Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50039265
TargetNuclear receptor subfamily 4 group A member 1(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50378798(CYTOSPORONE B)
Affinity DataKd:  1.51E+3nMAssay Description:Binding affinity to NuR77-LBD receptor expressed in human BGC823 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetNuclear receptor subfamily 4 group A member 1(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50378798(CYTOSPORONE B)
Affinity DataEC50:  0.115nMAssay Description:Agonist activity at nuclear orphan receptor Nur77 expressed in human BGC823 cells co-transfected with fused GAL4-LBD assessed as transactivation afte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetNuclear receptor subfamily 4 group A member 1(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50378798(CYTOSPORONE B)
Affinity DataEC50:  0.278nMAssay Description:Agonist activity at nuclear orphan receptor Nur77 expressed in human BGC823 cells co-transfected with fused GAL4-Nur77 assessed as transactivation af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetRetinoic acid receptor RXR-alpha(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM31892(CHEMBL705 | 9-cis retinoic acid | alitretinoin | P...)
Affinity DataKd:  240nMAssay Description:Binding affinity to RXRalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetNuclear receptor subfamily 4 group A member 1(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50378798(CYTOSPORONE B)
Affinity DataKd:  740nMAssay Description:Binding affinity to Nur77 receptor expressed in human BGC823 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)