Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50028844
TargetTestis-specific serine/threonine-protein kinase 1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50279383(sodium 2,2'-(biphenyl-4,4'-diyl)bis(1-hydroxy-2-ox...)
Affinity DataIC50: 1.44E+4nMAssay Description:Inhibition of TSSK1-catalyzed phosphorylation of AALVRQMSVAFFFK substrate by LC-MS based HTP assay in absence of Pep8-(O2)More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTestis-specific serine/threonine-protein kinase 1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50279383(sodium 2,2'-(biphenyl-4,4'-diyl)bis(1-hydroxy-2-ox...)
Affinity DataIC50: 1.91E+4nMAssay Description:Inhibition of TSSK1-catalyzed phosphorylation of AALVRQMSVAFFFK substrate by LC-MS based HTP assay in presence of Pep8-(O2)More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTestis-specific serine/threonine-protein kinase 1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50279383(sodium 2,2'-(biphenyl-4,4'-diyl)bis(1-hydroxy-2-ox...)
Affinity DataIC50: 2.48E+4nMAssay Description:Inhibition of TSSK1-catalyzed phosphorylation of AALVRQMSVAFFFK substrate by luminescent kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTestis-specific serine/threonine-protein kinase 1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50278920(4-(7-isopropyl-6-oxo-1-(3-phenylpropyl)-5,6-dihydr...)
Affinity DataIC50: 3.80E+4nMAssay Description:Inhibition of TSSK1-catalyzed phosphorylation of AALVRQMSVAFFFK substrate by LC-MS based HTP assay in presence of Pep8-(O2)More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTestis-specific serine/threonine-protein kinase 1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50279386(5-hydroxy-8-methyl-4-propyl-7,8-dihydropyrano[3,2-...)
Affinity DataIC50: 3.87E+4nMAssay Description:Inhibition of TSSK1-catalyzed phosphorylation of AALVRQMSVAFFFK substrate by luminescent kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTestis-specific serine/threonine-protein kinase 1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50279385(1,1'-(biphenyl-4,4'-diyl)bis(2,2-dihydroxyethanone...)
Affinity DataIC50: 4.32E+4nMAssay Description:Inhibition of TSSK1-catalyzed phosphorylation of AALVRQMSVAFFFK substrate by luminescent kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTestis-specific serine/threonine-protein kinase 1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50278919(2-(3,4-dihydroxyphenyl)-1-heptyl-7-isopropyl-1H-im...)
Affinity DataIC50: 7.20E+4nMAssay Description:Inhibition of TSSK1-catalyzed phosphorylation of AALVRQMSVAFFFK substrate by LC-MS based HTP assay in presence of Pep8-(O2)More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTestis-specific serine/threonine-protein kinase 1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50279384(N-(4-(7-methyl-6-oxo-1-(3-phenylpropyl)-5,6-dihydr...)
Affinity DataIC50: 9.80E+4nMAssay Description:Inhibition of TSSK1-catalyzed phosphorylation of AALVRQMSVAFFFK substrate by LC-MS based HTP assay in presence of Pep8-(O2)More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed