Compile Data Set for Download or QSAR
Report error Found 36 Enz. Inhib. hit(s) with all data for entry = 50026283
TargetCannabinoid receptor 2(Human)
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50244360(6,6,9-Trimethyl-3-(1-methyl-1-thiophen-2-yl-ethyl)...)
Affinity DataKi:  0.270nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50244359(3-[1-(3-Bromo-phenyl)-1-methyl-ethyl]-6,6,9-trimet...)
Affinity DataKi:  0.540nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50244284((6aR,10aR)-3-(2-(4-ethylphenyl)propan-2-yl)-6,6,9-...)
Affinity DataKi:  0.670nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50244252(6,6,9-Trimethyl-3-(1-methyl-1-p-tolyl-ethyl)-6a,7,...)
Affinity DataKi:  0.880nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50244322(3-[1-(3-Fluoro-phenyl)-1-methyl-ethyl]-6,6,9-trime...)
Affinity DataKi:  0.900nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50243718(3-(2-((6aR,10aR)-1-hydroxy-6,6,9-trimethyl-6a,7,10...)
Affinity DataKi:  0.910nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50133546((6aR,10aR)-6,6,9-trimethyl-3-(2-phenylpropan-2-yl)...)
Affinity DataKi:  0.910nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50244360(6,6,9-Trimethyl-3-(1-methyl-1-thiophen-2-yl-ethyl)...)
Affinity DataKi:  1.08nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50244281((6aR,10aR)-6,6,9-trimethyl-3-(2-m-tolylpropan-2-yl...)
Affinity DataKi:  1.13nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50244358(3-[1-(4-Bromo-phenyl)-1-methyl-ethyl]-6,6,9-trimet...)
Affinity DataKi:  1.54nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50244359(3-[1-(3-Bromo-phenyl)-1-methyl-ethyl]-6,6,9-trimet...)
Affinity DataKi:  1.59nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50244323((6aR,10aR)-3-(2-(4-chlorophenyl)propan-2-yl)-6,6,9...)
Affinity DataKi:  1.68nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50244320((6aR,10aR)-6,6,9-trimethyl-3-(2-(4-propylphenyl)pr...)
Affinity DataKi:  1.77nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50244284((6aR,10aR)-3-(2-(4-ethylphenyl)propan-2-yl)-6,6,9-...)
Affinity DataKi:  1.85nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50244281((6aR,10aR)-6,6,9-trimethyl-3-(2-m-tolylpropan-2-yl...)
Affinity DataKi:  2.53nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50243717(4-(2-((6aR,10aR)-1-hydroxy-6,6,9-trimethyl-6a,7,10...)
Affinity DataKi:  2.53nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50243718(3-(2-((6aR,10aR)-1-hydroxy-6,6,9-trimethyl-6a,7,10...)
Affinity DataKi:  2.72nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50244357(3-[1-(3-Chloro-phenyl)-1-methyl-ethyl]-6,6,9-trime...)
Affinity DataKi:  2.80nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50244252(6,6,9-Trimethyl-3-(1-methyl-1-p-tolyl-ethyl)-6a,7,...)
Affinity DataKi:  3.13nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50244357(3-[1-(3-Chloro-phenyl)-1-methyl-ethyl]-6,6,9-trime...)
Affinity DataKi:  3.54nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50244358(3-[1-(4-Bromo-phenyl)-1-methyl-ethyl]-6,6,9-trimet...)
Affinity DataKi:  5.03nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50244322(3-[1-(3-Fluoro-phenyl)-1-methyl-ethyl]-6,6,9-trime...)
Affinity DataKi:  5.26nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50244283(3-[1-(3,5-Dimethyl-phenyl)-1-methyl-ethyl]-6,6,9-t...)
Affinity DataKi:  7.45nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50244320((6aR,10aR)-6,6,9-trimethyl-3-(2-(4-propylphenyl)pr...)
Affinity DataKi:  7.83nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50243717(4-(2-((6aR,10aR)-1-hydroxy-6,6,9-trimethyl-6a,7,10...)
Affinity DataKi:  9.25nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50244282((6aR,10aR)-6,6,9-trimethyl-3-(2-o-tolylpropan-2-yl...)
Affinity DataKi:  10.7nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50244283(3-[1-(3,5-Dimethyl-phenyl)-1-methyl-ethyl]-6,6,9-t...)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50133546((6aR,10aR)-6,6,9-trimethyl-3-(2-phenylpropan-2-yl)...)
Affinity DataKi:  12.3nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50244321((6aR,10aR)-3-(2-(4-fluorophenyl)propan-2-yl)-6,6,9...)
Affinity DataKi:  12.4nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50243719(N-{3-[1-(1-hydroxy-6,6,9-trimethyl)-6a,7,10,10atet...)
Affinity DataKi:  13.6nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50243719(N-{3-[1-(1-hydroxy-6,6,9-trimethyl)-6a,7,10,10atet...)
Affinity DataKi:  13.7nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50244323((6aR,10aR)-3-(2-(4-chlorophenyl)propan-2-yl)-6,6,9...)
Affinity DataKi:  18.8nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50067734(6,6,9-Trimethyl-3-pentyl-6a,7,10,10a-tetrahydro-6H...)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50067734(6,6,9-Trimethyl-3-pentyl-6a,7,10,10a-tetrahydro-6H...)
Affinity DataKi:  28.5nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50244282((6aR,10aR)-6,6,9-trimethyl-3-(2-o-tolylpropan-2-yl...)
Affinity DataKi:  34.4nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50244321((6aR,10aR)-3-(2-(4-fluorophenyl)propan-2-yl)-6,6,9...)
Affinity DataKi:  76.1nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed