Compile Data Set for Download or QSAR
Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 3482
TargetGlycogen phosphorylase, liver form(Human)
Astellas Pharma

LigandPNGBDBM35353(indole-2-carboxamide derivative, 25e (R-isomer))
Affinity DataIC50: 20nMpH: 6.8 T: 2°CAssay Description:The activity of recombinant human liver GPa in the forward direction was measured by monitoring the production of NADPH. Enzyme activity was assayed...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Astellas Pharma

LigandPNGBDBM35351(indole-2-carboxamide derivative, 25e)
Affinity DataIC50: 36nMpH: 6.8 T: 2°CAssay Description:The activity of recombinant human liver GPa in the forward direction was measured by monitoring the production of NADPH. Enzyme activity was assayed...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Astellas Pharma

LigandPNGBDBM35350(indole-2-carboxamide derivative, 25d)
Affinity DataIC50: 48nMpH: 6.8 T: 2°CAssay Description:The activity of recombinant human liver GPa in the forward direction was measured by monitoring the production of NADPH. Enzyme activity was assayed...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Astellas Pharma

LigandPNGBDBM35349(indole-2-carboxamide derivative, 25c)
Affinity DataIC50: 63nMpH: 6.8 T: 2°CAssay Description:The activity of recombinant human liver GPa in the forward direction was measured by monitoring the production of NADPH. Enzyme activity was assayed...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Astellas Pharma

LigandPNGBDBM35345(indole-2-carboxamide derivative, 15)
Affinity DataIC50: 68nMpH: 6.8 T: 2°CAssay Description:The activity of recombinant human liver GPa in the forward direction was measured by monitoring the production of NADPH. Enzyme activity was assayed...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Astellas Pharma

LigandPNGBDBM35352(indole-2-carboxamide derivative, 25e (S-isomer))
Affinity DataIC50: 160nMpH: 6.8 T: 2°CAssay Description:The activity of recombinant human liver GPa in the forward direction was measured by monitoring the production of NADPH. Enzyme activity was assayed...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Astellas Pharma

LigandPNGBDBM35339(indole-2-carboxamide derivative, 5b)
Affinity DataIC50: 320nMpH: 6.8 T: 2°CAssay Description:The activity of recombinant human liver GPa in the forward direction was measured by monitoring the production of NADPH. Enzyme activity was assayed...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Astellas Pharma

LigandPNGBDBM35338(indole-2-carboxamide derivative, 3)
Affinity DataIC50: 440nMpH: 6.8 T: 2°CAssay Description:The activity of recombinant human liver GPa in the forward direction was measured by monitoring the production of NADPH. Enzyme activity was assayed...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Astellas Pharma

LigandPNGBDBM35348(indole-2-carboxamide derivative, 25b)
Affinity DataIC50: 590nMpH: 6.8 T: 2°CAssay Description:The activity of recombinant human liver GPa in the forward direction was measured by monitoring the production of NADPH. Enzyme activity was assayed...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Astellas Pharma

LigandPNGBDBM35343(trans-isomers+ 9a | indole-2-carboxamide derivativ...)
Affinity DataIC50: 800nMpH: 6.8 T: 2°CAssay Description:The activity of recombinant human liver GPa in the forward direction was measured by monitoring the production of NADPH. Enzyme activity was assayed...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Astellas Pharma

LigandPNGBDBM35347(indole-2-carboxamide derivative, 25a)
Affinity DataIC50: 810nMpH: 6.8 T: 2°CAssay Description:The activity of recombinant human liver GPa in the forward direction was measured by monitoring the production of NADPH. Enzyme activity was assayed...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Astellas Pharma

LigandPNGBDBM35341(indole-2-carboxamide derivative, 7)
Affinity DataIC50: 900nMpH: 6.8 T: 2°CAssay Description:The activity of recombinant human liver GPa in the forward direction was measured by monitoring the production of NADPH. Enzyme activity was assayed...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Astellas Pharma

LigandPNGBDBM35346(5-CHLORO-1H-INDOLE-2-CARBOXYLIC ACID [1-(4-FLUOROB...)
Affinity DataIC50: 920nMpH: 6.8 T: 2°CAssay Description:The activity of recombinant human liver GPa in the forward direction was measured by monitoring the production of NADPH. Enzyme activity was assayed...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Astellas Pharma

LigandPNGBDBM35340(indole-2-carboxamide derivative, 5c)
Affinity DataIC50: 1.20E+3nMpH: 6.8 T: 2°CAssay Description:The activity of recombinant human liver GPa in the forward direction was measured by monitoring the production of NADPH. Enzyme activity was assayed...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Astellas Pharma

LigandPNGBDBM35342(cis-isomers | indole-2-carboxamide derivative, 9a)
Affinity DataIC50: 8.50E+3nMpH: 6.8 T: 2°CAssay Description:The activity of recombinant human liver GPa in the forward direction was measured by monitoring the production of NADPH. Enzyme activity was assayed...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Astellas Pharma

LigandPNGBDBM35344(indole-2-carboxamide derivative, 12)
Affinity DataIC50: 1.00E+4nMpH: 6.8 T: 2°CAssay Description:The activity of recombinant human liver GPa in the forward direction was measured by monitoring the production of NADPH. Enzyme activity was assayed...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2009
Entry Details Article
PubMed