Compile Data Set for Download or QSAR
Report error Found 40 Enz. Inhib. hit(s) with all data for entry = 50026350
TargetAcetylcholinesterase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50267151(10-N-Demethyl-10-N-(6-(4-(piperidin-1-ylmethyl)phe...)
Affinity DataIC50: 5.62nMAssay Description:Inhibition of AChE from rat cortex homogenate by Ellmans methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAcetylcholinesterase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50267150(10-N-Demethyl-10-N-(5-(4-(piperidin-1-ylmethyl)phe...)
Affinity DataIC50: 6.52nMAssay Description:Inhibition of AChE from rat cortex homogenate by Ellmans methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAcetylcholinesterase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50267157(10-N-Demethyl-10-N-(6-(4-((diethylamino)methyl)-ph...)
Affinity DataIC50: 8.86nMAssay Description:Inhibition of AChE from rat cortex homogenate by Ellmans methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAcetylcholinesterase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50267106(10-N-Demethyl-10-N-(4-(4-(piperidin-1-ylmethyl)phe...)
Affinity DataIC50: 12.4nMAssay Description:Inhibition of AChE from rat cortex homogenate by Ellmans methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAcetylcholinesterase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50267156(10-N-Demethyl-10-N-(4-(4-((diethylamino)methyl)-ph...)
Affinity DataIC50: 14.6nMAssay Description:Inhibition of AChE from rat cortex homogenate by Ellmans methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAcetylcholinesterase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50267105(10-N-Demethyl-10-N-(3-(4-(piperidin-1-ylmethyl)phe...)
Affinity DataIC50: 18nMAssay Description:Inhibition of AChE from rat cortex homogenate by Ellmans methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAcetylcholinesterase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50267104(10-N-Demethyl-10-N-(2-(4-(piperidin-1-ylmethyl)phe...)
Affinity DataIC50: 24.5nMAssay Description:Inhibition of AChE from rat cortex homogenate by Ellmans methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAcetylcholinesterase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50267152(10-N-Demethyl-10-N-(8-(4-(piperidin-1-ylmethyl)phe...)
Affinity DataIC50: 34.7nMAssay Description:Inhibition of AChE from rat cortex homogenate by Ellmans methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAcetylcholinesterase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50267190(10-N-Demethyl-10-N-(4-(4-(pyrrolidine-1-carbonyl)-...)
Affinity DataIC50: 53.8nMAssay Description:Inhibition of AChE from rat cortex homogenate by Ellmans methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAcetylcholinesterase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50267155(10-N-Demethyl-10-N-(12-(4-(piperidin-1-ylmethyl)-p...)
Affinity DataIC50: 58.1nMAssay Description:Inhibition of AChE from rat cortex homogenate by Ellmans methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAcetylcholinesterase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50267154(10-N-Demethyl-10-N-(10-(4-(piperidin-1-ylmethyl)-p...)
Affinity DataIC50: 61.2nMAssay Description:Inhibition of AChE from rat cortex homogenate by Ellmans methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAcetylcholinesterase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50267153(10-N-Demethyl-10-N-(9-(4-(piperidin-1-ylmethyl)phe...)
Affinity DataIC50: 88.1nMAssay Description:Inhibition of AChE from rat cortex homogenate by Ellmans methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAcetylcholinesterase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50267188(10-N-Demethyl-10-N-(4-(3-(1-morpholinoethyl)phenox...)
Affinity DataIC50: 94.1nMAssay Description:Inhibition of AChE from rat cortex homogenate by Ellmans methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAcetylcholinesterase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50267186(10-N-Demethyl-10-N-(4-(4-(morpholinomethyl)phenoxy...)
Affinity DataIC50: 99.1nMAssay Description:Inhibition of AChE from rat cortex homogenate by Ellmans methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAcetylcholinesterase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50267187(10-N-Demethyl-10-N-(6-(4-(morpholinomethyl)phenoxy...)
Affinity DataIC50: 113nMAssay Description:Inhibition of AChE from rat cortex homogenate by Ellmans methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAcetylcholinesterase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50267191(10-N-Demethyl-10-N-(6-(4-(pyrrolidine-1-carbonyl)-...)
Affinity DataIC50: 122nMAssay Description:Inhibition of AChE from rat cortex homogenate by Ellmans methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAcetylcholinesterase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50267189(10-N-Demethyl-10-N-(6-(3-(1-morpholinoethyl)phenox...)
Affinity DataIC50: 154nMAssay Description:Inhibition of AChE from rat cortex homogenate by Ellmans methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAcetylcholinesterase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50267221(10-N-Demethyl-10-N-(6-(1-benzylpiperidin-4-yloxy)-...)
Affinity DataIC50: 222nMAssay Description:Inhibition of AChE from rat cortex homogenate by Ellmans methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAcetylcholinesterase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50267220(10-N-Demethyl-10-N-(4-(1-benzylpiperidin-4-yloxy)-...)
Affinity DataIC50: 306nMAssay Description:Inhibition of AChE from rat cortex homogenate by Ellmans methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAcetylcholinesterase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM10404(galantamine | (1S,12S,14R)-9-methoxy-4-methyl-11-o...)
Affinity DataIC50: 1.17E+3nMAssay Description:Inhibition of AChE from rat cortex homogenate by Ellmans methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50267155(10-N-Demethyl-10-N-(12-(4-(piperidin-1-ylmethyl)-p...)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of BChE from rat serum by Ellmans methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50267186(10-N-Demethyl-10-N-(4-(4-(morpholinomethyl)phenoxy...)
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of BChE from rat serum by Ellmans methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50267187(10-N-Demethyl-10-N-(6-(4-(morpholinomethyl)phenoxy...)
Affinity DataIC50: 3.90E+3nMAssay Description:Inhibition of BChE from rat serum by Ellmans methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50267220(10-N-Demethyl-10-N-(4-(1-benzylpiperidin-4-yloxy)-...)
Affinity DataIC50: 4.30E+3nMAssay Description:Inhibition of BChE from rat serum by Ellmans methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50267221(10-N-Demethyl-10-N-(6-(1-benzylpiperidin-4-yloxy)-...)
Affinity DataIC50: 5.50E+3nMAssay Description:Inhibition of BChE from rat serum by Ellmans methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50267190(10-N-Demethyl-10-N-(4-(4-(pyrrolidine-1-carbonyl)-...)
Affinity DataIC50: 5.60E+3nMAssay Description:Inhibition of BChE from rat serum by Ellmans methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50267189(10-N-Demethyl-10-N-(6-(3-(1-morpholinoethyl)phenox...)
Affinity DataIC50: 5.80E+3nMAssay Description:Inhibition of BChE from rat serum by Ellmans methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM10404(galantamine | (1S,12S,14R)-9-methoxy-4-methyl-11-o...)
Affinity DataIC50: 5.90E+3nMAssay Description:Inhibition of BChE from rat serum by Ellmans methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50267188(10-N-Demethyl-10-N-(4-(3-(1-morpholinoethyl)phenox...)
Affinity DataIC50: 7.10E+3nMAssay Description:Inhibition of BChE from rat serum by Ellmans methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50267191(10-N-Demethyl-10-N-(6-(4-(pyrrolidine-1-carbonyl)-...)
Affinity DataIC50: 9.40E+3nMAssay Description:Inhibition of BChE from rat serum by Ellmans methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50267104(10-N-Demethyl-10-N-(2-(4-(piperidin-1-ylmethyl)phe...)
Affinity DataIC50: 2.10E+4nMAssay Description:Inhibition of BChE from rat serum by Ellmans methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50267105(10-N-Demethyl-10-N-(3-(4-(piperidin-1-ylmethyl)phe...)
Affinity DataIC50: 2.40E+4nMAssay Description:Inhibition of BChE from rat serum by Ellmans methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50267106(10-N-Demethyl-10-N-(4-(4-(piperidin-1-ylmethyl)phe...)
Affinity DataIC50: 2.80E+4nMAssay Description:Inhibition of BChE from rat serum by Ellmans methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50267150(10-N-Demethyl-10-N-(5-(4-(piperidin-1-ylmethyl)phe...)
Affinity DataIC50: 2.90E+4nMAssay Description:Inhibition of BChE from rat serum by Ellmans methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50267151(10-N-Demethyl-10-N-(6-(4-(piperidin-1-ylmethyl)phe...)
Affinity DataIC50: 3.30E+4nMAssay Description:Inhibition of BChE from rat serum by Ellmans methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50267156(10-N-Demethyl-10-N-(4-(4-((diethylamino)methyl)-ph...)
Affinity DataIC50: 3.40E+4nMAssay Description:Inhibition of BChE from rat serum by Ellmans methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50267157(10-N-Demethyl-10-N-(6-(4-((diethylamino)methyl)-ph...)
Affinity DataIC50: 4.10E+4nMAssay Description:Inhibition of BChE from rat serum by Ellmans methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50267152(10-N-Demethyl-10-N-(8-(4-(piperidin-1-ylmethyl)phe...)
Affinity DataIC50: 5.30E+4nMAssay Description:Inhibition of BChE from rat serum by Ellmans methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50267153(10-N-Demethyl-10-N-(9-(4-(piperidin-1-ylmethyl)phe...)
Affinity DataIC50: 6.40E+4nMAssay Description:Inhibition of BChE from rat serum by Ellmans methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50267154(10-N-Demethyl-10-N-(10-(4-(piperidin-1-ylmethyl)-p...)
Affinity DataIC50: 9.30E+4nMAssay Description:Inhibition of BChE from rat serum by Ellmans methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed