Compile Data Set for Download or QSAR
Report error Found 23 Enz. Inhib. hit(s) with all data for entry = 50041652
TargetCorticotropin-releasing factor receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50116105(3-(6-(dimethylamino)-4-methylpyridin-3-yl)-2,5-dim...)
Affinity DataIC50: 28.2nMAssay Description:Displacement of [125I]sauvagine from human recombinant CRF1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50412811(CHEMBL458810)
Affinity DataIC50: 32.4nMAssay Description:Displacement of [125I]sauvagine from human recombinant CRF1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50084875(DMP696 | [8-(2,4-dichloro-phenyl)-2,7-dimethyl-pyr...)
Affinity DataIC50: 39.8nMAssay Description:Displacement of [125I]sauvagine from human recombinant CRF1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50412814(CHEMBL456660)
Affinity DataIC50: 50.1nMAssay Description:Displacement of [125I]sauvagine from human recombinant CRF1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50412812(CHEMBL459173)
Affinity DataIC50: 56.2nMAssay Description:Displacement of [125I]sauvagine from human recombinant CRF1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50412798(EMICERFONT)
Affinity DataIC50: 66.1nMAssay Description:Displacement of [125I]sauvagine from human recombinant CRF1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50412809(CHEMBL516170)
Affinity DataIC50: 67.6nMAssay Description:Displacement of [125I]sauvagine from human recombinant CRF1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50412808(CHEMBL456640)
Affinity DataIC50: 67.6nMAssay Description:Displacement of [125I]sauvagine from human recombinant CRF1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50412798(EMICERFONT)
Affinity DataKd:  72.4nMAssay Description:Antagonist activity at human CRF1 receptor expressed in CHO cells assessed as effect on sauvagine-induced cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50412817(CHEMBL464185)
Affinity DataIC50: 89.1nMAssay Description:Displacement of [125I]sauvagine from human recombinant CRF1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50412813(CHEMBL513937)
Affinity DataIC50: 120nMAssay Description:Displacement of [125I]sauvagine from human recombinant CRF1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50412802(CHEMBL515363)
Affinity DataIC50: 120nMAssay Description:Displacement of [125I]sauvagine from human recombinant CRF1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50412799(CHEMBL458599)
Affinity DataIC50: 123nMAssay Description:Displacement of [125I]sauvagine from human recombinant CRF1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50412803(CHEMBL456448)
Affinity DataIC50: 145nMAssay Description:Displacement of [125I]sauvagine from human recombinant CRF1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50412816(CHEMBL464184)
Affinity DataIC50: 158nMAssay Description:Displacement of [125I]sauvagine from human recombinant CRF1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50412804(CHEMBL456449)
Affinity DataIC50: 309nMAssay Description:Displacement of [125I]sauvagine from human recombinant CRF1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50412806(CHEMBL457710)
Affinity DataIC50: 316nMAssay Description:Displacement of [125I]sauvagine from human recombinant CRF1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50412815(CHEMBL457742)
Affinity DataIC50: 363nMAssay Description:Displacement of [125I]sauvagine from human recombinant CRF1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50412810(CHEMBL458626)
Affinity DataIC50: 372nMAssay Description:Displacement of [125I]sauvagine from human recombinant CRF1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50412800(CHEMBL515532)
Affinity DataIC50: 794nMAssay Description:Displacement of [125I]sauvagine from human recombinant CRF1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50412807(CHEMBL457975)
Affinity DataIC50: 1.23E+3nMAssay Description:Displacement of [125I]sauvagine from human recombinant CRF1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50412801(CHEMBL458600)
Affinity DataIC50: 1.95E+3nMAssay Description:Displacement of [125I]sauvagine from human recombinant CRF1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50412805(CHEMBL515503)
Affinity DataIC50: 3.24E+3nMAssay Description:Displacement of [125I]sauvagine from human recombinant CRF1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed