Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50027306
TargetPeroxisome proliferator-activated receptor alpha(Human)
University of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50264403(4-(2-(4-ethyl-5-(7-methoxybenzofuran-2-yl)-4H-1,2,...)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of fluorescent pan PPAR agonist form GST-tagged human PPARalpha ligand binding domain by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
University of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50264402(ethyl 3-((4-(methoxycarbonyl)phenyl)carbamoyl)-2-(...)
Affinity DataIC50: 1.50E+3nMAssay Description:Displacement of fluorescent pan PPAR agonist form GST-tagged human PPARalpha ligand binding domain by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
University of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50264405((S)-methyl 4-(2-(3-(4-methoxybenzyl)-1-(3-methoxyp...)
Affinity DataIC50: 7.20E+3nMAssay Description:Displacement of fluorescent pan PPAR agonist form GST-tagged human PPARdelta ligand binding domain by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
University of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50264405((S)-methyl 4-(2-(3-(4-methoxybenzyl)-1-(3-methoxyp...)
Affinity DataIC50: 1.30E+4nMAssay Description:Displacement of fluorescent pan PPAR agonist form GST-tagged human PPARgamma ligand binding domain by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
University of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50264404(4-((1-((4-morpholinophenylimino)methyl)naphthalen-...)
Affinity DataIC50: 2.00E+4nMAssay Description:Displacement of fluorescent pan PPAR agonist form GST-tagged human PPARgamma ligand binding domain by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
University of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50264404(4-((1-((4-morpholinophenylimino)methyl)naphthalen-...)
Affinity DataIC50: 3.40E+4nMAssay Description:Displacement of fluorescent pan PPAR agonist form GST-tagged human PPARdelta ligand binding domain by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
University of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50264403(4-(2-(4-ethyl-5-(7-methoxybenzofuran-2-yl)-4H-1,2,...)
Affinity DataIC50: 4.00E+4nMAssay Description:Displacement of fluorescent pan PPAR agonist form GST-tagged human PPARgamma ligand binding domain by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
University of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50264404(4-((1-((4-morpholinophenylimino)methyl)naphthalen-...)
Affinity DataIC50: 4.30E+4nMAssay Description:Displacement of fluorescent pan PPAR agonist form GST-tagged human PPARalpha ligand binding domain by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
University of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50264371((S)-ethyl 3-(2-(1-(2-chloro-6-fluorobenzoyl)piperi...)
Affinity DataIC50: 4.40E+4nMAssay Description:Displacement of fluorescent pan PPAR agonist form GST-tagged human PPARgamma ligand binding domain by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
University of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50264403(4-(2-(4-ethyl-5-(7-methoxybenzofuran-2-yl)-4H-1,2,...)
Affinity DataIC50: 3.90E+5nMAssay Description:Displacement of fluorescent pan PPAR agonist form GST-tagged human PPARdelta ligand binding domain by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed