Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 50000718
TargetMu-type opioid receptor(Guinea pig)
Anaquest

Curated by ChEMBL
LigandPNGBDBM50008984(N-(1-Phenethyl-piperidin-4-yl)-N-phenyl-propionami...)
Affinity DataIC50: 3.10nMAssay Description:In vitro binding activity against opioid receptor mu using [3H]-DAGO as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetMu-type opioid receptor(Guinea pig)
Anaquest

Curated by ChEMBL
LigandPNGBDBM50008980(CHEMBL169366 | 4-(Phenyl-propionyl-amino)-1-(2-pyr...)
Affinity DataIC50: 5.40nMAssay Description:In vitro binding activity against opioid receptor mu using [3H]DAGO) as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Anaquest

Curated by ChEMBL
LigandPNGBDBM50008982(CHEMBL168723 | N-[4-Methoxymethyl-1-(2-pyrazol-1-y...)
Affinity DataIC50: 10nMAssay Description:In vitro binding activity against opioid receptor mu using [3H]DAGO) as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Anaquest

Curated by ChEMBL
LigandPNGBDBM83450(N-[1-[2-(4-ethyl-5-oxidanylidene-1,2,3,4-tetrazol-...)
Affinity DataIC50: 15nMAssay Description:In vitro binding activity against opioid receptor mu using [3H]DAGO) as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Anaquest

Curated by ChEMBL
LigandPNGBDBM50008984(N-(1-Phenethyl-piperidin-4-yl)-N-phenyl-propionami...)
Affinity DataIC50: 187nMAssay Description:In vitro binding activity against opioid receptor delta using [3DPDPE] as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Anaquest

Curated by ChEMBL
LigandPNGBDBM50008980(CHEMBL169366 | 4-(Phenyl-propionyl-amino)-1-(2-pyr...)
Affinity DataIC50: 809nMAssay Description:In vitro binding activity against opioid receptor delta using [3H]DPDPE) as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Anaquest

Curated by ChEMBL
LigandPNGBDBM50008983(CHEMBL424400 | 1-[2-(1,3-Dioxo-1,3-dihydro-isoindo...)
Affinity DataIC50: 1.20E+3nMAssay Description:In vitro binding activity against opioid receptor mu using [3H]DAGO) as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Anaquest

Curated by ChEMBL
LigandPNGBDBM50008981(CHEMBL169587 | N-{1-[2-(1,3-Dioxo-1,3-dihydro-isoi...)
Affinity DataIC50: 1.60E+3nMAssay Description:In vitro binding activity against opioid receptor mu using [3H]DAGO) as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Anaquest

Curated by ChEMBL
LigandPNGBDBM50008982(CHEMBL168723 | N-[4-Methoxymethyl-1-(2-pyrazol-1-y...)
Affinity DataIC50: 1.70E+3nMAssay Description:In vitro binding activity against opioid receptor delta using [3H]DPDPE) as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Anaquest

Curated by ChEMBL
LigandPNGBDBM50008984(N-(1-Phenethyl-piperidin-4-yl)-N-phenyl-propionami...)
Affinity DataIC50: 5.89E+3nMAssay Description:In vitro binding activity against opioid receptor kappa using [3H]EKC as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Anaquest

Curated by ChEMBL
LigandPNGBDBM50008983(CHEMBL424400 | 1-[2-(1,3-Dioxo-1,3-dihydro-isoindo...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro binding activity against opioid receptor kappa using [3H]EKC as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Anaquest

Curated by ChEMBL
LigandPNGBDBM50008981(CHEMBL169587 | N-{1-[2-(1,3-Dioxo-1,3-dihydro-isoi...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro binding activity against opioid receptor kappa using [3H]EKC as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Anaquest

Curated by ChEMBL
LigandPNGBDBM83450(N-[1-[2-(4-ethyl-5-oxidanylidene-1,2,3,4-tetrazol-...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro binding activity against opioid receptor kappa using [3H]EKC as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed