Compile Data Set for Download or QSAR
Report error Found 28 Enz. Inhib. hit(s) with all data for entry = 50027431
TargetProto-oncogene tyrosine-protein kinase Src(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM4552(CHEMBL288441 | SKI-606 | 4-[(2,4-Dichloro-5-methox...)
Affinity DataIC50: 1.20nMAssay Description:Inhibition of cSrc by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetProto-oncogene tyrosine-protein kinase Src(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM4552(CHEMBL288441 | SKI-606 | 4-[(2,4-Dichloro-5-methox...)
Affinity DataIC50: 1.80nMAssay Description:Inhibition of cSrcMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetProto-oncogene tyrosine-protein kinase Src(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50271896(6-methyl-4-(6-methylbenzo[d]thiazol-2-ylamino)-7-(...)
Affinity DataIC50: 15.4nMAssay Description:Inhibition of cSrcMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50275877(4-(2-aminobenzo[d]thiazol-6-ylamino)-6-methoxy-7-(...)
Affinity DataIC50: 20.7nMAssay Description:Inhibition of cSrcMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50275756(4-(2-aminobenzo[d]thiazol-6-ylamino)-6-methyl-7-(2...)
Affinity DataIC50: 34.8nMAssay Description:Inhibition of cSrcMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50275812(4-(2-aminobenzo[d]thiazol-6-ylamino)-7-(3-(3,5-dim...)
Affinity DataIC50: 36.6nMAssay Description:Inhibition of cSrcMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50275813(4-(2-aminobenzo[d]thiazol-6-ylamino)-7-(3-(diethyl...)
Affinity DataIC50: 42nMAssay Description:Inhibition of cSrcMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50275757(4-(2-aminobenzo[d]thiazol-6-ylamino)-6-methyl-7-(3...)
Affinity DataIC50: 50.6nMAssay Description:Inhibition of cSrcMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50275811(4-(2-aminobenzo[d]thiazol-6-ylamino)-6-methyl-7-(3...)
Affinity DataIC50: 53.4nMAssay Description:Inhibition of cSrcMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50275758(4-(2-aminobenzo[d]thiazol-6-ylamino)-6-methyl-7-(3...)
Affinity DataIC50: 81.1nMAssay Description:Inhibition of cSrcMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50275759(4-(2-aminobenzo[d]thiazol-6-ylamino)-6-methyl-7-(3...)
Affinity DataIC50: 129nMAssay Description:Inhibition of cSrcMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50275875(4-(2-amino-1H-benzo[d]imidazol-6-ylamino)-7-(3-(di...)
Affinity DataIC50: 143nMAssay Description:Inhibition of cSrcMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50275876(4-(2-amino-1H-benzo[d]imidazol-6-ylamino)-6-methyl...)
Affinity DataIC50: 159nMAssay Description:Inhibition of cSrcMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50275814(4-(2-aminobenzo[d]thiazol-6-ylamino)-7-(3-(3,5-dim...)
Affinity DataIC50: 267nMAssay Description:Inhibition of cSrcMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetNitric oxide synthase, inducible(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50275814(4-(2-aminobenzo[d]thiazol-6-ylamino)-7-(3-(3,5-dim...)
Affinity DataIC50: 1.05E+4nMAssay Description:Inhibition of iNOS in mouse ANA1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetNitric oxide synthase, inducible(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50275811(4-(2-aminobenzo[d]thiazol-6-ylamino)-6-methyl-7-(3...)
Affinity DataIC50: 1.27E+4nMAssay Description:Inhibition of iNOS in mouse ANA1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetNitric oxide synthase, inducible(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50275875(4-(2-amino-1H-benzo[d]imidazol-6-ylamino)-7-(3-(di...)
Affinity DataIC50: 1.32E+4nMAssay Description:Inhibition of iNOS in mouse ANA1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetNitric oxide synthase, inducible(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50275759(4-(2-aminobenzo[d]thiazol-6-ylamino)-6-methyl-7-(3...)
Affinity DataIC50: 1.73E+4nMAssay Description:Inhibition of iNOS in mouse ANA1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetNitric oxide synthase, inducible(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50240843(Thiazol-2-ylamine | Basedol | thiazol-2-amine | 2-...)
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of iNOS in mouse ANA1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetNitric oxide synthase, inducible(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50275876(4-(2-amino-1H-benzo[d]imidazol-6-ylamino)-6-methyl...)
Affinity DataIC50: 2.48E+4nMAssay Description:Inhibition of iNOS in mouse ANA1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetNitric oxide synthase, inducible(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50275756(4-(2-aminobenzo[d]thiazol-6-ylamino)-6-methyl-7-(2...)
Affinity DataIC50: 2.67E+4nMAssay Description:Inhibition of iNOS in mouse ANA1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetNitric oxide synthase, inducible(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50275758(4-(2-aminobenzo[d]thiazol-6-ylamino)-6-methyl-7-(3...)
Affinity DataIC50: 3.18E+4nMAssay Description:Inhibition of iNOS in mouse ANA1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetNitric oxide synthase, inducible(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50275757(4-(2-aminobenzo[d]thiazol-6-ylamino)-6-methyl-7-(3...)
Affinity DataIC50: 3.71E+4nMAssay Description:Inhibition of iNOS in mouse ANA1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetNitric oxide synthase, inducible(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50275813(4-(2-aminobenzo[d]thiazol-6-ylamino)-7-(3-(diethyl...)
Affinity DataIC50: 4.68E+4nMAssay Description:Inhibition of iNOS in mouse ANA1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetNitric oxide synthase, inducible(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50271982(L-canavanine | CHEMBL443732)
Affinity DataIC50: 6.00E+4nMAssay Description:Inhibition of iNOS in mouse ANA1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetNitric oxide synthase, inducible(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50275812(4-(2-aminobenzo[d]thiazol-6-ylamino)-7-(3-(3,5-dim...)
Affinity DataIC50: 8.91E+4nMAssay Description:Inhibition of iNOS in mouse ANA1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetNitric oxide synthase, inducible(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50275877(4-(2-aminobenzo[d]thiazol-6-ylamino)-6-methoxy-7-(...)
Affinity DataIC50: 1.05E+5nMAssay Description:Inhibition of iNOS in mouse ANA1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetNitric oxide synthase, inducible(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50271896(6-methyl-4-(6-methylbenzo[d]thiazol-2-ylamino)-7-(...)
Affinity DataIC50: 3.13E+5nMAssay Description:Inhibition of iNOS in mouse ANA1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed