Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 2859
TargetAndrogen receptor(Human)
Pfizer

LigandPNGBDBM25428(4-[3-(4-hydroxybutyl)-4,4-dimethyl-2,5-dioxoimidaz...)
Affinity DataIC50: 16nMpH: 7.4 T: 2°CAssay Description:The competitive radio-ligand binding analysis was performed on human AR extracts from transfected Sf9 cells in the presence or absence of differing c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2008
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
Pfizer

LigandPNGBDBM25432(6-{methyl[(1R)-1-phenylethyl]amino}-4-(trifluorome...)
Affinity DataIC50: 20nMpH: 7.4 T: 2°CAssay Description:The competitive radio-ligand binding analysis was performed on human AR extracts from transfected Sf9 cells in the presence or absence of differing c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2008
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
Pfizer

LigandPNGBDBM25434(4-(2-hydroxycyclohexyl)-2-(trifluoromethyl)benzoni...)
Affinity DataIC50: 26nMpH: 7.4 T: 2°CAssay Description:The competitive radio-ligand binding analysis was performed on human AR extracts from transfected Sf9 cells in the presence or absence of differing c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2008
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
Pfizer

LigandPNGBDBM25431(4-(2-hydroxyphenyl)-2-methoxybenzonitrile | diaryl...)
Affinity DataIC50: 37nMpH: 7.4 T: 2°CAssay Description:The competitive radio-ligand binding analysis was performed on human AR extracts from transfected Sf9 cells in the presence or absence of differing c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2008
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
Pfizer

LigandPNGBDBM25436(PF-0998425 | 4-[(1R,2R)-2-hydroxycyclohexyl]-2-(tr...)
Affinity DataIC50: 37nMpH: 7.4 T: 2°CAssay Description:The competitive radio-ligand binding analysis was performed on human AR extracts from transfected Sf9 cells in the presence or absence of differing c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2008
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
Pfizer

LigandPNGBDBM25430(CHEMBL391548 | 4-(2-hydroxyphenyl)-2-(trifluoromet...)
Affinity DataIC50: 39.9nMpH: 7.4 T: 2°CAssay Description:The competitive radio-ligand binding analysis was performed on human AR extracts from transfected Sf9 cells in the presence or absence of differing c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2008
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
Pfizer

LigandPNGBDBM25437(4-{[(1R,2S)-2-cyanocyclohexyl]oxy}-2-(trifluoromet...)
Affinity DataIC50: 60nMpH: 7.4 T: 2°CAssay Description:The competitive radio-ligand binding analysis was performed on human AR extracts from transfected Sf9 cells in the presence or absence of differing c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2008
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
Pfizer

LigandPNGBDBM25435(4-[(1S,2S)-2-hydroxycyclohexyl]-2-(trifluoromethyl...)
Affinity DataIC50: 1.60E+3nMpH: 7.4 T: 2°CAssay Description:The competitive radio-ligand binding analysis was performed on human AR extracts from transfected Sf9 cells in the presence or absence of differing c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2008
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
Pfizer

LigandPNGBDBM25433(4-[(1R,2S)-2-hydroxycyclohexyl]-2-(trifluoromethyl...)
Affinity DataIC50: 3.00E+3nMpH: 7.4 T: 2°CAssay Description:The competitive radio-ligand binding analysis was performed on human AR extracts from transfected Sf9 cells in the presence or absence of differing c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2008
Entry Details Article
PubMed