Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50030488
Target3-phosphoinositide-dependent protein kinase 1(Human)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50296949(PS48 | (2Z)-5-(4-chlorophenyl)-3-phenylpent-2-enoi...)
Affinity DataKd:  1.03E+4nMAssay Description:Binding affinity to PDK1 (50 to 359) by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMedPDB3D3D Structure (crystal)
Target3-phosphoinositide-dependent protein kinase 1(Human)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50296950((Z)-5-(4-Bromophenyl)-3-phenylpent-2-enoic acid | ...)
Affinity DataKd:  2.09E+4nMAssay Description:Binding affinity to PDK1 (50 to 359) by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
Target3-phosphoinositide-dependent protein kinase 1(Human)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50296951((Z)-3-Phenyl-5-(4-(trifluoromethyl)phenyl)pent-2-e...)
Affinity DataKd:  1.04E+4nMAssay Description:Binding affinity to PDK1 (50 to 359) by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
Target3-phosphoinositide-dependent protein kinase 1(Human)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50296952((Z)-5-(3,4-Dichlorophenyl)-3-phenylpent-2-enoic Ac...)
Affinity DataKd:  1.39E+4nMAssay Description:Binding affinity to PDK1 (50 to 359) by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
Target3-phosphoinositide-dependent protein kinase 1(Human)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50296953((Z)-5-(2,4-Dichlorophenyl)-3-phenylpent-2-enoic Ac...)
Affinity DataKd:  5.90E+3nMAssay Description:Binding affinity to PDK1 (50 to 359) by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
Target3-phosphoinositide-dependent protein kinase 1(Human)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50296954((Z)-5-(4-bromo-2-fluorophenyl)-3-phenylpent-2-enoi...)
Affinity DataKd:  6.20E+3nMAssay Description:Binding affinity to PDK1 (50 to 359) by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
Target3-phosphoinositide-dependent protein kinase 1(Human)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50296955((Z)-5-(Naphthalen-2-yl)-3-phenylpent-2-enoic Acid ...)
Affinity DataKd:  1.38E+4nMAssay Description:Binding affinity to PDK1 (50 to 359) by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
Target3-phosphoinositide-dependent protein kinase 1(Human)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50296956((Z)-5-(1H-Indol-3-yl)-3-phenylpent-2-enoic Acid | ...)
Affinity DataKd:  1.00E+4nMAssay Description:Binding affinity to PDK1 (50 to 359) by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed