Compile Data Set for Download or QSAR
Report error Found 45 Enz. Inhib. hit(s) with all data for entry = 3258
TargetNociceptin receptor(Human)
Banyu Pharmaceutical

LigandPNGBDBM29988(benzimidazole analogue, 7h | benzimidazole derivat...)
Affinity DataIC50: 0.810nM EC50:  1.30nMpH: 7.4 T: 2°CAssay Description:Compounds were tested for their inhibitory effects on ligand binding to the human ORL1 receptor. Bound and free radioligands are separated by filtra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2009
Entry Details Article
PubMed
TargetNociceptin receptor(Human)
Banyu Pharmaceutical

LigandPNGBDBM30012(benzimidazole analogue, 7k)
Affinity DataIC50: 1nM EC50:  1.10nMpH: 7.4 T: 2°CAssay Description:Compounds were tested for their inhibitory effects on ligand binding to the human ORL1 receptor. Bound and free radioligands are separated by filtra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2009
Entry Details Article
PubMed
TargetNociceptin receptor(Human)
Banyu Pharmaceutical

LigandPNGBDBM30017(benzimidazole analogue, 7p)
Affinity DataIC50: 1.10nM EC50:  0.590nMpH: 7.4 T: 2°CAssay Description:Compounds were tested for their inhibitory effects on ligand binding to the human ORL1 receptor. Bound and free radioligands are separated by filtra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2009
Entry Details Article
PubMed
TargetNociceptin receptor(Human)
Banyu Pharmaceutical

LigandPNGBDBM30011(benzimidazole analogue, 7j)
Affinity DataIC50: 1.40nM EC50:  0.550nMpH: 7.4 T: 2°CAssay Description:Compounds were tested for their inhibitory effects on ligand binding to the human ORL1 receptor. Bound and free radioligands are separated by filtra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2009
Entry Details Article
PubMed
TargetNociceptin receptor(Human)
Banyu Pharmaceutical

LigandPNGBDBM30016(benzimidazole analogue, 7o)
Affinity DataIC50: 1.70nM EC50:  0.910nMpH: 7.4 T: 2°CAssay Description:Compounds were tested for their inhibitory effects on ligand binding to the human ORL1 receptor. Bound and free radioligands are separated by filtra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2009
Entry Details Article
PubMed
TargetNociceptin receptor(Human)
Banyu Pharmaceutical

LigandPNGBDBM30018(benzimidazole analogue, 7q)
Affinity DataIC50: 1.80nM EC50:  7.10nMpH: 7.4 T: 2°CAssay Description:Compounds were tested for their inhibitory effects on ligand binding to the human ORL1 receptor. Bound and free radioligands are separated by filtra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2009
Entry Details Article
PubMed
TargetNociceptin receptor(Human)
Banyu Pharmaceutical

LigandPNGBDBM30008(benzimidazole analogue, 7g)
Affinity DataIC50: 1.90nM EC50:  1.10nMpH: 7.4 T: 2°CAssay Description:Compounds were tested for their inhibitory effects on ligand binding to the human ORL1 receptor. Bound and free radioligands are separated by filtra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2009
Entry Details Article
PubMed
TargetNociceptin receptor(Human)
Banyu Pharmaceutical

LigandPNGBDBM30010(benzimidazole analogue, 7i)
Affinity DataIC50: 2.10nM EC50:  1.80nMpH: 7.4 T: 2°CAssay Description:Compounds were tested for their inhibitory effects on ligand binding to the human ORL1 receptor. Bound and free radioligands are separated by filtra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2009
Entry Details Article
PubMed
TargetNociceptin receptor(Human)
Banyu Pharmaceutical

LigandPNGBDBM30014(benzimidazole analogue, 7m)
Affinity DataIC50: 2.20nM EC50:  0.900nMpH: 7.4 T: 2°CAssay Description:Compounds were tested for their inhibitory effects on ligand binding to the human ORL1 receptor. Bound and free radioligands are separated by filtra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2009
Entry Details Article
PubMed
TargetNociceptin receptor(Human)
Banyu Pharmaceutical

LigandPNGBDBM29987(benzimidazole analogue, 7e | benzimidazole derivat...)
Affinity DataIC50: 2.40nM EC50:  0.720nMpH: 7.4 T: 2°CAssay Description:Compounds were tested for their inhibitory effects on ligand binding to the human ORL1 receptor. Bound and free radioligands are separated by filtra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2009
Entry Details Article
PubMed
TargetNociceptin receptor(Human)
Banyu Pharmaceutical

LigandPNGBDBM29995(CHEMBL494350 | benzimidazole-based antagonist, 1)
Affinity DataIC50: 2.60nM EC50:  0.650nMpH: 7.4 T: 2°CAssay Description:Compounds were tested for their inhibitory effects on ligand binding to the human ORL1 receptor. Bound and free radioligands are separated by filtra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2009
Entry Details Article
PubMed
TargetNociceptin receptor(Human)
Banyu Pharmaceutical

LigandPNGBDBM30004(benzimidazole analogue, 7c)
Affinity DataIC50: 4.30nM EC50:  1.10nMpH: 7.4 T: 2°CAssay Description:Compounds were tested for their inhibitory effects on ligand binding to the human ORL1 receptor. Bound and free radioligands are separated by filtra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2009
Entry Details Article
PubMed
TargetNociceptin receptor(Human)
Banyu Pharmaceutical

LigandPNGBDBM30013(benzimidazole analogue, 7l)
Affinity DataIC50: 6.90nM EC50:  4nMpH: 7.4 T: 2°CAssay Description:Compounds were tested for their inhibitory effects on ligand binding to the human ORL1 receptor. Bound and free radioligands are separated by filtra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2009
Entry Details Article
PubMed
TargetNociceptin receptor(Human)
Banyu Pharmaceutical

LigandPNGBDBM30015(benzimidazole analogue, 7n)
Affinity DataIC50: 7.40nM EC50:  3.70nMpH: 7.4 T: 2°CAssay Description:Compounds were tested for their inhibitory effects on ligand binding to the human ORL1 receptor. Bound and free radioligands are separated by filtra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2009
Entry Details Article
PubMed
TargetNociceptin receptor(Human)
Banyu Pharmaceutical

LigandPNGBDBM29996(benzimidazole analogue, 5a)
Affinity DataIC50: 9.20nM EC50:  2.90nMpH: 7.4 T: 2°CAssay Description:Compounds were tested for their inhibitory effects on ligand binding to the human ORL1 receptor. Bound and free radioligands are separated by filtra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2009
Entry Details Article
PubMed
TargetNociceptin receptor(Human)
Banyu Pharmaceutical

LigandPNGBDBM30005(benzimidazole analogue, 7d)
Affinity DataIC50: 9.5nM EC50:  2.10nMpH: 7.4 T: 2°CAssay Description:Compounds were tested for their inhibitory effects on ligand binding to the human ORL1 receptor. Bound and free radioligands are separated by filtra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2009
Entry Details Article
PubMed
TargetNociceptin receptor(Human)
Banyu Pharmaceutical

LigandPNGBDBM30007(Racemate | benzimidazole analogue, 7f)
Affinity DataIC50: 16nM EC50:  46nMpH: 7.4 T: 2°CAssay Description:Compounds were tested for their inhibitory effects on ligand binding to the human ORL1 receptor. Bound and free radioligands are separated by filtra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2009
Entry Details Article
PubMed
TargetNociceptin receptor(Human)
Banyu Pharmaceutical

LigandPNGBDBM30003(benzimidazole analogue, 7b)
Affinity DataIC50: 21nM EC50:  8.60nMpH: 7.4 T: 2°CAssay Description:Compounds were tested for their inhibitory effects on ligand binding to the human ORL1 receptor. Bound and free radioligands are separated by filtra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2009
Entry Details Article
PubMed
TargetNociceptin receptor(Human)
Banyu Pharmaceutical

LigandPNGBDBM30002(benzimidazole analogue, 7a)
Affinity DataIC50: 22nMpH: 7.4 T: 2°CAssay Description:Compounds were tested for their inhibitory effects on ligand binding to the human ORL1 receptor. Bound and free radioligands are separated by filtra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2009
Entry Details Article
PubMed
TargetNociceptin receptor(Human)
Banyu Pharmaceutical

LigandPNGBDBM29997(benzimidazole analogue, 5b)
Affinity DataIC50: 23nMpH: 7.4 T: 2°CAssay Description:Compounds were tested for their inhibitory effects on ligand binding to the human ORL1 receptor. Bound and free radioligands are separated by filtra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2009
Entry Details Article
PubMed
TargetNociceptin receptor(Human)
Banyu Pharmaceutical

LigandPNGBDBM30000(benzimidazole analogue, 5e)
Affinity DataIC50: 27nM EC50:  6.40nMpH: 7.4 T: 2°CAssay Description:Compounds were tested for their inhibitory effects on ligand binding to the human ORL1 receptor. Bound and free radioligands are separated by filtra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2009
Entry Details Article
PubMed
TargetNociceptin receptor(Human)
Banyu Pharmaceutical

LigandPNGBDBM30001(benzimidazole analogue, 5f)
Affinity DataIC50: 38nM EC50:  41nMpH: 7.4 T: 2°CAssay Description:Compounds were tested for their inhibitory effects on ligand binding to the human ORL1 receptor. Bound and free radioligands are separated by filtra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2009
Entry Details Article
PubMed
TargetNociceptin receptor(Human)
Banyu Pharmaceutical

LigandPNGBDBM29999(benzimidazole analogue, 5d)
Affinity DataIC50: 61nMpH: 7.4 T: 2°CAssay Description:Compounds were tested for their inhibitory effects on ligand binding to the human ORL1 receptor. Bound and free radioligands are separated by filtra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2009
Entry Details Article
PubMed
LigandPNGBDBM30016(benzimidazole analogue, 7o)
Affinity DataIC50: 380nMAssay Description:Compounds were tested for their inhibitory effects on ligand binding to the human ORL1 receptor. Bound and free radioligands are separated by filtra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2009
Entry Details Article
PubMed
TargetNociceptin receptor(Human)
Banyu Pharmaceutical

LigandPNGBDBM29998(benzimidazole analogue, 5c)
Affinity DataIC50: 630nMpH: 7.4 T: 2°CAssay Description:Compounds were tested for their inhibitory effects on ligand binding to the human ORL1 receptor. Bound and free radioligands are separated by filtra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2009
Entry Details Article
PubMed
LigandPNGBDBM29996(benzimidazole analogue, 5a)
Affinity DataIC50: 990nMAssay Description:Compounds were tested for their inhibitory effects on ligand binding to the human ORL1 receptor. Bound and free radioligands are separated by filtra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2009
Entry Details Article
PubMed
LigandPNGBDBM30005(benzimidazole analogue, 7d)
Affinity DataIC50: 1.50E+3nMAssay Description:Compounds were tested for their inhibitory effects on ligand binding to the human ORL1 receptor. Bound and free radioligands are separated by filtra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2009
Entry Details Article
PubMed
LigandPNGBDBM29995(CHEMBL494350 | benzimidazole-based antagonist, 1)
Affinity DataIC50: 1.60E+3nMAssay Description:Compounds were tested for their inhibitory effects on ligand binding to the human ORL1 receptor. Bound and free radioligands are separated by filtra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2009
Entry Details Article
PubMed
LigandPNGBDBM30007(Racemate | benzimidazole analogue, 7f)
Affinity DataIC50: 2.00E+3nMAssay Description:Compounds were tested for their inhibitory effects on ligand binding to the human ORL1 receptor. Bound and free radioligands are separated by filtra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2009
Entry Details Article
PubMed
LigandPNGBDBM30017(benzimidazole analogue, 7p)
Affinity DataIC50: 3.40E+3nMAssay Description:Compounds were tested for their inhibitory effects on ligand binding to the human ORL1 receptor. Bound and free radioligands are separated by filtra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2009
Entry Details Article
PubMed
LigandPNGBDBM29987(benzimidazole analogue, 7e | benzimidazole derivat...)
Affinity DataIC50: 3.50E+3nMAssay Description:Compounds were tested for their inhibitory effects on ligand binding to the human ORL1 receptor. Bound and free radioligands are separated by filtra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2009
Entry Details Article
PubMed
LigandPNGBDBM30004(benzimidazole analogue, 7c)
Affinity DataIC50: 3.90E+3nMAssay Description:Compounds were tested for their inhibitory effects on ligand binding to the human ORL1 receptor. Bound and free radioligands are separated by filtra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2009
Entry Details Article
PubMed
LigandPNGBDBM30014(benzimidazole analogue, 7m)
Affinity DataIC50: 4.40E+3nMAssay Description:Compounds were tested for their inhibitory effects on ligand binding to the human ORL1 receptor. Bound and free radioligands are separated by filtra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2009
Entry Details Article
PubMed
LigandPNGBDBM30015(benzimidazole analogue, 7n)
Affinity DataIC50: 6.30E+3nMAssay Description:Compounds were tested for their inhibitory effects on ligand binding to the human ORL1 receptor. Bound and free radioligands are separated by filtra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2009
Entry Details Article
PubMed
LigandPNGBDBM30001(benzimidazole analogue, 5f)
Affinity DataIC50: 1.00E+4nMAssay Description:Compounds were tested for their inhibitory effects on ligand binding to the human ORL1 receptor. Bound and free radioligands are separated by filtra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2009
Entry Details Article
PubMed
LigandPNGBDBM30000(benzimidazole analogue, 5e)
Affinity DataIC50: 1.00E+4nMAssay Description:Compounds were tested for their inhibitory effects on ligand binding to the human ORL1 receptor. Bound and free radioligands are separated by filtra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2009
Entry Details Article
PubMed
LigandPNGBDBM30008(benzimidazole analogue, 7g)
Affinity DataIC50: 1.00E+4nMAssay Description:Compounds were tested for their inhibitory effects on ligand binding to the human ORL1 receptor. Bound and free radioligands are separated by filtra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2009
Entry Details Article
PubMed
LigandPNGBDBM29988(benzimidazole analogue, 7h | benzimidazole derivat...)
Affinity DataIC50: 1.00E+4nMAssay Description:Compounds were tested for their inhibitory effects on ligand binding to the human ORL1 receptor. Bound and free radioligands are separated by filtra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2009
Entry Details Article
PubMed
LigandPNGBDBM30010(benzimidazole analogue, 7i)
Affinity DataIC50: 1.00E+4nMAssay Description:Compounds were tested for their inhibitory effects on ligand binding to the human ORL1 receptor. Bound and free radioligands are separated by filtra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2009
Entry Details Article
PubMed
LigandPNGBDBM30011(benzimidazole analogue, 7j)
Affinity DataIC50: 1.00E+4nMAssay Description:Compounds were tested for their inhibitory effects on ligand binding to the human ORL1 receptor. Bound and free radioligands are separated by filtra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2009
Entry Details Article
PubMed
LigandPNGBDBM30012(benzimidazole analogue, 7k)
Affinity DataIC50: 1.00E+4nMAssay Description:Compounds were tested for their inhibitory effects on ligand binding to the human ORL1 receptor. Bound and free radioligands are separated by filtra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2009
Entry Details Article
PubMed
LigandPNGBDBM30013(benzimidazole analogue, 7l)
Affinity DataIC50: 1.00E+4nMAssay Description:Compounds were tested for their inhibitory effects on ligand binding to the human ORL1 receptor. Bound and free radioligands are separated by filtra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2009
Entry Details Article
PubMed
LigandPNGBDBM29999(benzimidazole analogue, 5d)
Affinity DataIC50: 1.00E+4nMAssay Description:Compounds were tested for their inhibitory effects on ligand binding to the human ORL1 receptor. Bound and free radioligands are separated by filtra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2009
Entry Details Article
PubMed
LigandPNGBDBM29997(benzimidazole analogue, 5b)
Affinity DataIC50: 1.00E+4nMAssay Description:Compounds were tested for their inhibitory effects on ligand binding to the human ORL1 receptor. Bound and free radioligands are separated by filtra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2009
Entry Details Article
PubMed
LigandPNGBDBM30018(benzimidazole analogue, 7q)
Affinity DataIC50: 1.00E+4nMAssay Description:Compounds were tested for their inhibitory effects on ligand binding to the human ORL1 receptor. Bound and free radioligands are separated by filtra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2009
Entry Details Article
PubMed