Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with all data for entry = 50004482
TargetBifunctional protein GlmU(Escherichia coli (strain K12))
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50294336(5-amino-2-(4-aminophenylamino)benzenesulfonic acid...)
Affinity DataKi:  17nMAssay Description:Competitive inhibition of Acetyltransferase activity of Escherichia coli BL21(DE3) GlmU in presence of AcCoAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
TargetBifunctional protein GlmU(Escherichia coli (strain K12))
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50483325(Mac0029665 | CHEMBL1652297)
Affinity DataKi:  23nMAssay Description:Competitive inhibition of Acetyltransferase activity of Escherichia coli BL21(DE3) GlmU in presence of AcCoAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
TargetBifunctional protein GlmU(Escherichia coli (strain K12))
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50483326(Mac0008028 | CHEMBL1652296)
Affinity DataKi:  404nMAssay Description:Competitive inhibition of Acetyltransferase activity of Escherichia coli BL21(DE3) GlmU in presence of AcCoAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed