Compile Data Set for Download or QSAR
Report error Found 53 Enz. Inhib. hit(s) with all data for entry = 3362
TargetAurora kinase A(Human)
Genentech

LigandPNGBDBM31093(cid_11712649 | 4-[[7-[2,6-bis(fluoranyl)phenyl]-9-...)
Affinity DataIC50: 1nMpH: 7.5 T: 2°CAssay Description:Aurora kinase was assayed in ELISA format using a GST fusion of the N-terminus of Histone H3 as substrate. Plates were coated with substrate, and the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2009
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Genentech

LigandPNGBDBM31837(Aurora Inhibitor, 35 | 2,4-Bisanilinopyrimidine, 1...)
Affinity DataIC50: 3.40nMpH: 7.5 T: 2°CAssay Description:Aurora kinase was assayed in ELISA format using a GST fusion of the N-terminus of Histone H3 as substrate. Plates were coated with substrate, and the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2009
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Genentech

LigandPNGBDBM31836(2,4-Bisanilinopyrimidine, 9)
Affinity DataIC50: 4.30nMpH: 7.5 T: 2°CAssay Description:Aurora kinase was assayed in ELISA format using a GST fusion of the N-terminus of Histone H3 as substrate. Plates were coated with substrate, and the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAurora kinase A(Human)
Genentech

LigandPNGBDBM31833(2,4-Bisanilinopyrimidine, 5)
Affinity DataIC50: 6nMpH: 7.5 T: 2°CAssay Description:Aurora kinase was assayed in ELISA format using a GST fusion of the N-terminus of Histone H3 as substrate. Plates were coated with substrate, and the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAurora kinase A(Human)
Genentech

LigandPNGBDBM31858(2,4-Bisanilinopyrimidine, 23)
Affinity DataIC50: 8nMAssay Description:Aurora kinase was assayed in ELISA format using a GST fusion of the N-terminus of Histone H3 as substrate. Plates were coated with substrate, and the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2009
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Genentech

LigandPNGBDBM31842(2,4-Bisanilinopyrimidine, 49)
Affinity DataIC50: 9nMpH: 7.5 T: 2°CAssay Description:Aurora kinase was assayed in ELISA format using a GST fusion of the N-terminus of Histone H3 as substrate. Plates were coated with substrate, and the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2009
Entry Details Article
PubMed
TargetAurora kinase B(Human)
Genentech

LigandPNGBDBM31093(cid_11712649 | 4-[[7-[2,6-bis(fluoranyl)phenyl]-9-...)
Affinity DataIC50: 9.30nMpH: 7.5 T: 2°CAssay Description:Aurora kinase was assayed in ELISA format using a GST fusion of the N-terminus of Histone H3 as substrate. Plates were coated with substrate, and the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2009
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Genentech

LigandPNGBDBM31834(2,4-Bisanilinopyrimidine, 13)
Affinity DataIC50: 10nMpH: 7.5 T: 2°CAssay Description:Aurora kinase was assayed in ELISA format using a GST fusion of the N-terminus of Histone H3 as substrate. Plates were coated with substrate, and the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2009
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Genentech

LigandPNGBDBM31841(2,4-Bisanilinopyrimidine, 48)
Affinity DataIC50: 13nMpH: 7.5 T: 2°CAssay Description:Aurora kinase was assayed in ELISA format using a GST fusion of the N-terminus of Histone H3 as substrate. Plates were coated with substrate, and the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2009
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Genentech

LigandPNGBDBM31876(2,4-Bisanilinopyrimidine, 42)
Affinity DataIC50: 14nMAssay Description:Aurora kinase was assayed in ELISA format using a GST fusion of the N-terminus of Histone H3 as substrate. Plates were coated with substrate, and the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2009
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Genentech

LigandPNGBDBM31848(2,4-Bisanilinopyrimidine, 55)
Affinity DataIC50: 14nMpH: 7.5 T: 2°CAssay Description:Aurora kinase was assayed in ELISA format using a GST fusion of the N-terminus of Histone H3 as substrate. Plates were coated with substrate, and the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2009
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Genentech

