Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 50038805
TargetSerine/threonine-protein kinase pim-1(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50059889(3-methoxy-2-methyl-4-methylamino-(2S,3S,4S,6R)-29-...)
Affinity DataIC50: 10nMAssay Description:Inhibition of human recombinant Pim1 expressed in insect cells by HTRFMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2012
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM2681(3-{1-[3-(dimethylamino)propyl]-1H-indol-3-yl}-4-(1...)
Affinity DataIC50: 150nMAssay Description:Inhibition of human recombinant Pim1 expressed in insect cells by HTRFMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2012
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50267091(N-(2-(1H-indol-3-yl)ethyl)-4-chloro-N-(9-methyl-9-...)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of human recombinant Pim1 expressed in insect cells by HTRFMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2012
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50267023(1-(2-(1H-indol-3-yl)ethyl)-4-acetyl-5-(4-ethylphen...)
Affinity DataKi:  2.10E+3nMAssay Description:Inhibition of human recombinant Pim1 expressed in insect cells by HTRFMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2012
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50267025(BAS-8770954 | 1-(2-(1H-indol-3-yl)ethyl)-4-acetyl-...)
Affinity DataKi:  2.20E+3nMAssay Description:Inhibition of human recombinant Pim1 expressed in insect cells by HTRFMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2012
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50267089(LY-294002 | 2-morpholino-8-phenylchroman-4-one | C...)
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of human recombinant Pim1 expressed in insect cells by HTRFMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2012
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50267024(1-(2-(1H-indol-3-yl)ethyl)-4-acetyl-5-(4-ethoxyphe...)
Affinity DataKi:  4.20E+3nMAssay Description:Inhibition of human recombinant Pim1 expressed in insect cells by HTRFMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2012
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50267053(BAS-8770949 | 1-(2-(1H-indol-3-yl)ethyl)-4-acetyl-...)
Affinity DataKi:  4.50E+3nMAssay Description:Inhibition of human recombinant Pim1 expressed in insect cells by HTRFMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2012
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50267090(2-(3-(9H-carbazol-9-yl)-2-hydroxypropoxy)benzaldeh...)
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibition of human recombinant Pim1 expressed in insect cells by HTRFMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2012
Entry Details Article
PubMed