Compile Data Set for Download or QSAR
Report error Found 25 Enz. Inhib. hit(s) with all data for entry = 50004008
TargetEpidermal growth factor receptor(Human)
The University of Tokushima

Curated by ChEMBL
LigandPNGBDBM50478728(TX-2036 | CHEMBL490266)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of human A431 cell EGFRK assessed as 32P phosphorylation by scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
The University of Tokushima

Curated by ChEMBL
LigandPNGBDBM50478724(CHEMBL484119)
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of human A431 cell EGFRK assessed as 32P phosphorylation by scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 1(Human)
The University of Tokushima

Curated by ChEMBL
LigandPNGBDBM50478728(TX-2036 | CHEMBL490266)
Affinity DataIC50: 1.84E+4nMAssay Description:Inhibition of Flt1 expressed in mouse NIH3T3 cells by autoradiographyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
The University of Tokushima

Curated by ChEMBL
LigandPNGBDBM50478727(TX-2037 | CHEMBL490267)
Affinity DataIC50: 1.84E+4nMAssay Description:Inhibition of human A431 cell EGFRK assessed as 32P phosphorylation by scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 1(Human)
The University of Tokushima

Curated by ChEMBL
LigandPNGBDBM50478730(TX-2030 | CHEMBL484121)
Affinity DataIC50: 2.13E+4nMAssay Description:Inhibition of Flt1 expressed in mouse NIH3T3 cells by autoradiographyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
The University of Tokushima

Curated by ChEMBL
LigandPNGBDBM50478730(TX-2030 | CHEMBL484121)
Affinity DataIC50: 2.13E+4nMAssay Description:Inhibition of human A431 cell EGFRK assessed as 32P phosphorylation by scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
The University of Tokushima

Curated by ChEMBL
LigandPNGBDBM50478731(TX-2044 | CHEMBL484316)
Affinity DataIC50: 2.30E+4nMAssay Description:Inhibition of human A431 cell EGFRK assessed as 32P phosphorylation by scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 1(Human)
The University of Tokushima

Curated by ChEMBL
LigandPNGBDBM50478724(CHEMBL484119)
Affinity DataIC50: 2.34E+4nMAssay Description:Inhibition of Flt1 expressed in mouse NIH3T3 cells by autoradiographyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
The University of Tokushima

Curated by ChEMBL
LigandPNGBDBM50478724(CHEMBL484119)
Affinity DataIC50: 2.40E+4nMAssay Description:Inhibition of human bowes melanoma cell MMP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
The University of Tokushima

Curated by ChEMBL
LigandPNGBDBM50478730(TX-2030 | CHEMBL484121)
Affinity DataIC50: 4.90E+4nMAssay Description:Inhibition of human bowes melanoma cell MMP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
The University of Tokushima

Curated by ChEMBL
LigandPNGBDBM50478729(TX-2031 | CHEMBL484321)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human bowes melanoma cell MMP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Bovine)
The University of Tokushima

Curated by ChEMBL
LigandPNGBDBM50478724(CHEMBL484119)
Affinity DataIC50: 5.30E+4nMAssay Description:Inhibition of bovine arterial endothelial cell MMP9More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Bovine)
The University of Tokushima

Curated by ChEMBL
LigandPNGBDBM50478728(TX-2036 | CHEMBL490266)
Affinity DataIC50: 6.70E+4nMAssay Description:Inhibition of bovine arterial endothelial cell MMP9More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
The University of Tokushima

Curated by ChEMBL
LigandPNGBDBM50478728(TX-2036 | CHEMBL490266)
Affinity DataIC50: 7.70E+4nMAssay Description:Inhibition of human bowes melanoma cell MMP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Bovine)
The University of Tokushima

Curated by ChEMBL
LigandPNGBDBM50478730(TX-2030 | CHEMBL484121)
Affinity DataIC50: 1.02E+5nMAssay Description:Inhibition of bovine arterial endothelial cell MMP9More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Bovine)
The University of Tokushima

Curated by ChEMBL
LigandPNGBDBM50478727(TX-2037 | CHEMBL490267)
Affinity DataIC50: 1.03E+5nMAssay Description:Inhibition of bovine arterial endothelial cell MMP9More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Bovine)
The University of Tokushima

Curated by ChEMBL
LigandPNGBDBM50478729(TX-2031 | CHEMBL484321)
Affinity DataIC50: 1.28E+5nMAssay Description:Inhibition of bovine arterial endothelial cell MMP9More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
The University of Tokushima

Curated by ChEMBL
LigandPNGBDBM50478727(TX-2037 | CHEMBL490267)
Affinity DataIC50: 1.83E+5nMAssay Description:Inhibition of human bowes melanoma cell MMP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 1(Human)
The University of Tokushima

Curated by ChEMBL
LigandPNGBDBM50478727(TX-2037 | CHEMBL490267)
Affinity DataIC50: 1.84E+5nMAssay Description:Inhibition of Flt1 expressed in mouse NIH3T3 cells by autoradiographyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
The University of Tokushima

Curated by ChEMBL
LigandPNGBDBM50478729(TX-2031 | CHEMBL484321)
Affinity DataIC50: 2.13E+5nMAssay Description:Inhibition of human A431 cell EGFRK assessed as 32P phosphorylation by scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 1(Human)
The University of Tokushima

Curated by ChEMBL
LigandPNGBDBM50478729(TX-2031 | CHEMBL484321)
Affinity DataIC50: 2.13E+5nMAssay Description:Inhibition of Flt1 expressed in mouse NIH3T3 cells by autoradiographyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Bovine)
The University of Tokushima

Curated by ChEMBL
LigandPNGBDBM50478726(TX-2045 | CHEMBL484123)
Affinity DataIC50: 2.40E+5nMAssay Description:Inhibition of bovine arterial endothelial cell MMP9More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Bovine)
The University of Tokushima

Curated by ChEMBL
LigandPNGBDBM50478725(TX-2046 | CHEMBL484302)
Affinity DataIC50: 2.40E+5nMAssay Description:Inhibition of bovine arterial endothelial cell MMP9More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
The University of Tokushima

Curated by ChEMBL
LigandPNGBDBM50478725(TX-2046 | CHEMBL484302)
Affinity DataIC50: 2.40E+5nMAssay Description:Inhibition of human bowes melanoma cell MMP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
The University of Tokushima

Curated by ChEMBL
LigandPNGBDBM50478726(TX-2045 | CHEMBL484123)
Affinity DataIC50: 2.40E+5nMAssay Description:Inhibition of human bowes melanoma cell MMP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed