Compile Data Set for Download or QSAR
Report error Found 21 Enz. Inhib. hit(s) with all data for entry = 3269
TargetMelanin-concentrating hormone receptor 1(Human)
Banyu Pharmaceutical

LigandPNGBDBM30177(2-aminobenzimidazole-based compound, 25)
Affinity DataIC50: 2.70nMpH: 7.4 T: 2°CAssay Description:Compounds were evaluated for their binding affinity to the membranes of CHO-K1 cells expressing human MCH1R (hMCH1R) in a competition binding assay w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Banyu Pharmaceutical

LigandPNGBDBM30172(2-aminobenzimidazole-based compound, 20)
Affinity DataIC50: 3.10nMpH: 7.4 T: 2°CAssay Description:Compounds were evaluated for their binding affinity to the membranes of CHO-K1 cells expressing human MCH1R (hMCH1R) in a competition binding assay w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Banyu Pharmaceutical

LigandPNGBDBM30164(2-aminobenzimidazole-based compound, 12)
Affinity DataIC50: 4nM EC50:  22nMpH: 7.4 T: 2°CAssay Description:Compounds were evaluated for their binding affinity to the membranes of CHO-K1 cells expressing human MCH1R (hMCH1R) in a competition binding assay w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Banyu Pharmaceutical

LigandPNGBDBM30174(2-aminobenzimidazole-based compound, 22)
Affinity DataIC50: 5.5nMpH: 7.4 T: 2°CAssay Description:Compounds were evaluated for their binding affinity to the membranes of CHO-K1 cells expressing human MCH1R (hMCH1R) in a competition binding assay w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Banyu Pharmaceutical

LigandPNGBDBM30156(2-aminobenzimidazole-based compound, 8)
Affinity DataIC50: 5.90nM EC50:  21nMpH: 7.4 T: 2°CAssay Description:Compounds were evaluated for their binding affinity to the membranes of CHO-K1 cells expressing human MCH1R (hMCH1R) in a competition binding assay w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Banyu Pharmaceutical

LigandPNGBDBM30165(2-aminobenzimidazole-based compound, 13)
Affinity DataIC50: 6.70nM EC50:  27nMpH: 7.4 T: 2°CAssay Description:Compounds were evaluated for their binding affinity to the membranes of CHO-K1 cells expressing human MCH1R (hMCH1R) in a competition binding assay w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Banyu Pharmaceutical

LigandPNGBDBM30173(2-aminobenzimidazole-based compound, 21)
Affinity DataIC50: 8.80nMpH: 7.4 T: 2°CAssay Description:Compounds were evaluated for their binding affinity to the membranes of CHO-K1 cells expressing human MCH1R (hMCH1R) in a competition binding assay w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Banyu Pharmaceutical

LigandPNGBDBM30161(2-aminobenzimidazole-based compound, 9)
Affinity DataIC50: 12nMpH: 7.4 T: 2°CAssay Description:Compounds were evaluated for their binding affinity to the membranes of CHO-K1 cells expressing human MCH1R (hMCH1R) in a competition binding assay w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Banyu Pharmaceutical

LigandPNGBDBM30176(2-aminobenzimidazole-based compound, 24)
Affinity DataIC50: 15nMpH: 7.4 T: 2°CAssay Description:Compounds were evaluated for their binding affinity to the membranes of CHO-K1 cells expressing human MCH1R (hMCH1R) in a competition binding assay w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Banyu Pharmaceutical

LigandPNGBDBM30162(2-aminobenzimidazole-based compound, 10)
Affinity DataIC50: 19nMpH: 7.4 T: 2°CAssay Description:Compounds were evaluated for their binding affinity to the membranes of CHO-K1 cells expressing human MCH1R (hMCH1R) in a competition binding assay w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Banyu Pharmaceutical

LigandPNGBDBM30168(2-aminobenzimidazole-based compound, 16)
Affinity DataIC50: 23nMpH: 7.4 T: 2°CAssay Description:Compounds were evaluated for their binding affinity to the membranes of CHO-K1 cells expressing human MCH1R (hMCH1R) in a competition binding assay w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Banyu Pharmaceutical

LigandPNGBDBM30163(2-aminobenzimidazole-based compound, 11)
Affinity DataIC50: 24nMpH: 7.4 T: 2°CAssay Description:Compounds were evaluated for their binding affinity to the membranes of CHO-K1 cells expressing human MCH1R (hMCH1R) in a competition binding assay w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Banyu Pharmaceutical

LigandPNGBDBM30166(2-aminobenzimidazole-based compound, 14)
Affinity DataIC50: 27nMpH: 7.4 T: 2°CAssay Description:Compounds were evaluated for their binding affinity to the membranes of CHO-K1 cells expressing human MCH1R (hMCH1R) in a competition binding assay w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Banyu Pharmaceutical

LigandPNGBDBM30167(2-aminobenzimidazole-based compound, 15)
Affinity DataIC50: 30nMpH: 7.4 T: 2°CAssay Description:Compounds were evaluated for their binding affinity to the membranes of CHO-K1 cells expressing human MCH1R (hMCH1R) in a competition binding assay w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Banyu Pharmaceutical

LigandPNGBDBM30171(2-aminobenzimidazole-based compound, 19)
Affinity DataIC50: 41nMpH: 7.4 T: 2°CAssay Description:Compounds were evaluated for their binding affinity to the membranes of CHO-K1 cells expressing human MCH1R (hMCH1R) in a competition binding assay w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Banyu Pharmaceutical

LigandPNGBDBM30169(2-aminobenzimidazole-based compound, 17)
Affinity DataIC50: 135nMpH: 7.4 T: 2°CAssay Description:Compounds were evaluated for their binding affinity to the membranes of CHO-K1 cells expressing human MCH1R (hMCH1R) in a competition binding assay w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Banyu Pharmaceutical

LigandPNGBDBM30159(aminonaphthyridine-based compound, 36)
Affinity DataIC50: 365nMpH: 7.4 T: 2°CAssay Description:Compounds were evaluated for their binding affinity to the membranes of CHO-K1 cells expressing human MCH1R (hMCH1R) in a competition binding assay w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Banyu Pharmaceutical

LigandPNGBDBM30158(aminonaphthyridine-based compound, 31)
Affinity DataIC50: 375nMpH: 7.4 T: 2°CAssay Description:Compounds were evaluated for their binding affinity to the membranes of CHO-K1 cells expressing human MCH1R (hMCH1R) in a competition binding assay w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Banyu Pharmaceutical

LigandPNGBDBM30170(2-aminobenzimidazole-based compound, 18)
Affinity DataIC50: 428nMpH: 7.4 T: 2°CAssay Description:Compounds were evaluated for their binding affinity to the membranes of CHO-K1 cells expressing human MCH1R (hMCH1R) in a competition binding assay w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Banyu Pharmaceutical

LigandPNGBDBM30160(aminobenzothiazole-based compound, 39)
Affinity DataIC50: 750nMpH: 7.4 T: 2°CAssay Description:Compounds were evaluated for their binding affinity to the membranes of CHO-K1 cells expressing human MCH1R (hMCH1R) in a competition binding assay w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Banyu Pharmaceutical

LigandPNGBDBM30175(2-aminobenzimidazole-based compound, 23)
Affinity DataIC50: 900nMpH: 7.4 T: 2°CAssay Description:Compounds were evaluated for their binding affinity to the membranes of CHO-K1 cells expressing human MCH1R (hMCH1R) in a competition binding assay w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2009
Entry Details Article
PubMed