Compile Data Set for Download or QSAR
Report error Found 46 Enz. Inhib. hit(s) with all data for entry = 50028007
TargetTyrosine-protein kinase Lck(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50255312(2-(5-((dimethylamino)methyl)-2-methoxyphenyl)-4-(4...)
Affinity DataIC50: 6nMAssay Description:Inhibition of LckMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50239328(2-(3-((dimethylamino)methyl)phenyl)-4-(4-methyl-1H...)
Affinity DataIC50: 7.5nMAssay Description:Inhibition of human full length PKCthetaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50255312(2-(5-((dimethylamino)methyl)-2-methoxyphenyl)-4-(4...)
Affinity DataIC50: 8.70nMAssay Description:Inhibition of human full length PKCthetaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50255313(2-(5-((dimethylamino)methyl)-2-ethoxyphenyl)-4-(4-...)
Affinity DataIC50: 9.20nMAssay Description:Inhibition of human full length PKCthetaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50255315(2-(3-((dimethylamino)methyl)-2-methoxyphenyl)-4-(4...)
Affinity DataIC50: 12nMAssay Description:Inhibition of human full length PKCthetaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50256031(2-(4-((dimethylamino)methyl)phenyl)-4-(4-methyl-1H...)
Affinity DataIC50: 14nMAssay Description:Inhibition of human full length PKCthetaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50255252(2-(5-((dimethylamino)methyl)thiophen-3-yl)-4-(4-me...)
Affinity DataIC50: 16nMAssay Description:Inhibition of human full length PKCthetaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50255367(2-(2-((dimethylamino)methyl)-5-methoxyphenyl)-4-(4...)
Affinity DataIC50: 16nMAssay Description:Inhibition of human full length PKCthetaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lyn(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50255312(2-(5-((dimethylamino)methyl)-2-methoxyphenyl)-4-(4...)
Affinity DataIC50: 23nMAssay Description:Inhibition of LynMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50255254(2-(2-methoxyphenyl)-4-(4-methyl-1H-indol-5-ylamino...)
Affinity DataIC50: 23nMAssay Description:Inhibition of human full length PKCthetaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50255312(2-(5-((dimethylamino)methyl)-2-methoxyphenyl)-4-(4...)
Affinity DataIC50: 24nMAssay Description:Inhibition of human full length PKCdeltaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50239328(2-(3-((dimethylamino)methyl)phenyl)-4-(4-methyl-1H...)
Affinity DataIC50: 26nMAssay Description:Inhibition of human full length PKCdeltaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50255315(2-(3-((dimethylamino)methyl)-2-methoxyphenyl)-4-(4...)
Affinity DataIC50: 27nMAssay Description:Inhibition of human full length PKCdeltaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50239328(2-(3-((dimethylamino)methyl)phenyl)-4-(4-methyl-1H...)
Affinity DataIC50: 28nMAssay Description:Inhibition of LckMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50255252(2-(5-((dimethylamino)methyl)thiophen-3-yl)-4-(4-me...)
Affinity DataIC50: 51nMAssay Description:Inhibition of human full length PKCdeltaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50239331(4-(1H-indol-5-ylamino)-2-phenylthieno[2,3-b]pyridi...)
Affinity DataIC50: 52nMAssay Description:Inhibition of human full length PKCthetaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lyn(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50255313(2-(5-((dimethylamino)methyl)-2-ethoxyphenyl)-4-(4-...)
Affinity DataIC50: 74nMAssay Description:Inhibition of LynMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50255313(2-(5-((dimethylamino)methyl)-2-ethoxyphenyl)-4-(4-...)
Affinity DataIC50: 82nMAssay Description:Inhibition of human full length PKCdeltaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50255253(2-(5-((dimethylamino)methyl)pyridin-3-yl)-4-(4-met...)
Affinity DataIC50: 84nMAssay Description:Inhibition of human full length PKCthetaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50256031(2-(4-((dimethylamino)methyl)phenyl)-4-(4-methyl-1H...)
Affinity DataIC50: 88nMAssay Description:Inhibition of human full length PKCdeltaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50255251(2-(2-((dimethylamino)methyl)phenyl)-4-(4-methyl-1H...)
Affinity DataIC50: 93nMAssay Description:Inhibition of human full length PKCthetaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lyn(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50256031(2-(4-((dimethylamino)methyl)phenyl)-4-(4-methyl-1H...)
Affinity DataIC50: 100nMAssay Description:Inhibition of LynMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50255314(2-(5-((dimethylamino)methyl)-2-methylphenyl)-4-(4-...)
Affinity DataIC50: 100nMAssay Description:Inhibition of human full length PKCthetaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50255367(2-(2-((dimethylamino)methyl)-5-methoxyphenyl)-4-(4...)
Affinity DataIC50: 130nMAssay Description:Inhibition of human full length PKCdeltaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50255253(2-(5-((dimethylamino)methyl)pyridin-3-yl)-4-(4-met...)
Affinity DataIC50: 170nMAssay Description:Inhibition of human full length PKCdeltaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lyn(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50255314(2-(5-((dimethylamino)methyl)-2-methylphenyl)-4-(4-...)
Affinity DataIC50: 230nMAssay Description:Inhibition of LynMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50255254(2-(2-methoxyphenyl)-4-(4-methyl-1H-indol-5-ylamino...)
Affinity DataIC50: 250nMAssay Description:Inhibition of human full length PKCdeltaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lyn(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50255254(2-(2-methoxyphenyl)-4-(4-methyl-1H-indol-5-ylamino...)
Affinity DataIC50: 310nMAssay Description:Inhibition of LynMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50239331(4-(1H-indol-5-ylamino)-2-phenylthieno[2,3-b]pyridi...)
Affinity DataIC50: 370nMAssay Description:Inhibition of human full length PKCdeltaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50255251(2-(2-((dimethylamino)methyl)phenyl)-4-(4-methyl-1H...)
Affinity DataIC50: 380nMAssay Description:Inhibition of human full length PKCdeltaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lyn(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50255252(2-(5-((dimethylamino)methyl)thiophen-3-yl)-4-(4-me...)
Affinity DataIC50: 410nMAssay Description:Inhibition of LynMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50255314(2-(5-((dimethylamino)methyl)-2-methylphenyl)-4-(4-...)
Affinity DataIC50: 410nMAssay Description:Inhibition of human full length PKCdeltaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lyn(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50239328(2-(3-((dimethylamino)methyl)phenyl)-4-(4-methyl-1H...)
Affinity DataIC50: 520nMAssay Description:Inhibition of LynMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lyn(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50255315(2-(3-((dimethylamino)methyl)-2-methoxyphenyl)-4-(4...)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of LynMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lyn(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50255253(2-(5-((dimethylamino)methyl)pyridin-3-yl)-4-(4-met...)
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of LynMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lyn(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50239331(4-(1H-indol-5-ylamino)-2-phenylthieno[2,3-b]pyridi...)
Affinity DataIC50: 3.40E+3nMAssay Description:Inhibition of LynMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase Fyn(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50255367(2-(2-((dimethylamino)methyl)-5-methoxyphenyl)-4-(4...)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of FynMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase HCK(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50255367(2-(2-((dimethylamino)methyl)-5-methoxyphenyl)-4-(4...)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of HckMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50255367(2-(2-((dimethylamino)methyl)-5-methoxyphenyl)-4-(4...)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of MK2More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50255367(2-(2-((dimethylamino)methyl)-5-methoxyphenyl)-4-(4...)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of SrcMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lyn(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50255367(2-(2-((dimethylamino)methyl)-5-methoxyphenyl)-4-(4...)
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of LynMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProtein kinase C beta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50255367(2-(2-((dimethylamino)methyl)-5-methoxyphenyl)-4-(4...)
Affinity DataIC50: 2.20E+4nMAssay Description:Inhibition of human full length PKCbetaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lyn(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50255251(2-(2-((dimethylamino)methyl)phenyl)-4-(4-methyl-1H...)
Affinity DataIC50: 3.70E+4nMAssay Description:Inhibition of LynMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50255367(2-(2-((dimethylamino)methyl)-5-methoxyphenyl)-4-(4...)
Affinity DataIC50: 3.80E+4nMAssay Description:Inhibition of LckMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProtein kinase C epsilon type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50255367(2-(2-((dimethylamino)methyl)-5-methoxyphenyl)-4-(4...)
Affinity DataIC50: 9.50E+4nMAssay Description:Inhibition of human full length PKCepsilonMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProtein kinase C eta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50255367(2-(2-((dimethylamino)methyl)-5-methoxyphenyl)-4-(4...)
Affinity DataIC50: 3.60E+5nMAssay Description:Inhibition of human full length PKCetaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed