Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50026273
TargetMitogen-activated protein kinase kinase kinase 5(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50243867(STS-PEG-TAMRA | CHEMBL478889)
Affinity DataKd:  8.00E+3nMAssay Description:Binding affinity to ASK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase 5(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50059889(3-methoxy-2-methyl-4-methylamino-(2S,3S,4S,6R)-29-...)
Affinity DataKd:  110nMAssay Description:Binding affinity to ASK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase 5(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50059889(3-methoxy-2-methyl-4-methylamino-(2S,3S,4S,6R)-29-...)
Affinity DataIC50: 37nMAssay Description:Inhibition of ASK1 by luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase 5(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM7491(4-[2-Amino-5-oxo-1,5-dihydro-imidazol-(4Z)-ylidene...)
Affinity DataIC50: 150nMAssay Description:Inhibition of ASK1 by luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase 5(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50059889(3-methoxy-2-methyl-4-methylamino-(2S,3S,4S,6R)-29-...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of ASK1 by fluorescence correlation spectroscopyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase 5(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM7491(4-[2-Amino-5-oxo-1,5-dihydro-imidazol-(4Z)-ylidene...)
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of ASK1 by fluorescence correlation spectroscopyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase 5(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50243715(3-((1-methyl-1H-indol-3-yl)methylene)indolin-2-one...)
Affinity DataIC50: 8.27E+4nMAssay Description:Inhibition of ASK1 by luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase 5(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50243715(3-((1-methyl-1H-indol-3-yl)methylene)indolin-2-one...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of ASK1 by fluorescence correlation spectroscopyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed