Compile Data Set for Download or QSAR
Report error Found 24 Enz. Inhib. hit(s) with all data for entry = 50027297
TargetDipeptidyl peptidase 4(Human)
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50276045((R)-3-Amino-4-(5-chloro-2-fluoro-phenyl)-N-{4-[6-(...)
Affinity DataIC50: 0.640nMAssay Description:Inhibition of human Caco-2 cells-derived DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50276047((R)-3-Amino-N-{4-[6-(2-morpholin-4-yl-ethoxy)-benz...)
Affinity DataIC50: 0.790nMAssay Description:Inhibition of human Caco-2 cells-derived DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50276001((R)-3-Amino-N-{4-[6-(2-methoxy-ethoxy)-benzothiazo...)
Affinity DataIC50: 1nMAssay Description:Inhibition of human Caco-2 cells-derived DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50276046((R)-3-amino-4-(5-chloro-2-fluorophenyl)-N-(4-(6-(2...)
Affinity DataIC50: 1.90nMAssay Description:Inhibition of human Caco-2 cells-derived DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50275954((R)-3-Amino-N-[4-(6-methoxy-benzothiazol-2-yl)-1,1...)
Affinity DataIC50: 2.70nMAssay Description:Inhibition of human Caco-2 cells-derived DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50275955((R)-3-Amino-N-[4-(5-methoxy-benzothiazol-2-yl)-1,1...)
Affinity DataIC50: 3.30nMAssay Description:Inhibition of human Caco-2 cells-derived DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50276044((3R)-3-amino-4-(2,4,5-trifluorophenyl)-N-{4-[6-(2-...)
Affinity DataIC50: 3.60nMAssay Description:Inhibition of human Caco-2 cells-derived DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50275905((R)-3-Amino-4-(2-fluoro-phenyl)-N-[4-(6-methoxy-be...)
Affinity DataIC50: 12nMAssay Description:Inhibition of human Caco-2 cells-derived DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50275904((R)-3-Amino-N-(4-benzothiazol-2-yl-1,1-dioxo-hexah...)
Affinity DataIC50: 13nMAssay Description:Inhibition of human Caco-2 cells-derived DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50275957((R)-3-Amino-N-[4-(6-chloro-benzothiazol-2-yl)-1,1-...)
Affinity DataIC50: 35nMAssay Description:Inhibition of human Caco-2 cells-derived DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50275903((R)-3-Amino-N-(4-benzothiazol-2-yl-1,1-dioxo-hexah...)
Affinity DataIC50: 64nMAssay Description:Inhibition of human Caco-2 cells-derived DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50275999((R)-3-Amino-4-(2-fluoro-phenyl)-N-[4-(6-methyl-ben...)
Affinity DataIC50: 70nMAssay Description:Inhibition of human Caco-2 cells-derived DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50275998((R)-3-Amino-N-[4-(4-chloro-benzothiazol-2-yl)-1,1-...)
Affinity DataIC50: 130nMAssay Description:Inhibition of human Caco-2 cells-derived DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50275849((R)-3-Amino-N-(1,1-dioxo-4-thiazol-2-yl-hexahydro-...)
Affinity DataIC50: 190nMAssay Description:Inhibition of human Caco-2 cells-derived DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50275956((R)-3-Amino-4-(2-fluoro-phenyl)-N-[4-(4-methoxy-be...)
Affinity DataIC50: 270nMAssay Description:Inhibition of human Caco-2 cells-derived DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50276000((R)-3-Amino-4-(2-fluoro-phenyl)-N-[4-(4-methyl-ben...)
Affinity DataIC50: 350nMAssay Description:Inhibition of human Caco-2 cells-derived DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50275848((R)-3-Amino-N-(1,1-dioxo-4-pyridin-2-yl-hexahydro-...)
Affinity DataIC50: 470nMAssay Description:Inhibition of human Caco-2 cells-derived DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50275847((R)-3-Amino-N-(1,1-dioxo-4-phenyl-hexahydro-1lambd...)
Affinity DataIC50: 570nMAssay Description:Inhibition of human Caco-2 cells-derived DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50275791((R)-3-amino-4-(2-fluorophenyl)-N-(1-methyl-4-pheny...)
Affinity DataIC50: 870nMAssay Description:Inhibition of human Caco-2 cells-derived DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50275789((R)-3-amino-N-(1-benzyl-4-phenylpiperidin-4-yl)-4-...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human Caco-2 cells-derived DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50275790((R)-3-amino-N-(1,4-dibenzylpiperidin-4-yl)-4-(2-fl...)
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of human Caco-2 cells-derived DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50275845((R)-3-amino-4-(2-fluorophenyl)-N-(4-phenyltetrahyd...)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of human Caco-2 cells-derived DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50275846((R)-3-amino-4-(2-fluorophenyl)-N-(4-phenyltetrahyd...)
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of human Caco-2 cells-derived DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50275788((R)-3-amino-N-(1-benzyl-4-methylpiperidin-4-yl)-4-...)
Affinity DataIC50: 7.80E+3nMAssay Description:Inhibition of human Caco-2 cells-derived DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed