Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 50028674
TargetSodium channel protein type 2 subunit alpha(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50259542(2-(3-Trifluoromethylphenyl)-4(5)-(3-trifluoromethy...)
Affinity DataIC50: 200nMAssay Description:Inhibition of human Nav1.2 channel expressed in HEK cells by patch-clamp electrophysiology methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetSodium channel protein type 2 subunit alpha(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50259490(2-Phenyl-4(5)-(4-trifluoromethylphenyl)imidazole |...)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of human Nav1.2 channel expressed in HEK cells by patch-clamp electrophysiology methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetSodium channel protein type 2 subunit alpha(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50259388(2-(4-Chlorophenyl)-4(5)-phenylimidazole | CHEMBL50...)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of human Nav1.2 channel expressed in HEK cells by patch-clamp electrophysiology methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetSodium channel protein type 2 subunit alpha(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50259541(2-(4-Nitrophenyl)-4(5)-(3-trifluoromethylphenyl)-i...)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of human Nav1.2 channel expressed in HEK cells by patch-clamp electrophysiology methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetSodium channel protein type 2 subunit alpha(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50145044(2-Phenyl-4(5)-(3-trifluoromethylphenyl)imidazole |...)
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of human Nav1.2 channel expressed in HEK cells by patch-clamp electrophysiology methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetSodium channel protein type 2 subunit alpha(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50133778(2,5-Diphenyl-1H-imidazole | 2,4(5)-Diphenylimidazo...)
Affinity DataIC50: 4.06E+4nMAssay Description:Inhibition of human Nav1.2 channel expressed in HEK cells by patch-clamp electrophysiology methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetSodium channel protein type 2 subunit alpha(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50259540(2-(4-Chlorophenyl)-4(5)-(3-trifluoromethylphenyl)-...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human Nav1.2 channel expressed in HEK cells by patch-clamp electrophysiology methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetSodium channel protein type 2 subunit alpha(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50031299(CHEMBL741 | BW-430C | 6-(2,3-Dichloro-phenyl)-[1,2...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human Nav1.2 channel expressed in HEK cells by patch-clamp electrophysiology methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetSodium channel protein type 2 subunit alpha(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50003655(Phenytoin)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human Nav1.2 channel expressed in HEK cells by patch-clamp electrophysiology methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed