Compile Data Set for Download or QSAR
Report error Found 71 Enz. Inhib. hit(s) with all data for entry = 50028722
LigandPNGBDBM50278942(D-2-(4-(but-2-ynyloxy)phenylsulfonamido)-3-(1-(4-m...)
Affinity DataIC50: 80nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50279256(D-2-(4-(but-2-ynyloxy)phenylsulfonamido)-3-(5-meth...)
Affinity DataIC50: 140nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50278998(rac-2-(4-(but-2-ynyloxy)phenylsulfonamido)-3-(5-ch...)
Affinity DataIC50: 190nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50279026(rac-3-(1-benzyl-5-methoxy-2-methyl-1H-indol-3-yl)-...)
Affinity DataIC50: 250nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50279256(D-2-(4-(but-2-ynyloxy)phenylsulfonamido)-3-(5-meth...)
Affinity DataIC50: 270nMAssay Description:Inhibition of MMP2 by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50279255(2-(4-(but-2-ynyloxy)phenylsulfonamido)-3-(5-methyl...)
Affinity DataIC50: 280nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50279067(rac-2-(4-(but-2-ynyloxy)phenylsulfonamido)-3-(5-me...)
Affinity DataIC50: 280nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50279110(rac-2-(4-(but-2-ynyloxy)phenylsulfonamido)-3-(1-(4...)
Affinity DataIC50: 290nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50279071(rac-2-(4-(but-2-ynyloxy)phenylsulfonamido)-3-(1-(2...)
Affinity DataIC50: 300nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50278996(rac-2-(4-(but-2-ynyloxy)phenylsulfonamido)-3-(5-ch...)
Affinity DataIC50: 300nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50279109(rac-2-(4-(but-2-ynyloxy)phenylsulfonamido)-3-(1-(4...)
Affinity DataIC50: 320nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50279152(rac-2-(4-(but-2-ynyloxy)phenylsulfonamido)-3-(5-ch...)
Affinity DataIC50: 330nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50279028(rac-3-(1-(benzo[d][1,3]dioxol-5-ylmethyl)-5-methox...)
Affinity DataIC50: 330nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50279108(rac-2-(4-(but-2-ynyloxy)phenylsulfonamido)-3-(1-(3...)
Affinity DataIC50: 340nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50279153(2-(4-(but-2-ynyloxy)phenylsulfonamido)-3-(1-(3-cya...)
Affinity DataIC50: 410nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50279154(rac-2-(4-(but-2-ynyloxy)phenylsulfonamido)-3-(1-(4...)
Affinity DataIC50: 470nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50279069(rac-2-(4-(but-2-ynyloxy)phenylsulfonamido)-3-(5-me...)
Affinity DataIC50: 490nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50279068(rac-2-(4-(but-2-ynyloxy)phenylsulfonamido)-3-(5-me...)
Affinity DataIC50: 500nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50278888(D-3-(1-(4-(allyloxy)benzyl)-1H-indol-3-yl)-2-(4-(b...)
Affinity DataIC50: 540nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50279343(rac-3-(5-bromo-1H-indol-3-yl)-2-(4-(but-2-ynyloxy)...)
Affinity DataIC50: 630nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50278997(rac-2-(4-(but-2-ynyloxy)phenylsulfonamido)-3-(1-(4...)
Affinity DataIC50: 890nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50279025(rac-2-(4-(but-2-ynyloxy)phenylsulfonamido)-3-(5-me...)
Affinity DataIC50: 900nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50279416(D-3-(1-(biphenyl-2-ylmethyl)-1H-indol-3-yl)-2-(4-(...)
Affinity DataIC50: 970nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50278889(D-2-(4-(but-2-ynyloxy)phenylsulfonamido)-3-(1-(3,5...)
Affinity DataIC50: 980nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50278974(L-2-(4-(but-2-ynyloxy)phenylsulfonamido)-3-(1-(4-m...)
Affinity DataIC50: 1.18E+3nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50278995(rac-2-(4-(but-2-ynyloxy)phenylsulfonamido)-3-(1-is...)
Affinity DataIC50: 1.23E+3nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50279414(D-2-(4-(but-2-ynyloxy)phenylsulfonamido)-3-(1-(4-p...)
Affinity DataIC50: 1.25E+3nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50279257(2-(4-(but-2-ynyloxy)phenylsulfonamido)-3-(5-methox...)
Affinity DataIC50: 1.27E+3nMAssay Description:Inhibition of MMP2 by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50279377(D-2-(4-(but-2-ynyloxy)phenylsulfonamido)-3-(1-meth...)
Affinity DataIC50: 1.43E+3nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50278942(D-2-(4-(but-2-ynyloxy)phenylsulfonamido)-3-(1-(4-m...)
Affinity DataIC50: 1.44E+3nMAssay Description:Inhibition of MMP2 by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50279027(rac-3-(1-(benzo[d][1,3]dioxol-5-ylmethyl)-5-methox...)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50279341(rac-2-(4-(but-2-ynyloxy)phenylsulfonamido)-3-(5-fl...)
Affinity DataIC50: 1.56E+3nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50279375(rac-2-(4-(but-2-ynyloxy)phenylsulfonamido)-3-(6-me...)
Affinity DataIC50: 1.57E+3nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50279342(rac-2-(4-(but-2-ynyloxy)phenylsulfonamido)-3-(5-hy...)
Affinity DataIC50: 1.61E+3nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50279413(D-2-(4-(but-2-ynyloxy)phenylsulfonamido)-3-(1-(cyc...)
Affinity DataIC50: 1.71E+3nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50279256(D-2-(4-(but-2-ynyloxy)phenylsulfonamido)-3-(5-meth...)
Affinity DataIC50: 1.81E+3nMAssay Description:Inhibition of MMP13 by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50278940(D-2-(4-(but-2-ynyloxy)phenylsulfonamido)-3-(1-(4-f...)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50279415(D-3-(1-benzyl-1H-indol-3-yl)-2-(4-(but-2-ynyloxy)p...)
Affinity DataIC50: 2.15E+3nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50279070(rac-2-(4-(but-2-ynyloxy)phenylsulfonamido)-3-(1-(2...)
Affinity DataIC50: 2.24E+3nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50279029(rac-2-(4-(but-2-ynyloxy)phenylsulfonamido)-3-(5-me...)
Affinity DataIC50: 2.24E+3nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50278913(D-2-(4-(but-2-ynyloxy)phenylsulfonamido)-3-(1-(3-(...)
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50279412(D-2-(4-(but-2-ynyloxy)phenylsulfonamido)-3-(1-pent...)
Affinity DataIC50: 2.31E+3nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50279221(D-2-(4-(but-2-ynyloxy)phenylsulfonamido)-3-(1H-ind...)
Affinity DataIC50: 2.53E+3nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50279374(rac-2-(4-(but-2-ynyloxy)phenylsulfonamido)-3-(6-fl...)
Affinity DataIC50: 2.96E+3nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50279287(3-(5-(benzyloxy)-1H-indol-3-yl)-2-(4-(but-2-ynylox...)
Affinity DataIC50: 3.27E+3nMAssay Description:Inhibition of MMP2 by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50278941(D-2-(4-(but-2-ynyloxy)phenylsulfonamido)-3-(1-(4-c...)
Affinity DataIC50: 3.45E+3nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50278915(D-2-(4-(but-2-ynyloxy)phenylsulfonamido)-3-(1-(4-m...)
Affinity DataIC50: 3.59E+3nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50279376(D-2-(4-(but-2-ynyloxy)phenylsulfonamido)-3-(1-(ter...)
Affinity DataIC50: 3.67E+3nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50278914(D-2-(4-(but-2-ynyloxy)phenylsulfonamido)-3-(1-(4-(...)
Affinity DataIC50: 4.40E+3nMAssay Description:Inhibition of TACE by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50279287(3-(5-(benzyloxy)-1H-indol-3-yl)-2-(4-(but-2-ynylox...)
Affinity DataIC50: 4.44E+3nMAssay Description:Inhibition of MMP13 by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
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