Compile Data Set for Download or QSAR
Report error Found 34 Enz. Inhib. hit(s) with all data for entry = 50038841
TargetCannabinoid receptor 2(Human)
Universita Di Pisa

Curated by ChEMBL
LigandPNGBDBM50180022(5-(4-chloro-3-methyl-phenyl)-1-(4-methyl-benzyl)-1...)
Affinity DataKi:  0.600nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Universita Di Pisa

Curated by ChEMBL
LigandPNGBDBM50258604(N-Cycloheptyl-1-(p-fluorobenzyl)-1,8-naphthyridin-...)
Affinity DataKi:  0.700nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Universita Di Pisa

Curated by ChEMBL
LigandPNGBDBM50258654(cis-N-(4-Methylcyclohexyl)-1-(p-fluorobenzyl)-1,8-...)
Affinity DataKi:  0.700nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Universita Di Pisa

Curated by ChEMBL
LigandPNGBDBM50258652(N-(4-Methylcyclohexyl)-1-(p-fluorobenzyl)-1,8-naph...)
Affinity DataKi:  0.900nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Universita Di Pisa

Curated by ChEMBL
LigandPNGBDBM50258570(N-(4-Methylcyclohexyl)-1-(2-morpholin-4-ylethyl)-1...)
Affinity DataKi:  1.90nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Universita Di Pisa

Curated by ChEMBL
LigandPNGBDBM50258527(N-Cyclohexyl-1-(p-fluorobenzyl)-1,8-naphthyridin-2...)
Affinity DataKi:  2.20nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Universita Di Pisa

Curated by ChEMBL
LigandPNGBDBM50258605(N-Cycloheptyl-1-(2-morpholin-4-ylethyl)-1,8-naphth...)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Universita Di Pisa

Curated by ChEMBL
LigandPNGBDBM50180036(CHEMBL371214 | (6aR,10aR)-3-(1,1-dimethylbutyl)-6a...)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Universita Di Pisa

Curated by ChEMBL
LigandPNGBDBM50258608(cis-N-(4-Methylcyclohexyl)-1-benzyl-1,8-naphthyrid...)
Affinity DataKi:  5.80nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Universita Di Pisa

Curated by ChEMBL
LigandPNGBDBM50258606(N-(4-Methylcyclohexyl)-1-benzyl-1,8-naphthyridin-2...)
Affinity DataKi:  7.80nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Universita Di Pisa

Curated by ChEMBL
LigandPNGBDBM50258525(N-cyclohexyl-1-(2-morpholin-4-ylethyl)-1,8-naphthy...)
Affinity DataKi:  7.90nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Universita Di Pisa

Curated by ChEMBL
LigandPNGBDBM50258653(trans-N-(4-Methylcyclohexyl)-1-(p-fluorobenzyl)-1,...)
Affinity DataKi:  9nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Universita Di Pisa

Curated by ChEMBL
LigandPNGBDBM50258604(N-Cycloheptyl-1-(p-fluorobenzyl)-1,8-naphthyridin-...)
Affinity DataKi:  9.60nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Universita Di Pisa

Curated by ChEMBL
LigandPNGBDBM50258605(N-Cycloheptyl-1-(2-morpholin-4-ylethyl)-1,8-naphth...)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Universita Di Pisa

Curated by ChEMBL
LigandPNGBDBM50258572(N-Cycloheptyl-1-benzyl-1,8-naphthyridin-2(1H)-on-3...)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Universita Di Pisa

Curated by ChEMBL
LigandPNGBDBM50258526(N-Cyclohexyl-1-benzyl-1,8-naphthyridin-2(1H)-on-3-...)
Affinity DataKi:  31nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Universita Di Pisa

Curated by ChEMBL
LigandPNGBDBM50258607(trans-N-(4-Methylcyclohexyl)-1-benzyl-1,8-naphthyr...)
Affinity DataKi:  39.8nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Universita Di Pisa

Curated by ChEMBL
LigandPNGBDBM50258527(N-Cyclohexyl-1-(p-fluorobenzyl)-1,8-naphthyridin-2...)
Affinity DataKi:  56nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Universita Di Pisa

Curated by ChEMBL
LigandPNGBDBM50258571(N-(4-Fluorophenylethyl)-1-benzyl-1,8-naphthyridin-...)
Affinity DataKi:  69.8nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Universita Di Pisa

Curated by ChEMBL
LigandPNGBDBM50258569(N-Cyclohexyl-1-butyl-1,8-naphthyridin-2(1H)-on-3-c...)
Affinity DataKi:  70nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Universita Di Pisa

Curated by ChEMBL
LigandPNGBDBM50258652(N-(4-Methylcyclohexyl)-1-(p-fluorobenzyl)-1,8-naph...)
Affinity DataKi:  200nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Universita Di Pisa

Curated by ChEMBL
LigandPNGBDBM50258654(cis-N-(4-Methylcyclohexyl)-1-(p-fluorobenzyl)-1,8-...)
Affinity DataKi:  200nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Universita Di Pisa

Curated by ChEMBL
LigandPNGBDBM50258653(trans-N-(4-Methylcyclohexyl)-1-(p-fluorobenzyl)-1,...)
Affinity DataKi:  300nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Universita Di Pisa

Curated by ChEMBL
LigandPNGBDBM50180022(5-(4-chloro-3-methyl-phenyl)-1-(4-methyl-benzyl)-1...)
Affinity DataKi:  437nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Universita Di Pisa

Curated by ChEMBL
LigandPNGBDBM50258525(N-cyclohexyl-1-(2-morpholin-4-ylethyl)-1,8-naphthy...)
Affinity DataKi:  560nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Universita Di Pisa

Curated by ChEMBL
LigandPNGBDBM50258526(N-Cyclohexyl-1-benzyl-1,8-naphthyridin-2(1H)-on-3-...)
Affinity DataKi:  560nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Universita Di Pisa

Curated by ChEMBL
LigandPNGBDBM50180036(CHEMBL371214 | (6aR,10aR)-3-(1,1-dimethylbutyl)-6a...)
Affinity DataKi:  677nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Universita Di Pisa

Curated by ChEMBL
LigandPNGBDBM50258572(N-Cycloheptyl-1-benzyl-1,8-naphthyridin-2(1H)-on-3...)
Affinity DataKi:  960nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Universita Di Pisa

Curated by ChEMBL
LigandPNGBDBM50258570(N-(4-Methylcyclohexyl)-1-(2-morpholin-4-ylethyl)-1...)
Affinity DataKi:  1.00E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Universita Di Pisa

Curated by ChEMBL
LigandPNGBDBM50258608(cis-N-(4-Methylcyclohexyl)-1-benzyl-1,8-naphthyrid...)
Affinity DataKi:  1.52E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Universita Di Pisa

Curated by ChEMBL
LigandPNGBDBM50258606(N-(4-Methylcyclohexyl)-1-benzyl-1,8-naphthyridin-2...)
Affinity DataKi:  1.60E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Universita Di Pisa

Curated by ChEMBL
LigandPNGBDBM50258607(trans-N-(4-Methylcyclohexyl)-1-benzyl-1,8-naphthyr...)
Affinity DataKi:  5.26E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Universita Di Pisa

Curated by ChEMBL
LigandPNGBDBM50258569(N-Cyclohexyl-1-butyl-1,8-naphthyridin-2(1H)-on-3-c...)
Affinity DataKi:  5.60E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Universita Di Pisa

Curated by ChEMBL
LigandPNGBDBM50258571(N-(4-Fluorophenylethyl)-1-benzyl-1,8-naphthyridin-...)
Affinity DataKi:  6.95E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2012
Entry Details Article
PubMed