Compile Data Set for Download or QSAR
Report error Found 125 Enz. Inhib. hit(s) with all data for entry = 3281
TargetCollagenase 3(Human)
Novartis

LigandPNGBDBM30345(BOC-piperidinyl glycine derivative, 9)
Affinity DataIC50: 0.300nMpH: 7.5 T: 2°CAssay Description:Test compounds were serially diluted in the assay buffer. In each well of a 96-well microtiter plate (Immunofluor B, Dynatech), the inhibitor solutio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Novartis

LigandPNGBDBM30356(BOC-piperidinyl glycine derivative, 31)
Affinity DataIC50: 0.300nMpH: 7.5 T: 2°CAssay Description:Test compounds were serially diluted in the assay buffer. In each well of a 96-well microtiter plate (Immunofluor B, Dynatech), the inhibitor solutio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Novartis

LigandPNGBDBM30380(piperidinyl glycine derivative, 24q)
Affinity DataIC50: 0.400nMT: 2°CAssay Description:Test compounds were serially diluted in the assay buffer. In each well of a 96-well microtiter plate (Immunofluor B, Dynatech), the inhibitor solutio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Novartis

LigandPNGBDBM30384(piperidinyl glycine derivative, 24u)
Affinity DataIC50: 0.400nMT: 2°CAssay Description:Test compounds were serially diluted in the assay buffer. In each well of a 96-well microtiter plate (Immunofluor B, Dynatech), the inhibitor solutio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Novartis

LigandPNGBDBM30359(BOC-piperidinyl glycine derivative, 34)
Affinity DataIC50: 0.5nMpH: 7.5 T: 2°CAssay Description:Test compounds were serially diluted in the assay buffer. In each well of a 96-well microtiter plate (Immunofluor B, Dynatech), the inhibitor solutio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Novartis

LigandPNGBDBM30360(BOC-piperidinyl glycine derivative, 35)
Affinity DataIC50: 0.5nMpH: 7.5 T: 2°CAssay Description:Test compounds were serially diluted in the assay buffer. In each well of a 96-well microtiter plate (Immunofluor B, Dynatech), the inhibitor solutio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Novartis

LigandPNGBDBM30383(piperidinyl glycine derivative, 24t)
Affinity DataIC50: 0.5nMT: 2°CAssay Description:Test compounds were serially diluted in the assay buffer. In each well of a 96-well microtiter plate (Immunofluor B, Dynatech), the inhibitor solutio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Novartis

LigandPNGBDBM30367(piperidinyl glycine derivative, 24d)
Affinity DataIC50: 0.600nMpH: 7.5 T: 2°CAssay Description:Test compounds were serially diluted in the assay buffer. In each well of a 96-well microtiter plate (Immunofluor B, Dynatech), the inhibitor solutio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Novartis

LigandPNGBDBM30379(piperidinyl glycine derivative, 24p)
Affinity DataIC50: 0.600nMT: 2°CAssay Description:Test compounds were serially diluted in the assay buffer. In each well of a 96-well microtiter plate (Immunofluor B, Dynatech), the inhibitor solutio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Novartis

LigandPNGBDBM30382(piperidinyl glycine derivative, 24s)
Affinity DataIC50: 0.600nMT: 2°CAssay Description:Test compounds were serially diluted in the assay buffer. In each well of a 96-well microtiter plate (Immunofluor B, Dynatech), the inhibitor solutio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Novartis

LigandPNGBDBM30357(BOC-piperidinyl glycine derivative, 32)
Affinity DataIC50: 0.700nMpH: 7.5 T: 2°CAssay Description:Test compounds were serially diluted in the assay buffer. In each well of a 96-well microtiter plate (Immunofluor B, Dynatech), the inhibitor solutio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Novartis

LigandPNGBDBM30396(piperidinyl glycine derivative, 27c)
Affinity DataIC50: 0.700nMT: 2°CAssay Description:Test compounds were serially diluted in the assay buffer. In each well of a 96-well microtiter plate (Immunofluor B, Dynatech), the inhibitor solutio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Novartis

LigandPNGBDBM30397(piperidinyl glycine derivative, 27d)
Affinity DataIC50: 0.700nMT: 2°CAssay Description:Test compounds were serially diluted in the assay buffer. In each well of a 96-well microtiter plate (Immunofluor B, Dynatech), the inhibitor solutio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Novartis

LigandPNGBDBM30347(BOC-piperidinyl glycine derivative, 22a)
Affinity DataIC50: 0.75nMpH: 7.5 T: 2°CAssay Description:Test compounds were serially diluted in the assay buffer. In each well of a 96-well microtiter plate (Immunofluor B, Dynatech), the inhibitor solutio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Novartis

LigandPNGBDBM30370(piperidinyl glycine derivative, 24g)
Affinity DataIC50: 0.800nMpH: 7.5 T: 2°CAssay Description:Test compounds were serially diluted in the assay buffer. In each well of a 96-well microtiter plate (Immunofluor B, Dynatech), the inhibitor solutio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Novartis

LigandPNGBDBM30378(piperidinyl glycine derivative, 24o)
Affinity DataIC50: 0.800nMT: 2°CAssay Description:Test compounds were serially diluted in the assay buffer. In each well of a 96-well microtiter plate (Immunofluor B, Dynatech), the inhibitor solutio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Novartis

LigandPNGBDBM30387(piperidinyl glycine derivative, 25c)
Affinity DataIC50: 0.800nMT: 2°CAssay Description:Test compounds were serially diluted in the assay buffer. In each well of a 96-well microtiter plate (Immunofluor B, Dynatech), the inhibitor solutio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Novartis

LigandPNGBDBM30372(piperidinyl glycine derivative, 24i)
Affinity DataIC50: 0.900nMT: 2°CAssay Description:Test compounds were serially diluted in the assay buffer. In each well of a 96-well microtiter plate (Immunofluor B, Dynatech), the inhibitor solutio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Novartis

LigandPNGBDBM30381(piperidinyl glycine derivative, 24r)
Affinity DataIC50: 0.900nMT: 2°CAssay Description:Test compounds were serially diluted in the assay buffer. In each well of a 96-well microtiter plate (Immunofluor B, Dynatech), the inhibitor solutio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Novartis

LigandPNGBDBM30392(piperidinyl glycine derivative, 26d)
Affinity DataIC50: 0.900nMT: 2°CAssay Description:Test compounds were serially diluted in the assay buffer. In each well of a 96-well microtiter plate (Immunofluor B, Dynatech), the inhibitor solutio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Novartis

LigandPNGBDBM30377(piperidinyl glycine derivative, 24n)
Affinity DataIC50: 1nMT: 2°CAssay Description:Test compounds were serially diluted in the assay buffer. In each well of a 96-well microtiter plate (Immunofluor B, Dynatech), the inhibitor solutio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Novartis

LigandPNGBDBM30395(piperidinyl glycine derivative, 27b)
Affinity DataIC50: 1.20nMT: 2°CAssay Description:Test compounds were serially diluted in the assay buffer. In each well of a 96-well microtiter plate (Immunofluor B, Dynatech), the inhibitor solutio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Novartis

LigandPNGBDBM30364(piperidinyl glycine derivative, 24a)
Affinity DataIC50: 1.30nMpH: 7.5 T: 2°CAssay Description:Test compounds were serially diluted in the assay buffer. In each well of a 96-well microtiter plate (Immunofluor B, Dynatech), the inhibitor solutio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Novartis

LigandPNGBDBM30373(piperidinyl glycine derivative, 24j)
Affinity DataIC50: 1.30nMT: 2°CAssay Description:Test compounds were serially diluted in the assay buffer. In each well of a 96-well microtiter plate (Immunofluor B, Dynatech), the inhibitor solutio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Novartis

LigandPNGBDBM30385(piperidinyl glycine derivative, 25a)
Affinity DataIC50: 1.40nMT: 2°CAssay Description:Test compounds were serially diluted in the assay buffer. In each well of a 96-well microtiter plate (Immunofluor B, Dynatech), the inhibitor solutio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Novartis

LigandPNGBDBM30394(piperidinyl glycine derivative, 27a)
Affinity DataIC50: 1.40nMT: 2°CAssay Description:Test compounds were serially diluted in the assay buffer. In each well of a 96-well microtiter plate (Immunofluor B, Dynatech), the inhibitor solutio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Novartis

LigandPNGBDBM30386(piperidinyl glycine derivative, 25b)
Affinity DataIC50: 1.60nMT: 2°CAssay Description:Test compounds were serially diluted in the assay buffer. In each well of a 96-well microtiter plate (Immunofluor B, Dynatech), the inhibitor solutio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Novartis

LigandPNGBDBM30393(piperidinyl glycine derivative, 26e)
Affinity DataIC50: 1.70nMT: 2°CAssay Description:Test compounds were serially diluted in the assay buffer. In each well of a 96-well microtiter plate (Immunofluor B, Dynatech), the inhibitor solutio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Novartis

LigandPNGBDBM11863(CHEMBL440498 | alpha-tetrahydropyran beta-sulfone ...)
Affinity DataIC50: 2nMT: 2°CAssay Description:Test compounds were serially diluted in the assay buffer. In each well of a 96-well microtiter plate (Immunofluor B, Dynatech), the inhibitor solutio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Novartis

LigandPNGBDBM30376(piperidinyl glycine derivative, 24m)
Affinity DataIC50: 2nMT: 2°CAssay Description:Test compounds were serially diluted in the assay buffer. In each well of a 96-well microtiter plate (Immunofluor B, Dynatech), the inhibitor solutio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Novartis

LigandPNGBDBM30368(piperidinyl glycine derivative, 24e)
Affinity DataIC50: 2.20nMpH: 7.5 T: 2°CAssay Description:Test compounds were serially diluted in the assay buffer. In each well of a 96-well microtiter plate (Immunofluor B, Dynatech), the inhibitor solutio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2009
Entry Details Article
PubMed
TargetInterstitial collagenase(Human)
Novartis

LigandPNGBDBM30344(Trocade | Cipemastat)
Affinity DataIC50: 2.30nMT: 2°CAssay Description:Test compounds were serially diluted in the assay buffer. In each well of a 96-well microtiter plate (Immunofluor B, Dynatech), the inhibitor solutio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Novartis

LigandPNGBDBM30358(BOC-piperidinyl glycine derivative, 33)
Affinity DataIC50: 2.40nMpH: 7.5 T: 2°CAssay Description:Test compounds were serially diluted in the assay buffer. In each well of a 96-well microtiter plate (Immunofluor B, Dynatech), the inhibitor solutio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Novartis

LigandPNGBDBM30344(Trocade | Cipemastat)
Affinity DataIC50: 2.40nMT: 2°CAssay Description:Test compounds were serially diluted in the assay buffer. In each well of a 96-well microtiter plate (Immunofluor B, Dynatech), the inhibitor solutio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Novartis

LigandPNGBDBM30388(piperidinyl glycine derivative, 25d)
Affinity DataIC50: 2.80nMT: 2°CAssay Description:Test compounds were serially diluted in the assay buffer. In each well of a 96-well microtiter plate (Immunofluor B, Dynatech), the inhibitor solutio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Novartis

LigandPNGBDBM30366(piperidinyl glycine derivative, 24c)
Affinity DataIC50: 3.30nMpH: 7.5 T: 2°CAssay Description:Test compounds were serially diluted in the assay buffer. In each well of a 96-well microtiter plate (Immunofluor B, Dynatech), the inhibitor solutio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Novartis

LigandPNGBDBM30375(piperidinyl glycine derivative, 24l)
Affinity DataIC50: 3.5nMT: 2°CAssay Description:Test compounds were serially diluted in the assay buffer. In each well of a 96-well microtiter plate (Immunofluor B, Dynatech), the inhibitor solutio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Novartis

LigandPNGBDBM30391(piperidinyl glycine derivative, 26c)
Affinity DataIC50: 3.60nMT: 2°CAssay Description:Test compounds were serially diluted in the assay buffer. In each well of a 96-well microtiter plate (Immunofluor B, Dynatech), the inhibitor solutio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Novartis

