Compile Data Set for Download or QSAR
Report error Found 24 Enz. Inhib. hit(s) with all data for entry = 50030463
TargetFatty-acid amide hydrolase 1(Human)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM26740(N-phenyl-4-(quinolin-3-ylmethyl)piperidine-1-carbo...)
Affinity DataIC50: 16.2nMAssay Description:Inhibition of FAAHMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rat)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM26739(URB 597 | URB597 | CHEMBL184238 | 3-(3-carbamoylph...)
Affinity DataIC50: 22nMAssay Description:Inhibition of rat FAAH incubated 3 hrs prior to addition of arachidonyl-amino-methyl-coumarin amideMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1(Human)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM26741(N-phenyl-4-(quinolin-2-ylmethyl)piperazine-1-carbo...)
Affinity DataIC50: 33nMAssay Description:Inhibition of FAAHMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1(Human)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50244718(cid_2809273 | CHEMBL460273 | JNJ-1661010 | N-pheny...)
Affinity DataIC50: 33nMAssay Description:Inhibition of FAAHMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rat)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM26739(URB 597 | URB597 | CHEMBL184238 | 3-(3-carbamoylph...)
Affinity DataIC50: 63nMAssay Description:Inhibition of rat FAAH incubated 1 hr prior to addition of arachidonyl-amino-methyl-coumarin amideMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1(Human)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50296484(VER-156084 | (S)-{3-[(4-Chlorophenyl)-(2-chloropyr...)
Affinity DataIC50: 78nMAssay Description:Inhibition of human FAAH incubated 3 hrs prior to addition of arachidonyl-amino-methyl-coumarin amideMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1(Human)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM26739(URB 597 | URB597 | CHEMBL184238 | 3-(3-carbamoylph...)
Affinity DataIC50: 78nMAssay Description:Inhibition of human FAAH incubated 1 hr prior to addition of arachidonyl-amino-methyl-coumarin amideMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1(Human)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM26739(URB 597 | URB597 | CHEMBL184238 | 3-(3-carbamoylph...)
Affinity DataIC50: 109nMAssay Description:Inhibition of FAAHMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rat)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM23120(CHEMBL177577 | 7-phenyl-1-[5-(pyridin-2-yl)-1,3-ox...)
Affinity DataIC50: 112nMAssay Description:Inhibition of rat FAAH incubated 1 hr prior to addition of arachidonyl-amino-methyl-coumarin amideMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1(Human)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM23120(CHEMBL177577 | 7-phenyl-1-[5-(pyridin-2-yl)-1,3-ox...)
Affinity DataIC50: 119nMAssay Description:Inhibition of human FAAH incubated 1 hr prior to addition of arachidonyl-amino-methyl-coumarin amideMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1(Human)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50296484(VER-156084 | (S)-{3-[(4-Chlorophenyl)-(2-chloropyr...)
Affinity DataIC50: 140nMAssay Description:Inhibition of human FAAH incubated 1 hr prior to addition of arachidonyl-amino-methyl-coumarin amideMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1(Human)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50296484(VER-156084 | (S)-{3-[(4-Chlorophenyl)-(2-chloropyr...)
Affinity DataIC50: 188nMAssay Description:Inhibition of human FAAH incubated 3 hrs prior to addition of arachidonyl-amino-methyl-coumarin amideMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1(Human)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM23120(CHEMBL177577 | 7-phenyl-1-[5-(pyridin-2-yl)-1,3-ox...)
Affinity DataIC50: 230nMAssay Description:Inhibition of FAAHMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1(Human)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50296484(VER-156084 | (S)-{3-[(4-Chlorophenyl)-(2-chloropyr...)
Affinity DataIC50: 291nMAssay Description:Inhibition of human FAAH incubated 1 hr prior to addition of arachidonyl-amino-methyl-coumarin amideMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rat)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM23120(CHEMBL177577 | 7-phenyl-1-[5-(pyridin-2-yl)-1,3-ox...)
Affinity DataIC50: 306nMAssay Description:Inhibition of rat FAAH incubated 3 hrs prior to addition of arachidonyl-amino-methyl-coumarin amideMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rat)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50296484(VER-156084 | (S)-{3-[(4-Chlorophenyl)-(2-chloropyr...)
Affinity DataIC50: 531nMAssay Description:Inhibition of rat FAAH incubated 3 hrs prior to addition of arachidonyl-amino-methyl-coumarin amideMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50296484(VER-156084 | (S)-{3-[(4-Chlorophenyl)-(2-chloropyr...)
Affinity DataKi:  560nMAssay Description:Displacement of [3H]SR141716A from human CB1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rat)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50296484(VER-156084 | (S)-{3-[(4-Chlorophenyl)-(2-chloropyr...)
Affinity DataIC50: 1.03E+3nMAssay Description:Inhibition of rat FAAH incubated 1 hr prior to addition of arachidonyl-amino-methyl-coumarin amideMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50296484(VER-156084 | (S)-{3-[(4-Chlorophenyl)-(2-chloropyr...)
Affinity DataKi:  7.19E+3nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rat)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50296485((R)-{3-[(4-Chlorophenyl)-(2-chloropyridin-3-yl)met...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of rat FAAH incubated 1 hr prior to addition of arachidonyl-amino-methyl-coumarin amideMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rat)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50296485((R)-{3-[(4-Chlorophenyl)-(2-chloropyridin-3-yl)met...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of rat FAAH incubated 3 hrs prior to addition of arachidonyl-amino-methyl-coumarin amideMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1(Human)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50296485((R)-{3-[(4-Chlorophenyl)-(2-chloropyridin-3-yl)met...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human FAAH incubated 1 hr prior to addition of arachidonyl-amino-methyl-coumarin amideMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1(Human)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50296485((R)-{3-[(4-Chlorophenyl)-(2-chloropyridin-3-yl)met...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human FAAH incubated 3 hrs prior to addition of arachidonyl-amino-methyl-coumarin amideMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50296485((R)-{3-[(4-Chlorophenyl)-(2-chloropyridin-3-yl)met...)
Affinity DataKi:  1.09E+4nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed