Compile Data Set for Download or QSAR
Report error Found 97 Enz. Inhib. hit(s) with all data for entry = 50026355
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243218(2-(4-((4-(5-(6-oxo-1,6-dihydropyridin-3-yl)-4H-1,2...)
Affinity DataIC50: 1nMAssay Description:Inhibition of Akt1More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243221(2-(4-((4-(5-(6-methoxypyridin-3-yl)-4H-1,2,4-triaz...)
Affinity DataIC50: 3nMAssay Description:Inhibition of Akt1More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243215(3-phenyl-2-(4-((4-(5-(pyridin-2-yl)-4H-1,2,4-triaz...)
Affinity DataIC50: 3.5nMAssay Description:Inhibition of Akt1More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243216(N,N-dimethyl-2-(4-(6-phenyl-7-(4-((4-(5-(pyridin-2...)
Affinity DataIC50: 4nMAssay Description:Inhibition of Akt1More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetRAC-beta serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243216(N,N-dimethyl-2-(4-(6-phenyl-7-(4-((4-(5-(pyridin-2...)
Affinity DataIC50: 4nMAssay Description:Inhibition of Akt2More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243219(2-(4-((4-(5-(6-aminopyridin-3-yl)-4H-1,2,4-triazol...)
Affinity DataIC50: 4nMAssay Description:Inhibition of Akt1More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243220(3-phenyl-2-(4-((4-(5-(pyrazin-2-yl)-4H-1,2,4-triaz...)
Affinity DataIC50: 4nMAssay Description:Inhibition of Akt1More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243217(3-phenyl-2-(4-((4-(5-(pyrimidin-2-yl)-4H-1,2,4-tri...)
Affinity DataIC50: 7nMAssay Description:Inhibition of Akt1More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetRAC-beta serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243218(2-(4-((4-(5-(6-oxo-1,6-dihydropyridin-3-yl)-4H-1,2...)
Affinity DataIC50: 8nMAssay Description:Inhibition of Akt2More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243216(N,N-dimethyl-2-(4-(6-phenyl-7-(4-((4-(5-(pyridin-2...)
Affinity DataIC50: 10nMAssay Description:Inhibition of Akt1 by cellular assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243286(N,N-dimethyl-2-(4-(2-phenyl-3-(4-((4-(5-(pyridin-2...)
Affinity DataIC50: 10nMAssay Description:Inhibition of Akt1 by cellular assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243285(2-(4-(2-phenyl-3-(4-((4-(5-(pyridin-2-yl)-4H-1,2,4...)
Affinity DataIC50: 13nMAssay Description:Inhibition of Akt1 by cellular assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243215(3-phenyl-2-(4-((4-(5-(pyridin-2-yl)-4H-1,2,4-triaz...)
Affinity DataIC50: 16nMAssay Description:Inhibition of Akt1 by cellular assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetRAC-beta serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243221(2-(4-((4-(5-(6-methoxypyridin-3-yl)-4H-1,2,4-triaz...)
Affinity DataIC50: 16nMAssay Description:Inhibition of Akt2More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243284(6-(4-methylpiperazin-1-yl)-2-phenyl-3-(4-((4-(5-(p...)
Affinity DataIC50: 18nMAssay Description:Inhibition of Akt1 by cellular assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243275(5-(5-(1-((4-(2-(4-methylpiperazin-1-yl)-6-phenylpy...)
Affinity DataIC50: 20nMAssay Description:Inhibition of Akt1 by cellular assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetRAC-beta serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243220(3-phenyl-2-(4-((4-(5-(pyrazin-2-yl)-4H-1,2,4-triaz...)
Affinity DataIC50: 21nMAssay Description:Inhibition of Akt2More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243217(3-phenyl-2-(4-((4-(5-(pyrimidin-2-yl)-4H-1,2,4-tri...)
Affinity DataIC50: 23nMAssay Description:Inhibition of Akt1 by cellular assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243272(2-(4-methylpiperazin-1-yl)-6-phenyl-7-(4-((4-(5-(p...)
Affinity DataIC50: 25nMAssay Description:Inhibition of Akt1 by cellular assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243219(2-(4-((4-(5-(6-aminopyridin-3-yl)-4H-1,2,4-triazol...)
Affinity DataIC50: 26nMAssay Description:Inhibition of Akt1 by cellular assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetRAC-beta serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243215(3-phenyl-2-(4-((4-(5-(pyridin-2-yl)-4H-1,2,4-triaz...)
Affinity DataIC50: 26nMAssay Description:Inhibition of Akt2More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243283(Dimethyl-(2-{4-[7-(4-{4-[5-(1-oxy-pyridin-4-yl)-4H...)
Affinity DataIC50: 33nMAssay Description:Inhibition of Akt1 by cellular assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetRAC-beta serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243219(2-(4-((4-(5-(6-aminopyridin-3-yl)-4H-1,2,4-triazol...)
Affinity DataIC50: 33nMAssay Description:Inhibition of Akt2More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243274(N,N-dimethyl-2-(4-(6-phenyl-7-(4-((4-(5-(pyrimidin...)
Affinity DataIC50: 35nMAssay Description:Inhibition of Akt1 by cellular assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243273(2-(4-(6-phenyl-7-(4-((4-(5-(pyrimidin-2-yl)-4H-1,2...)
Affinity DataIC50: 37nMAssay Description:Inhibition of Akt1 by cellular assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243277(5-(5-(1-((4-(2-(4-(2-(dimethylamino)ethyl)piperazi...)
