry Details Article
PubMed