Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 50026276
TargetATP-dependent translocase ABCB1(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50197200(2-((2-(3-methoxyphenethyl)phenoxy)methyl)pyridine ...)
Affinity DataEC50:  2.76E+4nMAssay Description:Inhibition of P-glycoprotein-mediated [3H]vinblastine transport in human Caco-2 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetATP-dependent translocase ABCB1(Human)
Università

Curated by ChEMBL
LigandPNGBDBM20607((2-{4-[(1Z)-1,2-diphenylbut-1-en-1-yl]phenoxy}ethy...)
Affinity DataEC50:  5.65E+4nMAssay Description:Inhibition of P-glycoprotein-mediated [3H]vinblastine transport in human Caco-2 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetATP-dependent translocase ABCB1(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50022815((3S,6S,9S,12R,15S,18S,21S,24S,30S,33S)-30-ethyl-33...)
Affinity DataEC50:  4.55E+4nMAssay Description:Inhibition of P-glycoprotein-mediated [3H]vinblastine transport in human Caco-2 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetATP-dependent translocase ABCB1(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50338982((R)-5-((3,4-dimethoxyphenethyl)(methyl)amino)-2-(3...)
Affinity DataEC50:  2.00E+4nMAssay Description:Inhibition of P-glycoprotein-mediated [3H]vinblastine transport in human Caco-2 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed