Compile Data Set for Download or QSAR
Report error Found 72 Enz. Inhib. hit(s) with all data for entry = 50030483
TargetNeuropeptide Y receptor type 1(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50296870((1-((1R,4R)-4-((R)-1-(4-methoxyphenyl)ethylamino)-...)
Affinity DataKi:  7.30nMAssay Description:Displacement of [125I]PYY from human recombinant neuropeptide Y1 receptor expressed in CHO (NFAT-bla) cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50296879((4,4-diphenylpiperidin-1-yl)((1R,4R)-4-((R)-1-(4-m...)
Affinity DataKi:  7.40nMAssay Description:Displacement of [125I]PYY from human recombinant neuropeptide Y1 receptor expressed in CHO (NFAT-bla) cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50296876((4-(6-chloropyridin-3-yl)-4-phenylpiperidin-1-yl)(...)
Affinity DataIC50: 8nMAssay Description:Displacement of [3H]imipramine from human serotonin transporter expressed in CHO cell membrane by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50296884((1-((1R,4R)-2,2-dimethyl-4-((R)-1-p-tolylethylamin...)
Affinity DataKi:  10nMAssay Description:Displacement of [125I]PYY from human recombinant neuropeptide Y1 receptor expressed in CHO (NFAT-bla) cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50296873(1'-((1R,4R)-4-((R)-1-(4-methoxyphenyl)ethylamino)-...)
Affinity DataIC50: 11nMAssay Description:Displacement of [3H]imipramine from human serotonin transporter expressed in CHO cell membrane by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50296874(N-(4-((1R,4R)-4-((R)-1-(4-methoxyphenyl)ethylamino...)
Affinity DataIC50: 14nMAssay Description:Displacement of [3H]imipramine from human serotonin transporter expressed in CHO cell membrane by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50296877(((1R,4R)-4-((R)-1-(4-methoxyphenyl)ethylamino)-2,2...)
Affinity DataIC50: 14nMAssay Description:Displacement of [3H]imipramine from human serotonin transporter expressed in CHO cell membrane by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50296879((4,4-diphenylpiperidin-1-yl)((1R,4R)-4-((R)-1-(4-m...)
Affinity DataIC50: 15nMAssay Description:Displacement of [3H]imipramine from human serotonin transporter expressed in CHO cell membrane by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50296885(1-((1R,4R)-4-((R)-1-(4-methoxyphenyl)ethylamino)-2...)
Affinity DataKi:  15nMAssay Description:Displacement of [125I]PYY from human recombinant neuropeptide Y1 receptor expressed in CHO (NFAT-bla) cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50296872(3-(1-((1R,4R)-4-((R)-1-(4-methoxyphenyl)ethylamino...)
Affinity DataIC50: 17nMAssay Description:Displacement of [3H]imipramine from human serotonin transporter expressed in CHO cell membrane by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50296870((1-((1R,4R)-4-((R)-1-(4-methoxyphenyl)ethylamino)-...)
Affinity DataIC50: 17nMAssay Description:Displacement of [3H]imipramine from human serotonin transporter expressed in CHO cell membrane by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50296878(((1R,4R)-4-((R)-1-(4-methoxyphenyl)ethylamino)-2,2...)
Affinity DataIC50: 17nMAssay Description:Displacement of [3H]imipramine from human serotonin transporter expressed in CHO cell membrane by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50296873(1'-((1R,4R)-4-((R)-1-(4-methoxyphenyl)ethylamino)-...)
Affinity DataKi:  18nMAssay Description:Displacement of [125I]PYY from human recombinant neuropeptide Y1 receptor expressed in CHO (NFAT-bla) cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50296881((1-((1R,4R)-4-((S)-2,2-difluoro-1-(4-methoxyphenyl...)
Affinity DataKi:  22nMAssay Description:Displacement of [125I]PYY from human recombinant neuropeptide Y1 receptor expressed in CHO (NFAT-bla) cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50296871(1-(1-((1R,4R)-4-((R)-1-(4-methoxyphenyl)ethylamino...)
Affinity DataIC50: 24nMAssay Description:Displacement of [3H]imipramine from human serotonin transporter expressed in CHO cell membrane by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50296877(((1R,4R)-4-((R)-1-(4-methoxyphenyl)ethylamino)-2,2...)
Affinity DataKi:  24nMAssay Description:Displacement of [125I]PYY from human recombinant neuropeptide Y1 receptor expressed in CHO (NFAT-bla) cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50296875(N-(4-((1R,4R)-4-((R)-1-(4-methoxyphenyl)ethylamino...)
Affinity DataIC50: 26nMAssay Description:Displacement of [3H]imipramine from human serotonin transporter expressed in CHO cell membrane by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50296883((1-((1R,4R)-4-((R)-1-(4-chlorophenyl)ethylamino)-2...)
Affinity DataKi:  27nMAssay Description:Displacement of [125I]PYY from human recombinant neuropeptide Y1 receptor expressed in CHO (NFAT-bla) cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50296878(((1R,4R)-4-((R)-1-(4-methoxyphenyl)ethylamino)-2,2...)
Affinity DataKi:  29nMAssay Description:Displacement of [125I]PYY from human recombinant neuropeptide Y1 receptor expressed in CHO (NFAT-bla) cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50296876((4-(6-chloropyridin-3-yl)-4-phenylpiperidin-1-yl)(...)
Affinity DataKi:  32nMAssay Description:Displacement of [125I]PYY from human recombinant neuropeptide Y1 receptor expressed in CHO (NFAT-bla) cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50296885(1-((1R,4R)-4-((R)-1-(4-methoxyphenyl)ethylamino)-2...)
Affinity DataIC50: 38nMAssay Description:Displacement of [3H]imipramine from human serotonin transporter expressed in CHO cell membrane by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50296872(3-(1-((1R,4R)-4-((R)-1-(4-methoxyphenyl)ethylamino...)
Affinity DataKi:  42nMAssay Description:Displacement of [125I]PYY from human recombinant neuropeptide Y1 receptor expressed in CHO (NFAT-bla) cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50296880((1-((1R,4R)-2,2-dimethyl-4-((S)-2,2,2-trifluoro-1-...)
Affinity DataKi:  43nMAssay Description:Displacement of [125I]PYY from human recombinant neuropeptide Y1 receptor expressed in CHO (NFAT-bla) cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50296882((1-((1R,4R)-4-((R)-1-(4-fluorophenyl)ethylamino)-2...)
Affinity DataKi:  44nMAssay Description:Displacement of [125I]PYY from human recombinant neuropeptide Y1 receptor expressed in CHO (NFAT-bla) cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50296871(1-(1-((1R,4R)-4-((R)-1-(4-methoxyphenyl)ethylamino...)
Affinity DataKi:  45nMAssay Description:Displacement of [125I]PYY from human recombinant neuropeptide Y1 receptor expressed in CHO (NFAT-bla) cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50296875(N-(4-((1R,4R)-4-((R)-1-(4-methoxyphenyl)ethylamino...)
Affinity DataKi:  48nMAssay Description:Displacement of [125I]PYY from human recombinant neuropeptide Y1 receptor expressed in CHO (NFAT-bla) cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50296874(N-(4-((1R,4R)-4-((R)-1-(4-methoxyphenyl)ethylamino...)
Affinity DataKi:  49nMAssay Description:Displacement of [125I]PYY from human recombinant neuropeptide Y1 receptor expressed in CHO (NFAT-bla) cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50296883((1-((1R,4R)-4-((R)-1-(4-chlorophenyl)ethylamino)-2...)
Affinity DataIC50: 59nMAssay Description:Displacement of [3H]imipramine from human serotonin transporter expressed in CHO cell membrane by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50296884((1-((1R,4R)-2,2-dimethyl-4-((R)-1-p-tolylethylamin...)
Affinity DataIC50: 76nMAssay Description:Displacement of [3H]imipramine from human serotonin transporter expressed in CHO cell membrane by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50296894(((1R,4R)-4-((R)-1-(4-methoxyphenyl)ethylamino)-2,2...)
Affinity DataKi:  120nMAssay Description:Displacement of [125I]PYY from human recombinant neuropeptide Y1 receptor expressed in CHO (NFAT-bla) cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50296882((1-((1R,4R)-4-((R)-1-(4-fluorophenyl)ethylamino)-2...)
Affinity DataIC50: 130nMAssay Description:Displacement of [3H]imipramine from human serotonin transporter expressed in CHO cell membrane by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50296891((1-((1R,4R)-4-((R)-1-(4-methoxyphenyl)ethylamino)-...)
Affinity DataKi:  150nMAssay Description:Displacement of [125I]PYY from human recombinant neuropeptide Y1 receptor expressed in CHO (NFAT-bla) cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50296888((1-((1R,4R)-2,2-dimethyl-4-((R)-1-phenylethylamino...)
Affinity DataKi:  160nMAssay Description:Displacement of [125I]PYY from human recombinant neuropeptide Y1 receptor expressed in CHO (NFAT-bla) cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50296886((1-((1R,4R)-4-((R)-1-(3-methoxyphenyl)ethylamino)-...)
Affinity DataKi:  210nMAssay Description:Displacement of [125I]PYY from human recombinant neuropeptide Y1 receptor expressed in CHO (NFAT-bla) cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50296881((1-((1R,4R)-4-((S)-2,2-difluoro-1-(4-methoxyphenyl...)
Affinity DataIC50: 280nMAssay Description:Antagonist activity at human neuropeptide Y1 receptor expressed in HEK293 cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50296893(((1R,4R)-4-((R)-1-(4-methoxyphenyl)ethylamino)-2,2...)
Affinity DataKi:  330nMAssay Description:Displacement of [125I]PYY from human recombinant neuropeptide Y1 receptor expressed in CHO (NFAT-bla) cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50296889((1-((1R,4R)-4-(4-methoxybenzylamino)-2,2-dimethylc...)
Affinity DataKi:  470nMAssay Description:Displacement of [125I]PYY from human recombinant neuropeptide Y1 receptor expressed in CHO (NFAT-bla) cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50296877(((1R,4R)-4-((R)-1-(4-methoxyphenyl)ethylamino)-2,2...)
Affinity DataIC50: 520nMAssay Description:Displacement of [35S]MK499 from human ERG potassium channel expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50296879((4,4-diphenylpiperidin-1-yl)((1R,4R)-4-((R)-1-(4-m...)
Affinity DataIC50: 530nMAssay Description:Displacement of [35S]MK499 from human ERG potassium channel expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50296887((1-((1R,4R)-4-((R)-1-(2-methoxyphenyl)ethylamino)-...)
Affinity DataKi:  790nMAssay Description:Displacement of [125I]PYY from human recombinant neuropeptide Y1 receptor expressed in CHO (NFAT-bla) cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50296895((4-(1,3,4-oxadiazol-2-yl)-4-phenylpiperidin-1-yl)(...)
Affinity DataKi:  890nMAssay Description:Displacement of [125I]PYY from human recombinant neuropeptide Y1 receptor expressed in CHO (NFAT-bla) cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50296889((1-((1R,4R)-4-(4-methoxybenzylamino)-2,2-dimethylc...)
Affinity DataIC50: 900nMAssay Description:Displacement of [35S]MK499 from human ERG potassium channel expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50296890((1-((1R,4R)-4-((S)-1-(4-methoxyphenyl)ethylamino)-...)
Affinity DataKi:  1.10E+3nMAssay Description:Displacement of [125I]PYY from human recombinant neuropeptide Y1 receptor expressed in CHO (NFAT-bla) cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50296883((1-((1R,4R)-4-((R)-1-(4-chlorophenyl)ethylamino)-2...)
Affinity DataIC50: 1.30E+3nMAssay Description:Displacement of [35S]MK499 from human ERG potassium channel expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 2(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50296881((1-((1R,4R)-4-((S)-2,2-difluoro-1-(4-methoxyphenyl...)
Affinity DataIC50: 1.40E+3nMAssay Description:Antagonist activity at human neuropeptide Y2 receptor expressed in HEK293 cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50296876((4-(6-chloropyridin-3-yl)-4-phenylpiperidin-1-yl)(...)
Affinity DataIC50: 2.10E+3nMAssay Description:Displacement of [35S]MK499 from human ERG potassium channel expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50296892(((1R,4R)-4-((R)-1-(4-methoxyphenyl)ethylamino)-2,2...)
Affinity DataKi:  3.00E+3nMAssay Description:Displacement of [125I]PYY from human recombinant neuropeptide Y1 receptor expressed in CHO (NFAT-bla) cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50296890((1-((1R,4R)-4-((S)-1-(4-methoxyphenyl)ethylamino)-...)
Affinity DataIC50: 4.70E+3nMAssay Description:Displacement of [35S]MK499 from human ERG potassium channel expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50296881((1-((1R,4R)-4-((S)-2,2-difluoro-1-(4-methoxyphenyl...)
Affinity DataIC50: 4.80E+3nMAssay Description:Displacement of [3H]imipramine from human serotonin transporter expressed in CHO cell membrane by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50296892(((1R,4R)-4-((R)-1-(4-methoxyphenyl)ethylamino)-2,2...)
Affinity DataIC50: 6.70E+3nMAssay Description:Displacement of [35S]MK499 from human ERG potassium channel expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
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