Affinity DataIC50: 37nMAssay Description:Inhibition of Akt1 by cellular assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243276(2-(4-(7-(4-((4-(5-(6-aminopyridin-3-yl)-4H-1,2,4-t...)
Affinity DataIC50: 38nMAssay Description:Inhibition of Akt1 by cellular assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetRAC-beta serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243216(N,N-dimethyl-2-(4-(6-phenyl-7-(4-((4-(5-(pyridin-2...)
Affinity DataIC50: 39nMAssay Description:Inhibition of Akt2 by cellular assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243221(2-(4-((4-(5-(6-methoxypyridin-3-yl)-4H-1,2,4-triaz...)
Affinity DataIC50: 40nMAssay Description:Inhibition of Akt1 by cellular assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetRAC-beta serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243272(2-(4-methylpiperazin-1-yl)-6-phenyl-7-(4-((4-(5-(p...)
Affinity DataIC50: 40nMAssay Description:Inhibition of Akt2 by cellular assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetRAC-beta serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243286(N,N-dimethyl-2-(4-(2-phenyl-3-(4-((4-(5-(pyridin-2...)
Affinity DataIC50: 43nMAssay Description:Inhibition of Akt2 by cellular assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243220(3-phenyl-2-(4-((4-(5-(pyrazin-2-yl)-4H-1,2,4-triaz...)
Affinity DataIC50: 44nMAssay Description:Inhibition of Akt1 by cellular assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetRAC-beta serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243217(3-phenyl-2-(4-((4-(5-(pyrimidin-2-yl)-4H-1,2,4-tri...)
Affinity DataIC50: 44nMAssay Description:Inhibition of Akt2More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetRAC-beta serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243285(2-(4-(2-phenyl-3-(4-((4-(5-(pyridin-2-yl)-4H-1,2,4...)
Affinity DataIC50: 48nMAssay Description:Inhibition of Akt2 by cellular assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243287(6-(4-methylpiperazin-1-yl)-2-phenyl-3-(4-((4-(5-(p...)
Affinity DataIC50: 52nMAssay Description:Inhibition of Akt1 by cellular assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243218(2-(4-((4-(5-(6-oxo-1,6-dihydropyridin-3-yl)-4H-1,2...)
Affinity DataIC50: 62nMAssay Description:Inhibition of Akt1 by cellular assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243282(2-{4-[7-(4-{4-[5-(1-Oxy-pyridin-4-yl)-4H-[1,2,4]tr...)
Affinity DataIC50: 67nMAssay Description:Inhibition of Akt1 by cellular assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetRAC-beta serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243283(Dimethyl-(2-{4-[7-(4-{4-[5-(1-oxy-pyridin-4-yl)-4H...)
Affinity DataIC50: 68nMAssay Description:Inhibition of Akt2 by cellular assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243280(5-(5-(1-((4-(2-(4-(2-(dimethylamino)ethyl)piperazi...)
Affinity DataIC50: 69nMAssay Description:Inhibition of Akt1 by cellular assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetRAC-beta serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243217(3-phenyl-2-(4-((4-(5-(pyrimidin-2-yl)-4H-1,2,4-tri...)
Affinity DataIC50: 69nMAssay Description:Inhibition of Akt2 by cellular assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243290(5-(5-(1-((4-(6-(4-methylpiperazin-1-yl)-2-phenylpy...)
Affinity DataIC50: 70nMAssay Description:Inhibition of Akt1 by cellular assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243278(5-(5-(1-((4-(2-(4-methylpiperazin-1-yl)-6-phenylpy...)
Affinity DataIC50: 71nMAssay Description:Inhibition of Akt1 by cellular assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243288(2-(4-(2-phenyl-3-(4-((4-(5-(pyrimidin-2-yl)-4H-1,2...)
Affinity DataIC50: 72nMAssay Description:Inhibition of Akt1 by cellular assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetRAC-beta serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243273(2-(4-(6-phenyl-7-(4-((4-(5-(pyrimidin-2-yl)-4H-1,2...)
Affinity DataIC50: 80nMAssay Description:Inhibition of Akt2 by cellular assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetRAC-beta serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243275(5-(5-(1-((4-(2-(4-methylpiperazin-1-yl)-6-phenylpy...)
Affinity DataIC50: 84nMAssay Description:Inhibition of Akt2 by cellular assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243281(2-(4-Methyl-piperazin-1-yl)-7-(4-{4-[5-(1-oxy-pyri...)
Affinity DataIC50: 88nMAssay Description:Inhibition of Akt1 by cellular assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetRAC-beta serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243284(6-(4-methylpiperazin-1-yl)-2-phenyl-3-(4-((4-(5-(p...)
Affinity DataIC50: 92nMAssay Description:Inhibition of Akt2 by cellular assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetRAC-beta serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243280(5-(5-(1-((4-(2-(4-(2-(dimethylamino)ethyl)piperazi...)
Affinity DataIC50: 98nMAssay Description:Inhibition of Akt2 by cellular assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243289(N,N-dimethyl-2-(4-(2-phenyl-3-(4-((4-(5-(pyrimidin...)
Affinity DataIC50: 104nMAssay Description:Inhibition of Akt1 by cellular assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50243291(2-(4-(3-(4-((4-(5-(6-aminopyridin-3-yl)-4H-1,2,4-t...)
Affinity DataIC50: 115nMAssay Description:Inhibition of Akt1 by cellular assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
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