Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 50000706
TargetKappa-type opioid receptor(Guinea pig)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50007355(2-(3,4-Dichloro-phenyl)-N-methyl-N-((S)-2-methyl-1...)
Affinity DataIC50: 6.30nMAssay Description:Compound was evaluated for the Opioid receptor kappa 1 affinity using guinea pig brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50007344(2-(3,4-Dichloro-phenyl)-N-methyl-N-(1-phenyl-2-pyr...)
Affinity DataIC50: 6.90nMAssay Description:Compound was evaluated for the Opioid receptor kappa 1 affinity using guinea pig brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50008845(CHEMBL55543 | 2-(3,4-Dichloro-phenyl)-N-(2,2-dimet...)
Affinity DataIC50: 24nMAssay Description:Compound was evaluated for the opioid receptor kappa affinity using guinea pig brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50007361(CHEMBL56651 | 2-(3,4-Dichloro-phenyl)-N-methyl-N-(...)
Affinity DataIC50: 53nMAssay Description:Compound was evaluated for the Opioid receptor kappa 1 affinity using guinea pig brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50008843(CHEMBL55603 | 2-(3,4-Dichloro-phenyl)-N-methyl-N-(...)
Affinity DataIC50: 85nMAssay Description:Compound was evaluated for the opioid receptor kappa affinity using guinea pig brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50000296(CHEMBL441765 | CHEMBL482811 | U-50488H | US1149237...)
Affinity DataIC50: 96nMAssay Description:Compound was evaluated for the opioid receptor kappa affinity using guinea pig brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50008847(CHEMBL293973 | 2-(3,4-Dichloro-phenyl)-N-methyl-N-...)
Affinity DataIC50: 1.54E+3nMAssay Description:Compound was evaluated for the opioid receptor kappa affinity using guinea pig brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50008846(CHEMBL299068 | 2-(3,4-Dichloro-phenyl)-N-(1,1-dime...)
Affinity DataIC50: 2.06E+3nMAssay Description:Compound was evaluated for the opioid receptor kappa affinity using guinea pig brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50000092(Analog of 14-(Arylhydroxyamino)codeinone | 4-methy...)
Affinity DataIC50: 2.39E+3nMAssay Description:Compound was evaluated for the opioid receptor kappa affinity using guinea pig brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50008844(CHEMBL55020 | 2-(3,4-Dichloro-phenyl)-N-methyl-N-(...)
Affinity DataIC50: 3.41E+3nMAssay Description:Compound was evaluated for the opioid receptor kappa affinity using guinea pig brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50008850(CHEMBL56744 | 2-(3,4-Dichloro-phenyl)-N-methyl-N-(...)
Affinity DataIC50: 6.12E+3nMAssay Description:Compound was evaluated for the opioid receptor kappa affinity using guinea pig brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50008849(CHEMBL54451 | 2-(3,4-Dichloro-phenyl)-N-methyl-N-(...)
Affinity DataIC50: 1.00E+4nMAssay Description:Compound was evaluated for the opioid receptor kappa affinity using guinea pig brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed