Compile Data Set for Download or QSAR
Report error Found 31 Enz. Inhib. hit(s) with all data for entry = 50030422
TargetProstaglandin G/H synthase 2(Sheep)
Karl-Franzens-Universit£T Graz

Curated by ChEMBL
LigandPNGBDBM50295926(Magreth-14a | 5,3'-Diallyl-4'-methoxy-biphenyl-2-o...)
Affinity DataIC50: 60nMAssay Description:Inhibition of COX2 in sheep placental vesicle by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Sheep)
Karl-Franzens-Universit£T Graz

Curated by ChEMBL
LigandPNGBDBM50295926(Magreth-14a | 5,3'-Diallyl-4'-methoxy-biphenyl-2-o...)
Affinity DataIC50: 100nMAssay Description:Inhibition of COX1 in ram seminal vesicle by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Sheep)
Karl-Franzens-Universit£T Graz

Curated by ChEMBL
LigandPNGBDBM50295923(Magreth-3a | Magreth-3b | CHEMBL549698 | 4'-Methox...)
Affinity DataIC50: 200nMAssay Description:Inhibition of COX2 in sheep placental vesicle by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Sheep)
Karl-Franzens-Universit£T Graz

Curated by ChEMBL
LigandPNGBDBM50295925(Magreth-4 | CHEMBL569136 | (E)-3'-Propenyl)-5-(2-p...)
Affinity DataIC50: 600nMAssay Description:Inhibition of COX1 in ram seminal vesicle by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Sheep)
Karl-Franzens-Universit£T Graz

Curated by ChEMBL
LigandPNGBDBM50295923(Magreth-3a | Magreth-3b | CHEMBL549698 | 4'-Methox...)
Affinity DataIC50: 700nMAssay Description:Inhibition of COX1 in ram seminal vesicle by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Sheep)
Karl-Franzens-Universit£T Graz

Curated by ChEMBL
LigandPNGBDBM50157312(CHEMBL330227 | 5,3'-Dipropyl-biphenyl-2,4'-diol | ...)
Affinity DataIC50: 800nMAssay Description:Inhibition of COX1 in ram seminal vesicle by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Sheep)
Karl-Franzens-Universit£T Graz

Curated by ChEMBL
LigandPNGBDBM17638(indometacin | Indocin | 2-{1-[(4-chlorophenyl)carb...)
Affinity DataIC50: 900nMAssay Description:Inhibition of COX1 in ram seminal vesicle by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Sheep)
Karl-Franzens-Universit£T Graz

Curated by ChEMBL
LigandPNGBDBM50295924(4'-Methoxy-3'-(Z)-propenyl)-5-(2-propenyl)-bipheny...)
Affinity DataIC50: 900nMAssay Description:Inhibition of COX2 in sheep placental vesicle by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Human)
Karl-Franzens-Universit£T Graz

Curated by ChEMBL
LigandPNGBDBM50295925(Magreth-4 | CHEMBL569136 | (E)-3'-Propenyl)-5-(2-p...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of 5LOX-mediated LTB4 formation in stimulated human polymorphonuclear leukocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Human)
Karl-Franzens-Universit£T Graz

Curated by ChEMBL
LigandPNGBDBM50295924(4'-Methoxy-3'-(Z)-propenyl)-5-(2-propenyl)-bipheny...)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of 5LOX-mediated LTB4 formation in stimulated human polymorphonuclear leukocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Human)
Karl-Franzens-Universit£T Graz

Curated by ChEMBL
LigandPNGBDBM50295920(CHEMBL555297 | Magreth-1 | 4'-Methoxy-5,3'-dipropy...)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of 5LOX-mediated LTB4 formation in stimulated human polymorphonuclear leukocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Human)
Karl-Franzens-Universit£T Graz

Curated by ChEMBL
LigandPNGBDBM50295926(Magreth-14a | 5,3'-Diallyl-4'-methoxy-biphenyl-2-o...)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of 5LOX-mediated LTB4 formation in stimulated human polymorphonuclear leukocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Human)
Karl-Franzens-Universit£T Graz

Curated by ChEMBL
LigandPNGBDBM50157312(CHEMBL330227 | 5,3'-Dipropyl-biphenyl-2,4'-diol | ...)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of 5LOX-mediated LTB4 formation in stimulated human polymorphonuclear leukocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Sheep)
Karl-Franzens-Universit£T Graz

Curated by ChEMBL
LigandPNGBDBM50157304(3',5-diallylbiphenyl-2,4'-diol | CHEMBL16901 | cid...)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of COX1 in ram seminal vesicle by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Sheep)
Karl-Franzens-Universit£T Graz

Curated by ChEMBL
LigandPNGBDBM50157312(CHEMBL330227 | 5,3'-Dipropyl-biphenyl-2,4'-diol | ...)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of COX2 in sheep placental vesicle by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Sheep)
Karl-Franzens-Universit£T Graz

Curated by ChEMBL
LigandPNGBDBM50157304(3',5-diallylbiphenyl-2,4'-diol | CHEMBL16901 | cid...)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of COX2 in sheep placental vesicle by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Human)
Karl-Franzens-Universit£T Graz

Curated by ChEMBL
LigandPNGBDBM50295923(Magreth-3a | Magreth-3b | CHEMBL549698 | 4'-Methox...)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of 5LOX-mediated LTB4 formation in stimulated human polymorphonuclear leukocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Human)
Karl-Franzens-Universit£T Graz

Curated by ChEMBL
LigandPNGBDBM50295921(2-Acetoxy-4'-methoxy-5,3'-di-(2-propenyl)-biphenyl...)
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of 5LOX-mediated LTB4 formation in stimulated human polymorphonuclear leukocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Sheep)
Karl-Franzens-Universit£T Graz

Curated by ChEMBL
LigandPNGBDBM50029593(CHEMBL7162 | NS398 | NS-398 | N-(2-Cyclohexyloxy-4...)
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of COX2 in sheep placental vesicle by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetProstaglandin G/H synthase 2(Sheep)
Karl-Franzens-Universit£T Graz

Curated by ChEMBL
LigandPNGBDBM50295925(Magreth-4 | CHEMBL569136 | (E)-3'-Propenyl)-5-(2-p...)
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of COX2 in sheep placental vesicle by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Sheep)
Karl-Franzens-Universit£T Graz

Curated by ChEMBL
LigandPNGBDBM50295924(4'-Methoxy-3'-(Z)-propenyl)-5-(2-propenyl)-bipheny...)
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of COX1 in ram seminal vesicle by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Human)
Karl-Franzens-Universit£T Graz

Curated by ChEMBL
LigandPNGBDBM50157304(3',5-diallylbiphenyl-2,4'-diol | CHEMBL16901 | cid...)
Affinity DataIC50: 4.20E+3nMAssay Description:Inhibition of 5LOX-mediated LTB4 formation in stimulated human polymorphonuclear leukocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Human)
Karl-Franzens-Universit£T Graz

Curated by ChEMBL
LigandPNGBDBM50295922(2,4'-Diacetoxy-5,3'-di-(2-propenyl)-biphenyl | CHE...)
Affinity DataIC50: 4.50E+3nMAssay Description:Inhibition of 5LOX-mediated LTB4 formation in stimulated human polymorphonuclear leukocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Sheep)
Karl-Franzens-Universit£T Graz

Curated by ChEMBL
LigandPNGBDBM50295921(2-Acetoxy-4'-methoxy-5,3'-di-(2-propenyl)-biphenyl...)
Affinity DataIC50: 4.90E+3nMAssay Description:Inhibition of COX2 in sheep placental vesicle by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Human)
Karl-Franzens-Universit£T Graz

Curated by ChEMBL
LigandPNGBDBM50000541(Leutrol | CHEMBL93 | N-(1-Benzo(b)thien-2-ylethyl)...)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of 5LOX-mediated LTB4 formation in stimulated human polymorphonuclear leukocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Sheep)
Karl-Franzens-Universit£T Graz

Curated by ChEMBL
LigandPNGBDBM50295928(2,4'-Dimethoxy-5,3'-dipropyl-biphenyl | CHEMBL5602...)
Affinity DataIC50: 6.90E+3nMAssay Description:Inhibition of COX2 in sheep placental vesicle by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Sheep)
Karl-Franzens-Universit£T Graz

Curated by ChEMBL
LigandPNGBDBM50295927(5,3'-Diallyl-2,4'-dimethoxy-biphenyl | 2,4'-Dimeth...)
Affinity DataIC50: 7.70E+3nMAssay Description:Inhibition of COX2 in sheep placental vesicle by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Sheep)
Karl-Franzens-Universit£T Graz

Curated by ChEMBL
LigandPNGBDBM50295920(CHEMBL555297 | Magreth-1 | 4'-Methoxy-5,3'-dipropy...)
Affinity DataIC50: 7.70E+3nMAssay Description:Inhibition of COX1 in ram seminal vesicle by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Sheep)
Karl-Franzens-Universit£T Graz

Curated by ChEMBL
LigandPNGBDBM50295927(5,3'-Diallyl-2,4'-dimethoxy-biphenyl | 2,4'-Dimeth...)
Affinity DataIC50: 1.14E+4nMAssay Description:Inhibition of COX1 in ram seminal vesicle by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Human)
Karl-Franzens-Universit£T Graz

Curated by ChEMBL
LigandPNGBDBM50295927(5,3'-Diallyl-2,4'-dimethoxy-biphenyl | 2,4'-Dimeth...)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of 5LOX-mediated LTB4 formation in stimulated human polymorphonuclear leukocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Sheep)
Karl-Franzens-Universit£T Graz

Curated by ChEMBL
LigandPNGBDBM50295928(2,4'-Dimethoxy-5,3'-dipropyl-biphenyl | CHEMBL5602...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of COX1 in ram seminal vesicle by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed