Compile Data Set for Download or QSAR
Report error Found 94 Enz. Inhib. hit(s) with all data for entry = 50027681
TargetGlucocorticoid receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50254466(5-amino-N-(2-((2,6-dichloro-N-ethylbenzamido)methy...)
Affinity DataEC50:  2nMAssay Description:Agonist activity at human glucocorticoid receptor in human A549 cells assessed as transcriptional activity by MMTV luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50412614(CHEMBL465919)
Affinity DataEC50:  3.16nMAssay Description:Agonist activity at human glucocorticoid receptor in human A549 cells assessed as transcriptional activity by MMTV luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50254466(5-amino-N-(2-((2,6-dichloro-N-ethylbenzamido)methy...)
Affinity DataIC50: 3.16nMAssay Description:Displacement of fluorescent labelled Dexamethasone from glucocorticoid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50412614(CHEMBL465919)
Affinity DataIC50: 6.31nMAssay Description:Displacement of fluorescent labelled Dexamethasone from glucocorticoid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50254464(5-amino-N-(2-((2-chloro-N-ethylbenzamido)methyl)-3...)
Affinity DataEC50:  6.31nMAssay Description:Agonist activity at human glucocorticoid receptor in human A549 cells assessed as transcriptional activity by MMTV luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50254464(5-amino-N-(2-((2-chloro-N-ethylbenzamido)methyl)-3...)
Affinity DataEC50:  6.31nMAssay Description:Agonist activity at human glucocorticoid receptor in human A549 cells assessed as transcriptional activity by MMTV luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50412612(CHEMBL518451)
Affinity DataIC50: 6.31nMAssay Description:Displacement of fluorescent labelled Dexamethasone from glucocorticoid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50412609(CHEMBL520750)
Affinity DataIC50: 7.94nMAssay Description:Displacement of fluorescent labelled Dexamethasone from glucocorticoid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50254513(5-amino-N-(2-((N-ethyl-2,6-difluorobenzamido)methy...)
Affinity DataIC50: 7.94nMAssay Description:Displacement of fluorescent labelled Dexamethasone from glucocorticoid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50254513(5-amino-N-(2-((N-ethyl-2,6-difluorobenzamido)methy...)
Affinity DataEC50:  7.94nMAssay Description:Agonist activity at human glucocorticoid receptor in human A549 cells assessed as transcriptional activity by MMTV luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM19190((1S,2R,10S,11S,14R,15S,17S)-14,17-dihydroxy-14-(2-...)
Affinity DataIC50: 12.6nMAssay Description:Displacement of fluorescent labelled Dexamethasone from glucocorticoid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50412606(CHEMBL462282)
Affinity DataIC50: 12.6nMAssay Description:Displacement of fluorescent labelled Dexamethasone from glucocorticoid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50412608(CHEMBL519947)
Affinity DataIC50: 15.8nMAssay Description:Displacement of fluorescent labelled Dexamethasone from glucocorticoid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50412616(CHEMBL465927)
Affinity DataIC50: 15.8nMAssay Description:Displacement of fluorescent labelled Dexamethasone from glucocorticoid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50254760(5-amino-N-(2-((2,6-difluoro-N-(2-hydroxyethyl)benz...)
Affinity DataIC50: 15.8nMAssay Description:Displacement of fluorescent labelled Dexamethasone from glucocorticoid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50254759((+/-)-5-amino-N-(2-((2,6-difluoro-N-(2-fluoroethyl...)
Affinity DataIC50: 19.9nMAssay Description:Displacement of fluorescent labelled Dexamethasone from glucocorticoid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50412606(CHEMBL462282)
Affinity DataEC50:  19.9nMAssay Description:Agonist activity at human glucocorticoid receptor in human A549 cells assessed as transcriptional activity by MMTV luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50412611(CHEMBL479431)
Affinity DataIC50: 19.9nMAssay Description:Displacement of fluorescent labelled Dexamethasone from glucocorticoid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50412616(CHEMBL465927)
Affinity DataEC50:  25.1nMAssay Description:Agonist activity at human glucocorticoid receptor in human A549 cells assessed as transcriptional activity by MMTV luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50412607(CHEMBL516033)
Affinity DataEC50:  25.1nMAssay Description:Agonist activity at human glucocorticoid receptor in human A549 cells assessed as transcriptional activity by MMTV luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50254679(N-(2-((5-amino-1-(4-fluorophenyl)-1H-pyrazole-4-ca...)
