Compile Data Set for Download or QSAR
Report error Found 71 Enz. Inhib. hit(s) with all data for entry = 50028669
TargetAlpha-1D adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50259485(6-(2-(methoxymethyl)phenyl)-4,5,6,7-tetrahydro-1H-...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human cloned adrenergic Alpha-1D receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50259381(6-phenyl-6,7-di hydro-5H-pyrrolo[1,2-a]imidazole |...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human cloned adrenergic Alpha-1B receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50259333(6-phenyl-4,5,6,7-tetra hydro-1H-benzo[d]imidazole ...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human cloned adrenergic Alpha-1B receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50259332(2-(2,3-dihydro-1H-inden-2-yl)-1H-imidazole | CHEMB...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human cloned adrenergic Alpha-1B receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238822(2-(2,3-dihydro-1H-inden-1-yl)-1H-imidazole | CHEMB...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human cloned adrenergic Alpha-1B receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50259534(6-(2-fluorophenyl)-6,7-dihydro-5H-pyrrolo[1,2-a]im...)
Affinity DataEC50:  301nMAssay Description:Agonist activity at human cloned adrenergic Alpha-1D receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50259489(6-(3-methoxyphenyl)-6,7-dihydro-5H-pyrrolo[1,2-a]i...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human cloned adrenergic Alpha-1D receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50259487(6-(4-chlorophenyl)-6,7-dihydro-5H-pyrrolo[1,2-a]im...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human cloned adrenergic Alpha-1D receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50259486(6-(2-chlorophenyl)-6,7-dihydro-5H-pyrrolo[1,2-a]im...)
Affinity DataEC50:  364nMAssay Description:Agonist activity at human cloned adrenergic Alpha-1D receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50259382(6-phenyl-5,6,7,8-tetrahydroimidazo[1,2-a]pyridine ...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human cloned adrenergic Alpha-1B receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50259484(6-(4-methoxyphenyl)-4,5,6,7-tetrahydro-1H-benzo[d]...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human cloned adrenergic Alpha-1D receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50259387(6-(3-methoxyphenyl)-4,5,6,7-tetrahydro-1H-benzo[d]...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human cloned adrenergic Alpha-1D receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50259386(6-(2-methoxyphenyl)-4,5,6,7-tetrahydro-1H-benzo[d]...)
Affinity DataEC50:  3.50E+3nMAssay Description:Agonist activity at human cloned adrenergic Alpha-1D receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50259385(6-(4-chlorophenyl)-4,5,6,7-tetrahydro-1H-benzo[d]i...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human cloned adrenergic Alpha-1D receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50259384(6-(3-chlorophenyl)-4,5,6,7-tetrahydro-1H-benzo[d]i...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human cloned adrenergic Alpha-1D receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50259383(6-(2-chlorophenyl)-4,5,6,7-tetrahydro-1H-benzo[d]i...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human cloned adrenergic Alpha-1D receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50259382(6-phenyl-5,6,7,8-tetrahydroimidazo[1,2-a]pyridine ...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human cloned adrenergic Alpha-1D receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50259381(6-phenyl-6,7-di hydro-5H-pyrrolo[1,2-a]imidazole |...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human cloned adrenergic Alpha-1D receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50259487(6-(4-chlorophenyl)-6,7-dihydro-5H-pyrrolo[1,2-a]im...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human cloned adrenergic Alpha-1B receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50259381(6-phenyl-6,7-di hydro-5H-pyrrolo[1,2-a]imidazole |...)
Affinity DataEC50:  7.36E+3nMAssay Description:Agonist activity at human cloned adrenergic Alpha-1D receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50259333(6-phenyl-4,5,6,7-tetra hydro-1H-benzo[d]imidazole ...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human cloned adrenergic Alpha-1D receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50259332(2-(2,3-dihydro-1H-inden-2-yl)-1H-imidazole | CHEMB...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human cloned adrenergic Alpha-1D receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238822(2-(2,3-dihydro-1H-inden-1-yl)-1H-imidazole | CHEMB...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human cloned adrenergic Alpha-1D receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50259538(6-(2-(methoxymethyl)phenyl)-6,7-dihydro-5H-pyrrolo...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human cloned adrenergic Alpha-1B receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50259537(2-(6,7-dihydro-5H-pyrrolo[1,2-a]imidazol-6-yl)benz...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human cloned adrenergic Alpha-1B receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50259534(6-(2-fluorophenyl)-6,7-dihydro-5H-pyrrolo[1,2-a]im...)
Affinity DataEC50:  1.77E+3nMAssay Description:Agonist activity at human cloned adrenergic Alpha-1B receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50259489(6-(3-methoxyphenyl)-6,7-dihydro-5H-pyrrolo[1,2-a]i...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human cloned adrenergic Alpha-1B receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50259382(6-phenyl-5,6,7,8-tetrahydroimidazo[1,2-a]pyridine ...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human cloned adrenergic alpha2A receptor expressed in CHOK1 cells by beta-lactamase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50259486(6-(2-chlorophenyl)-6,7-dihydro-5H-pyrrolo[1,2-a]im...)
Affinity DataEC50:  1.10E+3nMAssay Description:Agonist activity at human cloned adrenergic Alpha-1B receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50259485(6-(2-(methoxymethyl)phenyl)-4,5,6,7-tetrahydro-1H-...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human cloned adrenergic Alpha-1B receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50259484(6-(4-methoxyphenyl)-4,5,6,7-tetrahydro-1H-benzo[d]...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human cloned adrenergic Alpha-1B receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50259387(6-(3-methoxyphenyl)-4,5,6,7-tetrahydro-1H-benzo[d]...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human cloned adrenergic Alpha-1B receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50259386(6-(2-methoxyphenyl)-4,5,6,7-tetrahydro-1H-benzo[d]...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human cloned adrenergic Alpha-1B receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50259385(6-(4-chlorophenyl)-4,5,6,7-tetrahydro-1H-benzo[d]i...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human cloned adrenergic Alpha-1B receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50259384(6-(3-chlorophenyl)-4,5,6,7-tetrahydro-1H-benzo[d]i...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human cloned adrenergic Alpha-1B receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50259383(6-(2-chlorophenyl)-4,5,6,7-tetrahydro-1H-benzo[d]i...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human cloned adrenergic Alpha-1B receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50259386(6-(2-methoxyphenyl)-4,5,6,7-tetrahydro-1H-benzo[d]...)
Affinity DataEC50:  144nMAssay Description:Agonist activity at human cloned adrenergic alpha1A receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50259488(6-(2-methoxyphenyl)-6,7-dihydro-5H-pyrrolo[1,2-a]i...)
Affinity DataEC50:  22nMAssay Description:Agonist activity at human cloned adrenergic alpha1A receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50259487(6-(4-chlorophenyl)-6,7-dihydro-5H-pyrrolo[1,2-a]im...)
Affinity DataEC50:  3.46E+3nMAssay Description:Agonist activity at human cloned adrenergic alpha1A receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50259486(6-(2-chlorophenyl)-6,7-dihydro-5H-pyrrolo[1,2-a]im...)
Affinity DataEC50:  19nMAssay Description:Agonist activity at human cloned adrenergic alpha1A receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50259381(6-phenyl-6,7-di hydro-5H-pyrrolo[1,2-a]imidazole |...)
Affinity DataEC50:  83nMAssay Description:Agonist activity at human cloned adrenergic alpha1A receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50259485(6-(2-(methoxymethyl)phenyl)-4,5,6,7-tetrahydro-1H-...)
Affinity DataEC50:  76nMAssay Description:Agonist activity at human cloned adrenergic alpha1A receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50259485(6-(2-(methoxymethyl)phenyl)-4,5,6,7-tetrahydro-1H-...)
Affinity DataEC50:  76nMAssay Description:Agonist activity at human cloned adrenergic alpha1A receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50259484(6-(4-methoxyphenyl)-4,5,6,7-tetrahydro-1H-benzo[d]...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human cloned adrenergic alpha1A receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50259387(6-(3-methoxyphenyl)-4,5,6,7-tetrahydro-1H-benzo[d]...)
Affinity DataEC50:  1.05E+3nMAssay Description:Agonist activity at human cloned adrenergic alpha1A receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50259489(6-(3-methoxyphenyl)-6,7-dihydro-5H-pyrrolo[1,2-a]i...)
Affinity DataEC50:  578nMAssay Description:Agonist activity at human cloned adrenergic alpha1A receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50259385(6-(4-chlorophenyl)-4,5,6,7-tetrahydro-1H-benzo[d]i...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human cloned adrenergic alpha1A receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50259384(6-(3-chlorophenyl)-4,5,6,7-tetrahydro-1H-benzo[d]i...)
Affinity DataEC50:  514nMAssay Description:Agonist activity at human cloned adrenergic alpha1A receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50259383(6-(2-chlorophenyl)-4,5,6,7-tetrahydro-1H-benzo[d]i...)
Affinity DataEC50:  276nMAssay Description:Agonist activity at human cloned adrenergic alpha1A receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50259382(6-phenyl-5,6,7,8-tetrahydroimidazo[1,2-a]pyridine ...)
Affinity DataEC50:  721nMAssay Description:Agonist activity at human cloned adrenergic alpha1A receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
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