LigandPNGBDBM31859(2,4-Bisanilinopyrimidine, 24)
Affinity DataIC50: 14nMAssay Description:Aurora kinase was assayed in ELISA format using a GST fusion of the N-terminus of Histone H3 as substrate. Plates were coated with substrate, and the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2009
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Genentech

LigandPNGBDBM31847(2,4-Bisanilinopyrimidine, 54)
Affinity DataIC50: 18nMpH: 7.5 T: 2°CAssay Description:Aurora kinase was assayed in ELISA format using a GST fusion of the N-terminus of Histone H3 as substrate. Plates were coated with substrate, and the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2009
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Genentech

LigandPNGBDBM31840(2,4-Bisanilinopyrimidine, 47)
Affinity DataIC50: 19nMpH: 7.5 T: 2°CAssay Description:Aurora kinase was assayed in ELISA format using a GST fusion of the N-terminus of Histone H3 as substrate. Plates were coated with substrate, and the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2009
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Genentech

LigandPNGBDBM31873(2,4-Bisanilinopyrimidine, 39)
Affinity DataIC50: 19nMAssay Description:Aurora kinase was assayed in ELISA format using a GST fusion of the N-terminus of Histone H3 as substrate. Plates were coated with substrate, and the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2009
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Genentech

LigandPNGBDBM31877(2,4-Bisanilinopyrimidine, 43)
Affinity DataIC50: 20nMAssay Description:Aurora kinase was assayed in ELISA format using a GST fusion of the N-terminus of Histone H3 as substrate. Plates were coated with substrate, and the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2009
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Genentech

LigandPNGBDBM31863(2,4-Bisanilinopyrimidine, 29)
Affinity DataIC50: 20nMAssay Description:Aurora kinase was assayed in ELISA format using a GST fusion of the N-terminus of Histone H3 as substrate. Plates were coated with substrate, and the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2009
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Genentech

LigandPNGBDBM31860(2,4-Bisanilinopyrimidine, 25)
Affinity DataIC50: 23nMAssay Description:Aurora kinase was assayed in ELISA format using a GST fusion of the N-terminus of Histone H3 as substrate. Plates were coated with substrate, and the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2009
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Genentech

LigandPNGBDBM31844(2,4-Bisanilinopyrimidine, 51)
Affinity DataIC50: 25nMpH: 7.5 T: 2°CAssay Description:Aurora kinase was assayed in ELISA format using a GST fusion of the N-terminus of Histone H3 as substrate. Plates were coated with substrate, and the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2009
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Genentech

LigandPNGBDBM31839(2,4-Bisanilinopyrimidine, 46)
Affinity DataIC50: 28nMpH: 7.5 T: 2°CAssay Description:Aurora kinase was assayed in ELISA format using a GST fusion of the N-terminus of Histone H3 as substrate. Plates were coated with substrate, and the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2009
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Genentech

LigandPNGBDBM31853(2,4-Bisanilinopyrimidine, 18)
Affinity DataIC50: 30nMAssay Description:Aurora kinase was assayed in ELISA format using a GST fusion of the N-terminus of Histone H3 as substrate. Plates were coated with substrate, and the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2009
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Genentech

LigandPNGBDBM31861(2,4-Bisanilinopyrimidine, 26)
Affinity DataIC50: 34nMAssay Description:Aurora kinase was assayed in ELISA format using a GST fusion of the N-terminus of Histone H3 as substrate. Plates were coated with substrate, and the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2009
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Genentech

LigandPNGBDBM31875(2,4-Bisanilinopyrimidine, 41)
Affinity DataIC50: 36nMAssay Description:Aurora kinase was assayed in ELISA format using a GST fusion of the N-terminus of Histone H3 as substrate. Plates were coated with substrate, and the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2009
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Genentech

LigandPNGBDBM31871(2,4-Bisanilinopyrimidine, 37)
Affinity DataIC50: 49nMAssay Description:Aurora kinase was assayed in ELISA format using a GST fusion of the N-terminus of Histone H3 as substrate. Plates were coated with substrate, and the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2009
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Genentech

LigandPNGBDBM31878(2,4-Bisanilinopyrimidine, 44)
Affinity DataIC50: 50nMAssay Description:Aurora kinase was assayed in ELISA format using a GST fusion of the N-terminus of Histone H3 as substrate. Plates were coated with substrate, and the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2009
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Genentech

LigandPNGBDBM31872(2,4-Bisanilinopyrimidine, 38)
Affinity DataIC50: 51nMAssay Description:Aurora kinase was assayed in ELISA format using a GST fusion of the N-terminus of Histone H3 as substrate. Plates were coated with substrate, and the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2009
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Genentech

LigandPNGBDBM31835(2,4-Bisanilinopyrimidine, 14)
Affinity DataIC50: 54nMpH: 7.5 T: 2°CAssay Description:Aurora kinase was assayed in ELISA format using a GST fusion of the N-terminus of Histone H3 as substrate. Plates were coated with substrate, and the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2009
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Genentech

LigandPNGBDBM31843(2,4-Bisanilinopyrimidine, 50)
Affinity DataIC50: 59nMpH: 7.5 T: 2°CAssay Description:Aurora kinase was assayed in ELISA format using a GST fusion of the N-terminus of Histone H3 as substrate. Plates were coated with substrate, and the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2009
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Genentech

LigandPNGBDBM31846(2,4-Bisanilinopyrimidine, 53)
Affinity DataIC50: 64nMpH: 7.5 T: 2°CAssay Description:Aurora kinase was assayed in ELISA format using a GST fusion of the N-terminus of Histone H3 as substrate. Plates were coated with substrate, and the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2009
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Genentech

LigandPNGBDBM31866(2,4-Bisanilinopyrimidine, 32)
Affinity DataIC50: 67nMAssay Description:Aurora kinase was assayed in ELISA format using a GST fusion of the N-terminus of Histone H3 as substrate. Plates were coated with substrate, and the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2009
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Genentech

LigandPNGBDBM31868(2,4-Bisanilinopyrimidine, 34)
Affinity DataIC50: 75nMAssay Description:Aurora kinase was assayed in ELISA format using a GST fusion of the N-terminus of Histone H3 as substrate. Plates were coated with substrate, and the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2009
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Genentech

LigandPNGBDBM31865(2,4-Bisanilinopyrimidine, 31)
Affinity DataIC50: 78nMAssay Description:Aurora kinase was assayed in ELISA format using a GST fusion of the N-terminus of Histone H3 as substrate. Plates were coated with substrate, and the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2009
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Genentech

LigandPNGBDBM31874(2,4-Bisanilinopyrimidine, 40)
Affinity DataIC50: 78nMAssay Description:Aurora kinase was assayed in ELISA format using a GST fusion of the N-terminus of Histone H3 as substrate. Plates were coated with substrate, and the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2009
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Genentech

LigandPNGBDBM31851(2,4-Bisanilinopyrimidine, 16)
Affinity DataIC50: 80nMAssay Description:Aurora kinase was assayed in ELISA format using a GST fusion of the N-terminus of Histone H3 as substrate. Plates were coated with substrate, and the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2009
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Genentech

LigandPNGBDBM31850(2,4-Bisanilinopyrimidine, 12)
Affinity DataIC50: 130nMAssay Description:Aurora kinase was assayed in ELISA format using a GST fusion of the N-terminus of Histone H3 as substrate. Plates were coated with substrate, and the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2009
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Genentech

LigandPNGBDBM31845(2,4-Bisanilinopyrimidine, 52)
Affinity DataIC50: 140nMpH: 7.5 T: 2°CAssay Description:Aurora kinase was assayed in ELISA format using a GST fusion of the N-terminus of Histone H3 as substrate. Plates were coated with substrate, and the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2009
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Genentech

LigandPNGBDBM31862(2,4-Bisanilinopyrimidine, 27)
Affinity DataIC50: 150nMAssay Description:Aurora kinase was assayed in ELISA format using a GST fusion of the N-terminus of Histone H3 as substrate. Plates were coated with substrate, and the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2009
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Genentech

LigandPNGBDBM31869(2,4-Bisanilinopyrimidine, 35)
Affinity DataIC50: 160nMAssay Description:Aurora kinase was assayed in ELISA format using a GST fusion of the N-terminus of Histone H3 as substrate. Plates were coated with substrate, and the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2009
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Genentech

LigandPNGBDBM31867(2,4-Bisanilinopyrimidine, 33)
Affinity DataIC50: 180nMAssay Description:Aurora kinase was assayed in ELISA format using a GST fusion of the N-terminus of Histone H3 as substrate. Plates were coated with substrate, and the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2009
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Genentech

LigandPNGBDBM31838(2,4-Bisanilinopyrimidine, 45)
Affinity DataIC50: 180nMpH: 7.5 T: 2°CAssay Description:Aurora kinase was assayed in ELISA format using a GST fusion of the N-terminus of Histone H3 as substrate. Plates were coated with substrate, and the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2009
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Genentech

LigandPNGBDBM31852(2,4-Bisanilinopyrimidine, 17)
Affinity DataIC50: 200nMAssay Description:Aurora kinase was assayed in ELISA format using a GST fusion of the N-terminus of Histone H3 as substrate. Plates were coated with substrate, and the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2009
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Genentech

LigandPNGBDBM31864(2,4-Bisanilinopyrimidine, 30)
Affinity DataIC50: 260nMAssay Description:Aurora kinase was assayed in ELISA format using a GST fusion of the N-terminus of Histone H3 as substrate. Plates were coated with substrate, and the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2009
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Genentech

LigandPNGBDBM31857(2,4-Bisanilinopyrimidine, 22)
Affinity DataIC50: 490nMAssay Description:Aurora kinase was assayed in ELISA format using a GST fusion of the N-terminus of Histone H3 as substrate. Plates were coated with substrate, and the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2009
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Genentech

LigandPNGBDBM31870(2,4-Bisanilinopyrimidine, 36)
Affinity DataIC50: 640nMAssay Description:Aurora kinase was assayed in ELISA format using a GST fusion of the N-terminus of Histone H3 as substrate. Plates were coated with substrate, and the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2009
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Genentech

LigandPNGBDBM31849(2,4-Bisanilinopyrimidine, 11)
Affinity DataIC50: 680nMAssay Description:Aurora kinase was assayed in ELISA format using a GST fusion of the N-terminus of Histone H3 as substrate. Plates were coated with substrate, and the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2009
Entry Details Article
PubMed
TargetAurora kinase B(Human)
Genentech

LigandPNGBDBM31833(2,4-Bisanilinopyrimidine, 5)
Affinity DataIC50: 1.40E+3nMpH: 7.5 T: 2°CAssay Description:Aurora kinase was assayed in ELISA format using a GST fusion of the N-terminus of Histone H3 as substrate. Plates were coated with substrate, and the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2009
Entry Details Article
PubMed
TargetAurora kinase B(Human)
Genentech

LigandPNGBDBM31834(2,4-Bisanilinopyrimidine, 13)
Affinity DataIC50: 1.90E+3nMpH: 7.5 T: 2°CAssay Description:Aurora kinase was assayed in ELISA format using a GST fusion of the N-terminus of Histone H3 as substrate. Plates were coated with substrate, and the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2009
Entry Details Article
PubMed
TargetAurora kinase B(Human)
Genentech

LigandPNGBDBM31837(Aurora Inhibitor, 35 | 2,4-Bisanilinopyrimidine, 1...)
Affinity DataIC50: 3.40E+3nMpH: 7.5 T: 2°CAssay Description:Aurora kinase was assayed in ELISA format using a GST fusion of the N-terminus of Histone H3 as substrate. Plates were coated with substrate, and the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2009
Entry Details Article
PubMed
TargetAurora kinase B(Human)
Genentech

LigandPNGBDBM31836(2,4-Bisanilinopyrimidine, 9)
Affinity DataIC50: 3.70E+3nMpH: 7.5 T: 2°CAssay Description:Aurora kinase was assayed in ELISA format using a GST fusion of the N-terminus of Histone H3 as substrate. Plates were coated with substrate, and the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2009
Entry Details Article
PubMed
TargetAurora kinase B(Human)
Genentech

LigandPNGBDBM31835(2,4-Bisanilinopyrimidine, 14)
Affinity DataIC50: 3.80E+3nMpH: 7.5 T: 2°CAssay Description:Aurora kinase was assayed in ELISA format using a GST fusion of the N-terminus of Histone H3 as substrate. Plates were coated with substrate, and the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2009
Entry Details Article
PubMed
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