Affinity DataEC50:  39.8nMAssay Description:Agonist activity at human glucocorticoid receptor in human A549 cells assessed as transcriptional activity by MMTV luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50412613(CHEMBL481784)
Affinity DataIC50: 39.8nMAssay Description:Displacement of fluorescent labelled Dexamethasone from glucocorticoid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50412605(CHEMBL481185)
Affinity DataIC50: 50.1nMAssay Description:Displacement of fluorescent labelled Dexamethasone from glucocorticoid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50412605(CHEMBL481185)
Affinity DataEC50:  50.1nMAssay Description:Agonist activity at human glucocorticoid receptor in human A549 cells assessed as transcriptional activity by MMTV luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50412605(CHEMBL481185)
Affinity DataIC50: 50.1nMAssay Description:Displacement of fluorescent labelled Dexamethasone from glucocorticoid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50412609(CHEMBL520750)
Affinity DataEC50:  50.1nMAssay Description:Agonist activity at human glucocorticoid receptor in human A549 cells assessed as transcriptional activity by MMTV luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50412605(CHEMBL481185)
Affinity DataEC50:  50.1nMAssay Description:Agonist activity at human glucocorticoid receptor in human A549 cells assessed as transcriptional activity by MMTV luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50412612(CHEMBL518451)
Affinity DataEC50:  50.1nMAssay Description:Agonist activity at human glucocorticoid receptor in human A549 cells assessed as transcriptional activity by MMTV luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM19190((1S,2R,10S,11S,14R,15S,17S)-14,17-dihydroxy-14-(2-...)
Affinity DataEC50:  50.1nMAssay Description:Agonist activity at human glucocorticoid receptor in human A549 cells assessed as transcriptional activity by MMTV luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50412607(CHEMBL516033)
Affinity DataIC50: 50.1nMAssay Description:Displacement of fluorescent labelled Dexamethasone from glucocorticoid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50254760(5-amino-N-(2-((2,6-difluoro-N-(2-hydroxyethyl)benz...)
Affinity DataEC50:  50.1nMAssay Description:Agonist activity at human glucocorticoid receptor in human A549 cells assessed as transcriptional activity by MMTV luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50254759((+/-)-5-amino-N-(2-((2,6-difluoro-N-(2-fluoroethyl...)
Affinity DataEC50:  50.1nMAssay Description:Agonist activity at human glucocorticoid receptor in human A549 cells assessed as transcriptional activity by MMTV luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50254465((+/-)-5-amino-N-(2-((N-ethyl-2-(methylsulfonyl)ben...)
Affinity DataIC50: 63.1nMAssay Description:Displacement of fluorescent labelled Dexamethasone from glucocorticoid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50254723((+/-)-5-amino-N-(2-((2,6-difluoro-N-methylbenzamid...)
Affinity DataIC50: 79.4nMAssay Description:Displacement of fluorescent labelled Dexamethasone from glucocorticoid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50412605(CHEMBL481185)
Affinity DataIC50: 125nMAssay Description:Displacement of fluorescent labelled Dexamethasone from glucocorticoid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50254465((+/-)-5-amino-N-(2-((N-ethyl-2-(methylsulfonyl)ben...)
Affinity DataEC50:  158nMAssay Description:Agonist activity at human glucocorticoid receptor in human A549 cells assessed as transcriptional activity by MMTV luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50412608(CHEMBL519947)
Affinity DataEC50:  251nMAssay Description:Agonist activity at human glucocorticoid receptor in human A549 cells assessed as transcriptional activity by MMTV luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50254723((+/-)-5-amino-N-(2-((2,6-difluoro-N-methylbenzamid...)
Affinity DataEC50:  251nMAssay Description:Agonist activity at human glucocorticoid receptor in human A549 cells assessed as transcriptional activity by MMTV luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50412611(CHEMBL479431)
Affinity DataEC50:  316nMAssay Description:Agonist activity at human glucocorticoid receptor in human A549 cells assessed as transcriptional activity by MMTV luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50412610(CHEMBL480800)
Affinity DataIC50: 316nMAssay Description:Displacement of fluorescent labelled Dexamethasone from glucocorticoid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50412615(CHEMBL465920)
Affinity DataIC50: 398nMAssay Description:Displacement of fluorescent labelled Dexamethasone from glucocorticoid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50254759((+/-)-5-amino-N-(2-((2,6-difluoro-N-(2-fluoroethyl...)
Affinity DataIC50: 500nMAssay Description:Inhibition of CYP3A4More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50254466(5-amino-N-(2-((2,6-dichloro-N-ethylbenzamido)methy...)
Affinity DataIC50: 700nMAssay Description:Inhibition of CYP3A4More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50412613(CHEMBL481784)
Affinity DataEC50:  794nMAssay Description:Agonist activity at human glucocorticoid receptor in human A549 cells assessed as transcriptional activity by MMTV luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCytochrome P450 2C9(Human)
Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50254466(5-amino-N-(2-((2,6-dichloro-N-ethylbenzamido)methy...)
Affinity DataIC50: 800nMAssay Description:Inhibition of CYP2C9More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50254464(5-amino-N-(2-((2-chloro-N-ethylbenzamido)methyl)-3...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of CYP3A4More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50254464(5-amino-N-(2-((2-chloro-N-ethylbenzamido)methyl)-3...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of CYP3A4More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50254513(5-amino-N-(2-((N-ethyl-2,6-difluorobenzamido)methy...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of CYP3A4More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50254465((+/-)-5-amino-N-(2-((N-ethyl-2-(methylsulfonyl)ben...)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of CYP3A4More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCytochrome P450 2C9(Human)
Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50254761(5-amino-N-(2-((2,6-dichloro-N-(2-hydroxyethyl)benz...)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of CYP2C9More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
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