Compile Data Set for Download or QSAR
Report error Found 55 Enz. Inhib. hit(s) with all data for entry = 50038572
TargetCannabinoid receptor 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50260753((S)-N-(1-amino-3,3-dimethyl-1-oxobutan-2-yl)-3-(3-...)
Affinity DataEC50:  2nMAssay Description:Agonist activity at human CB2 receptor assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50261053(1-(2-morpholinoethyl)-N-(naphthalen-1-yl)-2-oxo-1,...)
Affinity DataEC50:  22nMAssay Description:Agonist activity at human CB2 receptor assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50261052((R)-3-(2-morpholinoethyl)-2-oxo-N-(1,2,3,4-tetrahy...)
Affinity DataEC50:  0.700nMAssay Description:Agonist activity at human CB2 receptor assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50261051(3-(2-morpholinoethyl)-N-(naphthalen-1-yl)-2-oxo-2,...)
Affinity DataEC50:  8nMAssay Description:Agonist activity at human CB2 receptor assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50261101(N-cyclohexyl-N-methyl-3-(2-morpholinoethyl)-2-oxo-...)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50260671((S)-N-(1-amino-1-oxo-3-phenylpropan-2-yl)-3-(2-mor...)
Affinity DataIC50: 2.50E+3nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50260629((S)-N-(2-amino-2-oxo-1-phenylethyl)-3-(2-morpholin...)
Affinity DataIC50: 2.50E+3nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50260672((S)-N-(1-cyano-2,2-dimethylpropyl)-3-(2-morpholino...)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [3H]SR141716A from human CB1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50260752((S)-N-(1-amino-3,3-dimethyl-1-oxobutan-2-yl)-3-(2-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [3H]SR141716A from human CB1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50260751((S)-N-(1-amino-3,3-dimethyl-1-oxobutan-2-yl)-3-(2-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [3H]SR141716A from human CB1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50260674((S)-N-(2,2-dimethyl-1-(3-methyl-1,2,4-oxadiazol-5-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [3H]SR141716A from human CB1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50261102(N-(1-(4-fluorophenyl)ethyl)-3-(2-morpholinoethyl)-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [3H]SR141716A from human CB1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50260627((S)-N-(1-amino-3,3-dimethyl-1-oxobutan-2-yl)-3-(2-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [3H]SR141716A from human CB1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50261100(N-cyclohexyl-3-(2-morpholinoethyl)-2-oxo-2,3-dihyd...)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [3H]SR141716A from human CB1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50260538((S)-N-(1-(dimethylamino)-3,3-dimethyl-1-oxobutan-2...)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [3H]SR141716A from human CB1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50260514((S)-N-(1-hydroxy-3,3-dimethylbutan-2-yl)-3-(2-morp...)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [3H]SR141716A from human CB1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50260513(N-((1S,2S)-2-hydroxycyclohexyl)-3-(2-morpholinoeth...)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [3H]SR141716A from human CB1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50260512(N-(2-hydroxy-1,2,3,4-tetrahydronaphthalen-1-yl)-3-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [3H]SR141716A from human CB1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50260712((S)-N-(1-amino-3,3-dimethyl-1-oxobutan-2-yl)-3-iso...)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50377918(CHEMBL1162994)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50260627((S)-N-(1-amino-3,3-dimethyl-1-oxobutan-2-yl)-3-(2-...)
Affinity DataKi:  5nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50260672((S)-N-(1-cyano-2,2-dimethylpropyl)-3-(2-morpholino...)
Affinity DataKi:  5nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50260673((S)-N-(2,2-dimethyl-1-(2-methyl-2H-tetrazol-5-yl)p...)
Affinity DataKi:  5nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50260709(N-((S)-1-amino-3,3-dimethyl-1-oxobutan-2-yl)-2-oxo...)
Affinity DataKi:  6nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50261052((R)-3-(2-morpholinoethyl)-2-oxo-N-(1,2,3,4-tetrahy...)
Affinity DataKi:  7nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50261051(3-(2-morpholinoethyl)-N-(naphthalen-1-yl)-2-oxo-2,...)
Affinity DataKi:  8nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50260753((S)-N-(1-amino-3,3-dimethyl-1-oxobutan-2-yl)-3-(3-...)
Affinity DataKi:  8nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50261099((R)-1-(2-morpholinoethyl)-2-oxo-N-(1,2,3,4-tetrahy...)
Affinity DataKi:  9nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50260674((S)-N-(2,2-dimethyl-1-(3-methyl-1,2,4-oxadiazol-5-...)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50260514((S)-N-(1-hydroxy-3,3-dimethylbutan-2-yl)-3-(2-morp...)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50260626((S)-N'-(3,3-dimethyl-1-(methylamino)-1-oxobutan-2-...)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50260538((S)-N-(1-(dimethylamino)-3,3-dimethyl-1-oxobutan-2...)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50261053(1-(2-morpholinoethyl)-N-(naphthalen-1-yl)-2-oxo-1,...)
Affinity DataKi:  41nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50260512(N-(2-hydroxy-1,2,3,4-tetrahydronaphthalen-1-yl)-3-...)
Affinity DataKi:  51nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50261100(N-cyclohexyl-3-(2-morpholinoethyl)-2-oxo-2,3-dihyd...)
Affinity DataKi:  60nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50260628(N-((2S,3S)-1-amino-3-methyl-1-oxopentan-2-yl)-3-(2...)
Affinity DataKi:  67nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50260712((S)-N-(1-amino-3,3-dimethyl-1-oxobutan-2-yl)-3-iso...)
Affinity DataKi:  69nMAssay Description:Displacement of [3H]SR141716A from human CB1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50260511(N-(chroman-4-yl)-3-(2-morpholinoethyl)-2-oxo-2,3-d...)
Affinity DataKi:  74nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50260750((S)-N-(1-amino-3,3-dimethyl-1-oxobutan-2-yl)-3-((4...)
Affinity DataKi:  92nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50260751((S)-N-(1-amino-3,3-dimethyl-1-oxobutan-2-yl)-3-(2-...)
Affinity DataKi:  144nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50260752((S)-N-(1-amino-3,3-dimethyl-1-oxobutan-2-yl)-3-(2-...)
Affinity DataKi:  196nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50261102(N-(1-(4-fluorophenyl)ethyl)-3-(2-morpholinoethyl)-...)
Affinity DataKi:  232nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50260710((S)-N-(1-amino-3,3-dimethyl-1-oxobutan-2-yl)-2-oxo...)
Affinity DataKi:  242nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50260711((S)-N-(1-amino-3,3-dimethyl-1-oxobutan-2-yl)-3-(2-...)
Affinity DataKi:  338nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50260513(N-((1S,2S)-2-hydroxycyclohexyl)-3-(2-morpholinoeth...)
Affinity DataKi:  484nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50260709(N-((S)-1-amino-3,3-dimethyl-1-oxobutan-2-yl)-2-oxo...)
Affinity DataKi:  1.32E+3nMAssay Description:Displacement of [3H]SR141716A from human CB1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50260753((S)-N-(1-amino-3,3-dimethyl-1-oxobutan-2-yl)-3-(3-...)
Affinity DataKi:  1.46E+3nMAssay Description:Displacement of [3H]SR141716A from human CB1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50377918(CHEMBL1162994)
Affinity DataKi:  1.47E+3nMAssay Description:Displacement of [3H]SR141716A from human CB1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50260673((S)-N-(2,2-dimethyl-1-(2-methyl-2H-tetrazol-5-yl)p...)
Affinity DataKi:  1.48E+3nMAssay Description:Displacement of [3H]SR141716A from human CB1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50261099((R)-1-(2-morpholinoethyl)-2-oxo-N-(1,2,3,4-tetrahy...)
Affinity DataKi:  1.51E+3nMAssay Description:Displacement of [3H]SR141716A from human CB1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
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