LigandPNGBDBM30374(piperidinyl glycine derivative, 24k)
Affinity DataIC50: 3.90nMT: 2°CAssay Description:Test compounds were serially diluted in the assay buffer. In each well of a 96-well microtiter plate (Immunofluor B, Dynatech), the inhibitor solutio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Novartis

LigandPNGBDBM30371(piperidinyl glycine derivative, 24h)
Affinity DataIC50: 4nMT: 2°CAssay Description:Test compounds were serially diluted in the assay buffer. In each well of a 96-well microtiter plate (Immunofluor B, Dynatech), the inhibitor solutio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Novartis

LigandPNGBDBM30399(piperidinyl glycine derivative, 27f)
Affinity DataIC50: 4nMT: 2°CAssay Description:Test compounds were serially diluted in the assay buffer. In each well of a 96-well microtiter plate (Immunofluor B, Dynatech), the inhibitor solutio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Novartis

LigandPNGBDBM30400(piperidinyl glycine derivative, 27g)
Affinity DataIC50: 4.70nMT: 2°CAssay Description:Test compounds were serially diluted in the assay buffer. In each well of a 96-well microtiter plate (Immunofluor B, Dynatech), the inhibitor solutio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Novartis

LigandPNGBDBM30398(piperidinyl glycine derivative, 27e)
Affinity DataIC50: 5.5nMT: 2°CAssay Description:Test compounds were serially diluted in the assay buffer. In each well of a 96-well microtiter plate (Immunofluor B, Dynatech), the inhibitor solutio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Novartis

LigandPNGBDBM30348(BOC-piperidinyl glycine derivative, 22b)
Affinity DataIC50: 6.80nMpH: 7.5 T: 2°CAssay Description:Test compounds were serially diluted in the assay buffer. In each well of a 96-well microtiter plate (Immunofluor B, Dynatech), the inhibitor solutio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Novartis

LigandPNGBDBM8465(CGS 27023 | CHEMBL514138 | hydroxamate analogue 1 ...)
Affinity DataIC50: 6.80nMT: 2°CAssay Description:Test compounds were serially diluted in the assay buffer. In each well of a 96-well microtiter plate (Immunofluor B, Dynatech), the inhibitor solutio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Novartis

LigandPNGBDBM30401(piperidinyl glycine derivative, 27h)
Affinity DataIC50: 6.90nMT: 2°CAssay Description:Test compounds were serially diluted in the assay buffer. In each well of a 96-well microtiter plate (Immunofluor B, Dynatech), the inhibitor solutio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2009
Entry Details Article
PubMed
TargetStromelysin-1(Human)
Novartis

LigandPNGBDBM11863(CHEMBL440498 | alpha-tetrahydropyran beta-sulfone ...)
Affinity DataIC50: 7.10nMT: 2°CAssay Description:Test compounds were serially diluted in the assay buffer. In each well of a 96-well microtiter plate (Immunofluor B, Dynatech), the inhibitor solutio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Novartis

LigandPNGBDBM30403(piperidinyl glycine derivative, 28a)
Affinity DataIC50: 7.60nMT: 2°CAssay Description:Test compounds were serially diluted in the assay buffer. In each well of a 96-well microtiter plate (Immunofluor B, Dynatech), the inhibitor solutio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Novartis

LigandPNGBDBM30390(piperidinyl glycine derivative, 26b)
Affinity DataIC50: 8nMT: 2°CAssay Description:Test compounds were serially diluted in the assay buffer. In each well of a 96-well microtiter plate (Immunofluor B, Dynatech), the inhibitor solutio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Novartis

LigandPNGBDBM30369(piperidinyl glycine derivative, 24f)
Affinity DataIC50: 10nMT: 2°CAssay Description:Test compounds were serially diluted in the assay buffer. In each well of a 96-well microtiter plate (Immunofluor B, Dynatech), the inhibitor solutio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2009
Entry Details Article
PubMed
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